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La ricerca find articoli where soggetti phrase all words 'human leukocyte elastase' sort by level,fasc_key/DESCEND, pagina_ini_num/ASCEND ha restituito 345 riferimenti
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    1. Rodis, NP; Digenis, GA
      Synthesis and in-vitro evaluation of novel low molecular weight thiocarbamates as inhibitors of human leukocyte elastase

      JOURNAL OF ENZYME INHIBITION
    2. Vicentini, CB; Guarneri, M; Andrisano, V; Guccione, S; Langer, T; Marschhofer, R; Chabin, R; Edison, AM; Huang, X; Knight, WB; Giori, P
      Potential of pyrazolooxadiazinone derivatives as serine protease inhibitors

      JOURNAL OF ENZYME INHIBITION
    3. Hinchliffe, PS; Wood, JM; Davis, AM; Austin, RP; Beckett, RP; Page, MI
      Unusual steric effects in sulfonyl transfer reactions

      JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 2
    4. De Angelis, F; Attorrese, G; Cavicchio, G; Ciampa, S; Di Tullio, A; Fattori, D; Nicoletti, R; Domenici, E
      Synthesis and preliminary biological evaluation of 3 '-substituted cephem sulfones as potential beta-lactamase inhibitors

      EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
    5. Walker, B; Lynas, JF
      Strategies for the inhibition of serine proteases

      CELLULAR AND MOLECULAR LIFE SCIENCES
    6. Naumov, P; Jovanovski, G
      An update to the combined vibrational-diffraction experimental and theoretical studies of small biologically important cyclic imides: Reference to saccharin

      CURRENT ORGANIC CHEMISTRY
    7. Okada, Y
      Synthesis of peptides by solution methods

      CURRENT ORGANIC CHEMISTRY
    8. Beardsell, M; Hinchliffe, PS; Wood, JM; Wilmouth, RC; Schofield, CJ; Page, MI
      beta-Sultams - A novel class of serine protease inhibitors

      CHEMICAL COMMUNICATIONS
    9. Gorrini, M; Lupi, A; Viglio, S; Pamparana, F; Cetta, G; Iadarola, P; Powers, JC; Luisetti, M
      Inhibition of human neutrophil elastase by erythromycin and flurythromycin, two macrolide antibiotics

      AMERICAN JOURNAL OF RESPIRATORY CELL AND MOLECULAR BIOLOGY
    10. Ying, QL; Simon, SR
      Kinetics of the inhibition of proteinase 3 by elafin

      AMERICAN JOURNAL OF RESPIRATORY CELL AND MOLECULAR BIOLOGY
    11. Groutas, WC; He, S; Kuang, RZ; Ruan, S; Tu, J; Chan, HK
      Inhibition of serine proteases by functionalized sulfonamides coupled to the 1,2,5-thiadiazolidin-3-one 1,1 dioxide scaffold

      BIOORGANIC & MEDICINAL CHEMISTRY
    12. Ohmoto, K; Okuma, M; Yamamoto, T; Kijima, H; Sekioka, T; Kitagawa, K; Yamamoto, S; Tanaka, K; Kawabata, K; Sakata, A; Imawaka, H; Nakai, H; Toda, M
      Design and synthesis of new orally active inhibitors of human neutrophil elastase

      BIOORGANIC & MEDICINAL CHEMISTRY
    13. Neumann, U; Schechter, NM; Gutschow, M
      Inhibition of human chymase by 2-amino-3,1-benzoxazin-4-ones

      BIOORGANIC & MEDICINAL CHEMISTRY
    14. Odagaki, Y; Ohmoto, K; Matsuoka, S; Hamanaka, N; Nakai, H; Toda, M; Katsuya, Y
      The crystal structure of the complex of non-peptidic inhibitor of human neutrophil elastase ONO-6818 and porcine pancreatic elastase

      BIOORGANIC & MEDICINAL CHEMISTRY
    15. Akahoshi, F; Ashimori, A; Yoshimura, T; Imada, T; Nakajima, M; Mitsutomi, N; Kuwahara, S; Ohtsuka, T; Fukaya, C; Miyazaki, M; Nakamura, N
      Non-peptidic inhibitors of human chymase. Synthesis, structure-activity relationships, and pharmacokinetic profiles of a series of 5-amino-6-oxo-1,6-dihydropyrimidine-containing trifluoromethyl ketones

      BIOORGANIC & MEDICINAL CHEMISTRY
    16. Aoyama, Y; Uenaka, M; Kii, M; Tanaka, M; Konoike, T; Hayasaki-Kajiwara, Y; Naya, N; Nakajima, M
      Design, synthesis and pharmacological evaluation of 3-benzylazetidine-2-one-based human chymase inhibitors

      BIOORGANIC & MEDICINAL CHEMISTRY
    17. Mcdonold, SJF; Dowle, MD; Harrison, LA; Shah, P; Johnson, MR; Inglis, GGA; Clarke, GDE; Smith, RA; Humphreys, D; Molloy, CR; Amour, A; Dixon, M; Murkitt, G; Godward, RE; Padfield, T; Skarzynski, T; Singh, OMP; Kumar, KA; Fleetwood, G; Hodgson, ST; Hardy, GW; Fincha, H
      The discovery of a potent, intracellular, orally bioavailable, long duration inhibitor of human neutrophil Elastase - GW311616A a development candidate

      BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
    18. Macdonald, SJF; Dowle, MD; Harrison, LA; Spooner, JE; Shah, P; Johnson, MR; Inglis, GGA; Clarke, GDE; Belton, DJ; Smith, RA; Molloy, CR; Dixon, M; Murkitt, G; Godward, RE; Skarzynski, T; Singh, OMP; Kumar, KA; Hodgson, ST; McDonald, E; Hardy, GW; Finch, H
      Intracellular inhibition of human neutrophil elastase by orally active pyrrolidine-trans-lactams

      BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
    19. Chen, ZL; Demuth, TP; Wireko, FC
      Stereoselective synthesis and antibacterial evaluation of 4-amido-isothiazolidinone oxides

      BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
    20. Ohmoto, K; Yamamoto, T; Horiuchi, T; Kojima, T; Hachiya, K; Hashimoto, S; Kawamura, M; Nakai, H; Toda, M
      Improved synthesis of a new nonpeptidic inhibitor of human neutrophil elastase

      SYNLETT
    21. Ginzberg, HH; Cherapanov, V; Dong, Q; Cantin, A; McCulloch, CAG; Shannon, PT; Downey, GP
      Neutrophil-mediated epithelial injury during transmigration: role of elastase

      AMERICAN JOURNAL OF PHYSIOLOGY-GASTROINTESTINAL AND LIVER PHYSIOLOGY
    22. Kawase, M
      Synthetic and medicinal chemistry of trifluoromethyl ketones

      JOURNAL OF SYNTHETIC ORGANIC CHEMISTRY JAPAN
    23. Ghani, U; Ng, KKS; Atta-ur-Rahman; Choudhary, MI; Ullah, N; James, MNG
      Crystal structure of gamma-chymotrypsin in complex with 7-hydroxycoumarin

      JOURNAL OF MOLECULAR BIOLOGY
    24. Ohmoto, K; Yamamoto, T; Okuma, M; Horiuchi, T; Imanishi, H; Odagaki, Y; Kawabata, K; Sekioka, T; Hirota, Y; Matsuoka, S; Nakai, H; Toda, M; Cheronis, JC; Spruce, LW; Gyorkos, A; Wieczorek, M
      Development of orally active nonpeptidic inhibitors of human neutrophil elastase

      JOURNAL OF MEDICINAL CHEMISTRY
    25. Akahoshi, F; Ashimori, A; Sakashita, H; Yoshimura, T; Imada, T; Nakajima, M; Mitsutomi, N; Kuwahara, S; Ohtsuka, T; Fukaya, C; Miyazaki, M; Nakamura, N
      Synthesis, structure-activity relationships, and pharmacokinetic profiles of nonpeptidic alpha-keto heterocycles as novel inhibitors of human chymase

      JOURNAL OF MEDICINAL CHEMISTRY
    26. Akahoshi, F; Ashimori, A; Sakashita, H; Yoshimura, T; Eda, M; Imada, T; Nakajima, M; Mitsutomi, N; Kuwahara, S; Ohtsuka, T; Fukaya, C; Miyazaki, M; Nakamura, N
      Synthesis, structure-activity relationships, and pharmacokinetic profiles of nonpeptidic difluoromethylene ketones as novel inhibitors of human chymase

      JOURNAL OF MEDICINAL CHEMISTRY
    27. Boackle, RJ; Dutton, SL; Fei, H; Vesely, J; Malamud, D; Furness, AR
      Salivary non-immunoglobulin agglutinin inhibits human leukocyte elastase digestion of acidic proline-rich salivary proteins

      JOURNAL OF DENTAL RESEARCH
    28. Li, FQ; Horwitz, M
      Characterization of mutant neutrophil elastase in severe congenital neutropenia

      JOURNAL OF BIOLOGICAL CHEMISTRY
    29. Naumov, P; Jovanovski, G; Drew, MGB; Ng, SW
      Outer-sphere coordination, N-coordination and O-coordination of the deprotonated saccharin in copper(II) saccharinato complexes. Implications for thesaccharinato carbonyl stretching frequency

      INORGANICA CHIMICA ACTA
    30. Wright, PA; Wilmouth, RC; Clifton, IJ; Schofield, CJ
      Kinetic and crystallographic analysis of complexes formed between elastaseand peptides from beta-casein

      EUROPEAN JOURNAL OF BIOCHEMISTRY
    31. Baskova, IP; Zavalova, LL
      Proteinase inhibitors from the medicinal leech Hirudo medicinalis

      BIOCHEMISTRY-MOSCOW
    32. Gladysheva, IP; Moroz, NA; Papisova, AI; Larionova, NI
      Soybean Bowman-Birk inhibitor conjugates with clinical dextran. Synthesis and antiproteolytic activity

      BIOCHEMISTRY-MOSCOW
    33. Stein, RL; DeCicco, C; Nelson, D; Thomas, B
      Slow-binding inhibition of gamma-glutamyl transpeptidase by gamma-boroGlu

      BIOCHEMISTRY
    34. Groutas, WC; Epp, JB; Kuang, RZ; Ruan, SM; Chong, LS; Venkataraman, R; Tu, J; He, S; Yu, HY; Fu, QH; Li, YH; Truong, TM; Vu, NT
      1,2,5-Thiadiazolidin-3-one 1,1 dioxide: A powerful scaffold for probing the S ' subsites of (chymo)trypsin-like serine proteases

      ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS
    35. Prakash, GKS; Mandal, M; Schweizer, S; Petasis, NA; Olah, GA
      A facile stereocontrolled synthesis of anti-alpha-(trifluoromethyl)-beta-amino alcohols

      ORGANIC LETTERS
    36. Valueva, TA; Revina, TA; Mosolov, VV; Mentele, R
      Primary structure of potato Kunitz-type serine proteinase inhibitor

      BIOLOGICAL CHEMISTRY
    37. Laborde, MA; Mascaretti, OA
      Synthesis and elastase inhibitory evaluation of phosphate esters and mixedphosphate anhydride of penam sulfones

      MOLECULES
    38. Kawabata, K; Hagio, T; Matsumoto, S; Nakao, S; Orita, S; Aze, Y; Ohno, H
      Delayed neutrophil elastase inhibition prevents subsequent progression of acute lung injury induced by endotoxin inhalation in hamsters

      AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE
    39. Kim, KY; Lim, HK; Lee, KJ; Park, DH; Kang, KW; Chung, SI; Jung, KH
      Production and characterization of recombinant guamerin, an elastase-specific inhibitor, in the methylotrophic yeast Pichia pastoris

      PROTEIN EXPRESSION AND PURIFICATION
    40. Ying, QL; Simon, SR
      DNA from bronchial secretions modulates elastase inhibition by alpha(1)-proteinase inhibitor and oxidized secretory leukoprotease inhibitor

      AMERICAN JOURNAL OF RESPIRATORY CELL AND MOLECULAR BIOLOGY
    41. Viglio, S; Lupi, A; Luisetti, M; Zanaboni, G; Cetta, G; Iadarola, P
      Activity of different proteases in a complex mixture and in vitro study oftheir reciprocal interferences by micellar electrokinetic chromatography

      JOURNAL OF MICROCOLUMN SEPARATIONS
    42. He, S; Kuang, RZ; Venkataraman, R; Tu, J; Truong, TM; Chan, HK; Groutas, WC
      Potent inhibition of serine proteases by heterocyclic sulfide derivatives of 1,2,5-thiadiazolidin-3-one 1,1 dioxide

      BIOORGANIC & MEDICINAL CHEMISTRY
    43. Kuang, RZ; Epp, JB; Ruan, S; Chong, LS; Venkataraman, R; Tu, J; He, S; Truong, TM; Groutas, WC
      Utilization of the 1,2,5-thiadiazolidin-3-one 1,1 dioxide scaffold in the design of potent inhibitors of serine proteases: SAR studies using carboxylates

      BIOORGANIC & MEDICINAL CHEMISTRY
    44. Jakobsen, P; Horneman, AM; Persson, E
      Inhibitors of the tissue factor/factor VIIa-induced coagulation: Synthesisand in vitro evaluation of novel 2-aryl substituted pyrido[3,4-d][1,3]-, pyrido[2,3-d][1,3]-, pyrazino[2,3-d][1,3]-, pyrimido[4,5-d][1,3]-, pyrazolo[3,4-d][1,3]-, thieno[3,2-d][1,3]- and thieno[2,3-d][1,3]-oxazin-4-ones

      BIOORGANIC & MEDICINAL CHEMISTRY
    45. Buynak, JD; Doppalapudi, VR; Rao, AS; Nidamarthy, SD; Adam, G
      The synthesis and evaluation of 2-substituted-7(alkylidene)cephalosporin sulfones as beta-lactamase inhibitors

      BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
    46. Waxman, L; Darke, PL
      The herpesvirus proteases as targets for antiviral chemotherapy

      ANTIVIRAL CHEMISTRY & CHEMOTHERAPY
    47. Filippusson, H; Erlendsson, LS; Lowe, CR
      Design, synthesis and evaluation of biomimetic affinity ligands for elastases

      JOURNAL OF MOLECULAR RECOGNITION
    48. Saturnino, C; Fusco, B; Saturnino, P; De Martino, G; Rocco, F; Lancelot, JC
      Evaluation of analgesic and anti-inflammatory activity of novel beta-lactam monocyclic compounds

      BIOLOGICAL & PHARMACEUTICAL BULLETIN
    49. Vaday, GG; Lider, O
      Extracellular matrix moieties, cytokines, and enzymes: dynamic effects on immune cell behavior and inflammation

      JOURNAL OF LEUKOCYTE BIOLOGY
    50. Achilles, K; Schirmeister, T; Otto, HH
      beta-lactam derivatives as enzyme inhibitors: 1-peptidyl derivatives of 4-phenylazetidin-2-one as inhibitors of elastase and papain

      ARCHIV DER PHARMAZIE
    51. Wright, PA; Wilmouth, RC; Clifton, IJ; Schofield, CJ
      'pH-jump' crystallographic analyses of gamma-lactam-porcine pancreatic elastase complexes

      BIOCHEMICAL JOURNAL
    52. Veinberg, G; Vorona, M; Grigan, N; Kanepe, I; Shestakova, I; Strakov, A; Lukevics, E
      Cephalosporins with carbonate functions at positions 3 and 7

      KHIMIYA GETEROTSIKLICHESKIKH SOEDINENII
    53. Grigan, N; Veinberg, G; Shestakova, I; Kanepe, I; Lukevics, E
      Synthesis and biological properties of 3-(dihydroxybenzoyloxy)methyl- and 3-(diacetoxybenzoyloxy)methyl-7 alpha-chlorocephalosporanate sulfones

      KHIMIYA GETEROTSIKLICHESKIKH SOEDINENII
    54. Liu, Z; Zhou, XY; Shapiro, SD; Shipley, JM; Twining, SS; Diaz, LA; Senior, RM; Werb, Z
      The serpin alpha 1-proteinase inhibitor is a critical substrate for gelatinase B/MMP-9 in vivo

      CELL
    55. Mellor, JM; Reid, G; El-Sagheer, AH; El-Tamany, ESH
      Reaction of alkyl and aryl grignard reagents with trifluoroacetyldihydropyrans and other cyclic beta-alkoxy-alpha,beta-unsaturated trifluoromethylketones

      TETRAHEDRON
    56. Dougherty, JM; Probst, DA; Robinson, RE; Moore, JD; Klein, TA; Snelgrove, KA; Hanson, PR
      Ring-closing metathesis strategies to cyclic sulfamide peptidomimetics

      TETRAHEDRON
    57. Page, MI; Laws, AP
      The chemical reactivity of beta-lactams, beta-sultams and beta-phospholactams

      TETRAHEDRON
    58. Wilmouth, RC; Li, YH; Wright, PA; Claridge, TDW; Aplin, RT; Schofield, CJ
      Reaction of clavams with elastase reveals a general method for inhibiting 'serine' enzymes

      TETRAHEDRON
    59. Wang, ZJ; Neidlein, R; Krieger, C
      A new approach to the synthesis of heteroannulated 3,1-oxazin-4-ones from beta-enamino esters and phosgeneiminium salts

      SYNTHESIS-STUTTGART
    60. Leung, D; Abbenante, G; Fairlie, DP
      Protease inhibitors: Current status and future prospects

      JOURNAL OF MEDICINAL CHEMISTRY
    61. Coppola, GM
      Synthesis and reactions of 2-hetero-4H-3,1-benzoxazin-4-ones

      JOURNAL OF HETEROCYCLIC CHEMISTRY
    62. Liu, Z; Shapiro, SD; Zhou, XY; Twining, SS; Senior, RM; Giudice, GJ; Fairley, JA; Diaz, LA
      A critical role for neutrophil elastase in experimental bullous pemphigoid

      JOURNAL OF CLINICAL INVESTIGATION
    63. Nakanishi, I; Kinoshita, T; Sato, A; Tada, T
      Structure of porcine pancreatic elastase complexed with FR901277, a novel macrocyclic inhibitor of elastases, at 1.6 angstrom resolution

      BIOPOLYMERS
    64. Gladysheva, IP; Balabushevich, NG; Moroz, NA; Larionova, NI
      Isolation and characterization of soybean Bowman-Birk inhibitor from different sources

      BIOCHEMISTRY-MOSCOW
    65. Hill, AT; Campbell, EJ; Hill, SL; Bayley, DL; Stockley, RA
      Association between airway bacterial load and markers of airway inflammation in patients with stable chronic bronchitis

      AMERICAN JOURNAL OF MEDICINE
    66. Li-Pan, ZS; Joshi, HV; Digenis, GA
      Synthesis and mechanism of action of novel thiocarbamate inhibitors of human leukocyte elastase

      JOURNAL OF ENZYME INHIBITION
    67. Larksarp, C; Alper, H
      A simple synthesis of 2-substituted-4H-3,1-benzoxazin-4-ones by palladium-catalyzed cyclocarbonylation of o-odoanilines with acid chlorides

      ORGANIC LETTERS
    68. Beauve, C; Tjoens, G; Touillaux, R; Lamotte-Brasseur, J; Marchand-Brynaert, J; Fastrez, J
      1-alkoxycarbonyl-3-bromoazetidin-2-ones as potential elastase inhibitors

      EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
    69. Martyn, DC; Moore, MJB; Abell, AD
      Succinimide and saccharin-based enzyme-activated inhibitors of serine proteases

      CURRENT PHARMACEUTICAL DESIGN
    70. Metz, WA; Peet, NP
      Inhibitors of human neutrophil elastase as a potential treatment for inflammatory diseases

      EXPERT OPINION ON THERAPEUTIC PATENTS
    71. Gibson, TLB; Cohen, P
      Inflammation-related neutrophil proteases, cathepsin G and elastase, function as insulin-like growth factor binding protein proteases

      GROWTH HORMONE & IGF RESEARCH
    72. Fujita, J; Skold, CM; Daughton, DM; Ertl, RF; Takahara, J; Rennard, SI
      Modulation of elastase binding to elastin by human alveolar macrophage-derived lipids

      AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE
    73. Edwards, JV; Bopp, AF; Batiste, S; Ullah, AJ; Cohen, IK; Diegelmann, RF; Montante, SJ
      Inhibition of elastase by a synthetic cotton-bound serine protease inhibitor: in vitro kinetics and inhibitor release

      WOUND REPAIR AND REGENERATION
    74. Witko-Sarsat, V; Halbwachs-Mecarelli, L; Schuster, A; Nusbaum, P; Ueki, I; Canteloup, S; Lenoir, G; Descamps-Latscha, B; Nadel, JA
      Proteinase 3, a potent secretagogue in airways, is present in cystic fibrosis sputum

      AMERICAN JOURNAL OF RESPIRATORY CELL AND MOLECULAR BIOLOGY
    75. Fujie, K; Shinguh, Y; Yamazaki, A; Hatanaka, H; Okamoto, M; Okuhara, M
      Inhibition of elastase-induced acute inflammation and pulmonary emphysema in hamsters by a novel neutrophil elastase inhibitor FR901277

      INFLAMMATION RESEARCH
    76. Reiner, JE; Lim-Wilby, MS; Brunck, TK; Ha-Uong, T; Goldman, EA; Abelman, MA; Nutt, RF; Semple, JE; Tamura, SY
      Investigation of the S-3 site of thrombin: Design, synthesis and biological activity of 4-substituted 3-amino-2-pyridones incorporating P-1-argininals

      BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
    77. Yu, KL; Civiello, R; Roberts, DGM; Seiler, SM; Meanwell, NA
      Solid-phase synthesis of benzisothiazolones as serine protease inhibitors

      BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
    78. Garrett, GS; McPhail, SJ; Tornheim, K; Correa, PE; McIver, JM
      Synthesis of potent and selective inhibitors of human plasma kallikrein

      BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
    79. Pryor, KE; La Clair, JJ
      A rapid method to identify exo-protease inhibitors

      BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
    80. Khan, JK; Bu, HZ; Samarendra, ZZ; Maiti, N; Micetich, RG
      A rapid and reliable solid-phase extraction-LC/MS/MS assay for the determination of two novel human leukocyte elastase inhibitors, SYN-1390 and SYN-1396, in rat plasma

      JOURNAL OF PHARMACEUTICAL AND BIOMEDICAL ANALYSIS
    81. Konttinen, YT; Kaapa, E; Hukkanen, M; Gu, XH; Takagi, M; Santavirta, S; Alaranta, H; Li, TF; Suda, A
      Cathepsin G in degenerating and healthy discal tissue

      CLINICAL AND EXPERIMENTAL RHEUMATOLOGY
    82. Hamilton-Miller, JMT
      beta-lactams: variations on a chemical theme, with some surprising biological results

      Journal of antimicrobial chemotherapy
    83. Tamas, L; Gunda, TE; Sztaricskai, F
      On the preparation of 2-substituted cephalosporin sulfoxides via anionic intermediates

      JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1
    84. Dall'Acqua, W; Halin, C; Rodrigues, ML; Carter, P
      Elastase substrate specificity tailored through substrate-assisted catalysis and phage display

      PROTEIN ENGINEERING
    85. Sanderson, PEJ
      Small, noncovalent serine protease inhibitors

      MEDICINAL RESEARCH REVIEWS
    86. Dallegri, F; Dapino, P; Arduino, N; Bertolotto, M; Ottonello, L
      Cefoperazone prevents the inactivation of alpha(1)-antitrypsin by activated neutrophils

      ANTIMICROBIAL AGENTS AND CHEMOTHERAPY
    87. Murcko, MA; Caron, PR; Charifson, PS
      Structure-based drug design

      ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 34
    88. Beauve, C; Bouchet, M; Touillaux, R; Fastrez, J; Marchand-Brynaert, J
      Synthesis, reactivity and biochemical evaluation of 1,3-substituted azetidin-2-ones as enzyme inhibitors

      TETRAHEDRON
    89. Palomo, C; Aizpurua, JM; Gracenea, JJ
      Diastereoselective conjugate reduction and enolate trapping with glyoxylate imines. A concise approach to beta-lactams that involves a ternary combination of components

      JOURNAL OF ORGANIC CHEMISTRY
    90. Poupart, MA; Fazal, G; Goulet, S; Mar, LT
      Solid-phase synthesis of peptidyl trifluoromethyl ketones

      JOURNAL OF ORGANIC CHEMISTRY
    91. Cabaret, D; Adediran, SA; Gonzalez, MJG; Pratt, RF; Wakselman, M
      Synthesis and reactivity with beta-lactamases of "penicillin-like" cyclic depsipeptides

      JOURNAL OF ORGANIC CHEMISTRY
    92. Gutschow, M
      One-pot reactions of N-(mesyloxy)phthalimides with secondary amines to 2-ureidobenzamides, 2-ureidobenzoic acids, ethyl 2-ureidobenzoates, or isatoicanhydrides

      JOURNAL OF ORGANIC CHEMISTRY
    93. MacDonald, SJF; Clarke, GDE; Dowle, MD; Harrison, LA; Hodgson, ST; Inglis, GGA; Johnson, MR; Shah, P; Upton, RJ; Walls, SB
      A flexible, practical, and stereoselective synthesis of enantiomerically pure trans-5-oxohexahydropyrrolo[3,2-b]pyrroles (pyrrolidine-trans-lactams),a new class of serine protease inhibitors, using acyliminium methodology

      JOURNAL OF ORGANIC CHEMISTRY
    94. Iijima, K; Katada, J; Yasuda, E; Uno, I; Hayashi, Y
      N-[2,2-dimethyl-3-(N-(4-cyanobenzoyl)amino)nonanoyl]-L-phenylalalanine ethyl ester as a stable ester-type inhibitor of chymotrypsin-like serine proteases: Structural requirements for potent inhibition of alpha-chymotrypsin

      JOURNAL OF MEDICINAL CHEMISTRY
    95. Coppola, GM
      The Chemistry of 4H-3,1-benzoxazin-4-ones

      JOURNAL OF HETEROCYCLIC CHEMISTRY
    96. Taylor, P; Anderson, V; Dowden, J; Flitsch, SL; Turner, NJ; Loughran, K; Walkinshaw, MD
      Novel mechanism of inhibition of elastase by beta-lactams is defined by two inhibitor crystal complexes

      JOURNAL OF BIOLOGICAL CHEMISTRY
    97. Buczek-Thomas, JA; Nugent, MA
      Elastase-mediated release of heparan sulfate proteoglycans from pulmonary fibroblast cultures - A mechanism for basic fibroblast growth factor (bFGF)release and attenuation of bFGF binding following elastase-induced injury

      JOURNAL OF BIOLOGICAL CHEMISTRY
    98. Fujie, K; Shinguh, Y; Inamura, N; Yasumitsu, R; Okamoto, M; Okuhara, M
      Release of neutrophil elastase and its role in tissue injury in acute inflammation: effect of the elastase inhibitor, FR134043

      EUROPEAN JOURNAL OF PHARMACOLOGY
    99. McBride, JD; Freeman, HNM; Leatherbarrow, RJ
      Selection of human elastase inhibitors from a conformationally-constrainedcombinatorial peptide library

      EUROPEAN JOURNAL OF BIOCHEMISTRY
    100. Czapinska, H; Otlewski, J
      Structural and energetic determinants of the S-1-site specificity in serine proteases

      EUROPEAN JOURNAL OF BIOCHEMISTRY


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Documento generato il 06/06/20 alle ore 12:34:39