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La ricerca find articoli where soggetti phrase all words 'PORCINE PANCREATIC ELASTASE' sort by level,fasc_key/DESCEND, pagina_ini_num/ASCEND ha restituito 126 riferimenti
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    1. Rodis, NP; Digenis, GA
      Synthesis and in-vitro evaluation of novel low molecular weight thiocarbamates as inhibitors of human leukocyte elastase

      JOURNAL OF ENZYME INHIBITION
    2. Walker, B; Lynas, JF
      Strategies for the inhibition of serine proteases

      CELLULAR AND MOLECULAR LIFE SCIENCES
    3. Beardsell, M; Hinchliffe, PS; Wood, JM; Wilmouth, RC; Schofield, CJ; Page, MI
      beta-Sultams - A novel class of serine protease inhibitors

      CHEMICAL COMMUNICATIONS
    4. Wilmouth, RC; Edman, K; Neutze, R; Wright, PA; Clifton, IJ; Schneider, TR; Schofield, CJ; Hajdu, J
      X-ray snapshots of serine protease catalysis reveal a tetrahedral intermediate

      NATURE STRUCTURAL BIOLOGY
    5. Vagnoni, LM; Gronostaj, M; Kerrigan, JE
      6-Acylamino-2-[(ethylsulfonyl)oxy]-1H-isoindole-1,3-diones mechanism-basedinhibitors of human leukocyte elastase and cathepsin G: Effect of chirality in the 6-acylamino substituent on inhibitory potency and selectivity

      BIOORGANIC & MEDICINAL CHEMISTRY
    6. Akahoshi, F; Ashimori, A; Yoshimura, T; Imada, T; Nakajima, M; Mitsutomi, N; Kuwahara, S; Ohtsuka, T; Fukaya, C; Miyazaki, M; Nakamura, N
      Non-peptidic inhibitors of human chymase. Synthesis, structure-activity relationships, and pharmacokinetic profiles of a series of 5-amino-6-oxo-1,6-dihydropyrimidine-containing trifluoromethyl ketones

      BIOORGANIC & MEDICINAL CHEMISTRY
    7. Ghani, U; Ng, KKS; Atta-ur-Rahman; Choudhary, MI; Ullah, N; James, MNG
      Crystal structure of gamma-chymotrypsin in complex with 7-hydroxycoumarin

      JOURNAL OF MOLECULAR BIOLOGY
    8. Wright, PA; Wilmouth, RC; Clifton, IJ; Schofield, CJ
      Kinetic and crystallographic analysis of complexes formed between elastaseand peptides from beta-casein

      EUROPEAN JOURNAL OF BIOCHEMISTRY
    9. Koteva, KP; Cantin, AM; Neugebauer, WA; Escher, E
      Synthesis and evaluation of novel beta-lactam inhibitors of human leukocyte elastase

      CANADIAN JOURNAL OF CHEMISTRY-REVUE CANADIENNE DE CHIMIE
    10. Waxman, L; Darke, PL
      The herpesvirus proteases as targets for antiviral chemotherapy

      ANTIVIRAL CHEMISTRY & CHEMOTHERAPY
    11. Filippusson, H; Erlendsson, LS; Lowe, CR
      Design, synthesis and evaluation of biomimetic affinity ligands for elastases

      JOURNAL OF MOLECULAR RECOGNITION
    12. Donkor, IO
      A survey of calpain inhibitors

      CURRENT MEDICINAL CHEMISTRY
    13. Achilles, K; Schirmeister, T; Otto, HH
      beta-lactam derivatives as enzyme inhibitors: 1-peptidyl derivatives of 4-phenylazetidin-2-one as inhibitors of elastase and papain

      ARCHIV DER PHARMAZIE
    14. Vogt, W
      Cleavage of the fifth component of complement and generation of a functionally active C5b6-like complex by human leukocyte elastase

      IMMUNOBIOLOGY
    15. Wilmouth, RC; Li, YH; Wright, PA; Claridge, TDW; Aplin, RT; Schofield, CJ
      Reaction of clavams with elastase reveals a general method for inhibiting 'serine' enzymes

      TETRAHEDRON
    16. Botos, I; Meyer, E; Nguyen, M; Swanson, SM; Koomen, JM; Russell, DH; Meyer, EF
      The structure of an insect chymotrypsin

      JOURNAL OF MOLECULAR BIOLOGY
    17. Hilpert, K; Hansen, G; Wessner, H; Schneider-Mergener, J; Hohne, W
      Characterizing and optimizing protease/peptide inhibitor interactions, a new application for spot synthesis

      JOURNAL OF BIOCHEMISTRY
    18. Nakanishi, I; Kinoshita, T; Sato, A; Tada, T
      Structure of porcine pancreatic elastase complexed with FR901277, a novel macrocyclic inhibitor of elastases, at 1.6 angstrom resolution

      BIOPOLYMERS
    19. Schalkwijk, J; Wiedow, O; Hirose, S
      The trappin gene family: proteins defined by an N-terminal transglutaminase substrate domain and a C-terminal four-disulphide core

      BIOCHEMICAL JOURNAL
    20. Barbato, G; Cicero, DO; Nardi, MC; Steinkuhler, C; Cortese, R; De Francesco, R; Bazzo, R
      The solution structure of the N-terminal proteinase domain of the hepatitis C virus (HCV) NS3 protein provides new insights into its activation and catalytic mechanism

      JOURNAL OF MOLECULAR BIOLOGY
    21. Boatman, PD; Ogbu, CO; Eguchi, M; Kim, HO; Nakanishi, H; Cao, BL; Shea, JP; Kahn, M
      Secondary structure peptide mimetics: Design, synthesis, and evaluation ofbeta-strand mimetic thrombin inhibitors

      JOURNAL OF MEDICINAL CHEMISTRY
    22. Iijima, K; Katada, J; Yasuda, E; Uno, I; Hayashi, Y
      N-[2,2-dimethyl-3-(N-(4-cyanobenzoyl)amino)nonanoyl]-L-phenylalalanine ethyl ester as a stable ester-type inhibitor of chymotrypsin-like serine proteases: Structural requirements for potent inhibition of alpha-chymotrypsin

      JOURNAL OF MEDICINAL CHEMISTRY
    23. Taylor, P; Anderson, V; Dowden, J; Flitsch, SL; Turner, NJ; Loughran, K; Walkinshaw, MD
      Novel mechanism of inhibition of elastase by beta-lactams is defined by two inhibitor crystal complexes

      JOURNAL OF BIOLOGICAL CHEMISTRY
    24. McBride, JD; Freeman, HNM; Leatherbarrow, RJ
      Selection of human elastase inhibitors from a conformationally-constrainedcombinatorial peptide library

      EUROPEAN JOURNAL OF BIOCHEMISTRY
    25. Hudaky, P; Kaslik, G; Venekei, I; Graf, L
      The differential specificity of chymotrypsin A and B is determined by amino acid 226

      EUROPEAN JOURNAL OF BIOCHEMISTRY
    26. Wilmouth, RC; Kassamally, S; Westwood, NJ; Sheppard, RJ; Claridge, TDW; Aplin, RT; Wright, PA; Pritchard, GJ; Schofield, CJ
      Mechanistic insights into the inhibition of serine proteases by monocycliclactams

      BIOCHEMISTRY
    27. Simons, JWFA; Cox, RC; Egmond, MR; Verheij, HM
      Rational design of alpha-keto triglyceride analogues as inhibitors for Staphylococcus hyicus lipase

      BIOCHEMISTRY
    28. Wieczorek, M; Gyorkos, A; Spruce, LW; Ettinger, A; Ross, SE; Kroona, HS; Burgos-Lepley, CE; Bratton, LD; Drennan, TS; Garnert, DL; Von Burg, G; Pilkington, CG; Cheronis, JC
      Biochemical characterization of alpha-ketooxadiazoie inhibitors of elastases

      ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS
    29. YAVIN EJ; FRIDKIN M
      PEPTIDES DERIVED FROM HUMAN C-REACTIVE PROTEIN INHIBIT THE ENZYMATIC-ACTIVITIES OF HUMAN-LEUKOCYTE ELASTASE AND CATHEPSIN-G - USE OF OVERLAPPING PEPTIDE SEQUENCES TO IDENTIFY A UNIQUE INHIBITOR

      The journal of peptide research
    30. NEGRINI D; PASSI A; DELUCA G; MISEROCCHI G
      PROTEOGLYCAN INVOLVEMENT DURING DEVELOPMENT OF LESIONAL PULMONARY-EDEMA

      American journal of physiology. Lung cellular and molecular physiology
    31. JING H; BABU YS; MOORE D; KILPATRICK JM; LIU XY; VOLANAKIS JE; NARAYANA SVL
      STRUCTURES OF NATIVE AND COMPLEXED COMPLEMENT FACTOR-D - IMPLICATIONSOF THE ATYPICAL HIS57 CONFORMATION AND SELF-INHIBITORY LOOP IN THE REGULATION OF SPECIFIC SERINE-PROTEASE ACTIVITY

      Journal of Molecular Biology
    32. GUY L; VIDAL J; COLLET A; AMOUR A; REBOUDRAVAUX M
      DESIGN AND SYNTHESIS OF HYDRAZINOPEPTIDES AND THEIR EVALUATION AS HUMAN-LEUKOCYTE ELASTASE INHIBITORS

      Journal of medicinal chemistry
    33. CREGGE RJ; DURHAM SL; FARR RA; GALLION SL; HARE CM; HOFFMAN RV; JANUSZ MJ; KIM HO; KOEHL JR; MEHDI S; METZ WA; PEET NP; PELTON JT; SCHREUDER HA; SUNDER S; TARDIF C
      INHIBITION OF HUMAN NEUTROPHIL ELASTASE - 4 - DESIGN, SYNTHESIS, X-RAY CRYSTALLOGRAPHIC ANALYSIS, AND STRUCTURE-ACTIVITY-RELATIONSHIPS FOR A SERIES OF P-2-MODIFIED, ORALLY-ACTIVE PEPTIDYL PENTAFLUOROETHYL KETONES

      Journal of medicinal chemistry
    34. GUTSCHOW M; NEUMANN U
      NOVEL THIENO[2,3-D][1,3]OXAZIN-4-ONES AS INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE

      Journal of medicinal chemistry
    35. Wilmouth, RC; Westwood, NJ; Anderson, K; Brownlee, W; Claridge, TDW; Clifton, IJ; Pritchard, GJ; Aplin, RT; Schofield, CJ
      Inhibition of elastase by N-sulfonylaryl beta-lactams: Anatomy of a stableacyl-enzyme complex

      BIOCHEMISTRY
    36. KOSTOULAS G; HORLER D; NAGGI A; CASU B; BAICI A
      ELECTROSTATIC INTERACTIONS BETWEEN HUMAN-LEUKOCYTE ELASTASE AND SULFATED GLYCOSAMINOGLYCANS - PHYSIOLOGICAL IMPLICATIONS

      Biological chemistry
    37. DIDIERJEAN C; DELDUCA V; BENEDETTI E; AUBRY A; ZOUIKRI M; MARRAUD M; BOUSSARD G
      X-RAY STRUCTURES OF AZA-PROLINE-CONTAINING PEPTIDES

      The journal of peptide research
    38. VANKUPPEVELT TH; VANDELEST CHA; VERSTEEG EMM; DEKHUIJZEN PNR; VEERKAMP JH
      INDUCTION OF EMPHYSEMATOUS LESIONS IN RAT LUNG BY BETA-D-XYLOSIDE, ANINHIBITOR OF PROTEOGLYCAN SYNTHESIS

      American journal of respiratory cell and molecular biology
    39. GUTSCHOW M; NEUMANN U
      INHIBITION OF CATHEPSIN-G BY 4H-3,1-BENZOXAZIN-4-ONES

      Bioorganic & medicinal chemistry
    40. LYNAS J; WALKER B
      PEPTIDYL INVERSE ESTERS OF P-METHOXYBENZOIC ACID - A NOVEL CLASS OF POTENT INACTIVATOR OF THE SERINE PROTEASES

      Biochemical journal
    41. CUNNINGHAM MA; BLAJCHMAN MA; SHEFFIELD WP
      IMPACT OF MUTATIONS AT THE P4 AND P5 POSITIONS ON THE REACTION OF ANTITHROMBIN WITH THROMBIN AND ELASTASE

      Thrombosis research
    42. WASSERMAN HH; PETERSEN AK
      A CONVERGENT SYNTHESIS OF POSTSTATIN - APPLICATION OF THE ACYL CYANOPHOSPHORANE COUPLING PROCEDURE IN THE FORMATION OF A PEPTIDIC ALPHA-KETO AMIDE

      Tetrahedron letters
    43. HOFFMAN RV; SAENZ JE
      A SHORT, EFFICIENT SYNTHESIS OF MONOFLUORO KETOMETHYLENE PEPTIDE ISOSTERE CORE UNITS

      Tetrahedron letters
    44. ABELL AD; OLDHAM MD
      SYNTHESIS AND X-RAY CRYSTALLOGRAPHIC STRUCTURE OF LEUCINE-PHENYLALANYL SUCCINIMIDE-BASED PSEUDOPEPTIDES

      Journal of organic chemistry
    45. BAKER BM; MURPHY KP
      DISSECTING THE ENERGETICS OF A PROTEIN-PROTEIN INTERACTION - THE BINDING OF OVOMUCOID 3RD-DOMAIN TO ELASTASE

      Journal of Molecular Biology
    46. LU WY; APOSTOL I; QASIM MA; WARNE N; WYNN R; ZHANG WL; ANDERSON S; CHIANG YW; OGIN E; ROTHBERG I; RYAN K; LASKOWSKI M
      BINDING OF AMINO-ACID SIDE-CHAINS TO S-1 CAVITIES OF SERINE PROTEINASES

      Journal of Molecular Biology
    47. REGAN J; MCGARRY D; BRUNO J; GREEN D; NEWMAN J; HSU CY; KLINE J; BARTON J; TRAVIS J; CHOI YM; VOLZ F; PAULS H; HARRISON R; ZILBERSTEIN A; BENSASSON SA; CHANG M
      ANIONIC-MEDIATED AND LIPOPHILIC-MEDIATED SURFACE BINDING INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE

      Journal of medicinal chemistry
    48. BABINE RE; BENDER SL
      MOLECULAR RECOGNITION OF PROTEIN-LIGAND COMPLEXES - APPLICATIONS TO DRUG DESIGN

      Chemical reviews
    49. PLOTNICK MI; SCHECHTER NM; WANG ZM; LIU XZ; RUBIN H
      ROLE OF THE P6-P3' REGION OF THE SERPIN REACTIVE LOOP IN THE FORMATION AND BREAKDOWN OF THE INHIBITORY COMPLEX

      Biochemistry
    50. ORLOWSKI M; CARDOZO C; ELEUTERI AM; KOHANSKI R; KAM CM; POWERS JC
      REACTIONS OF [C-14] 3,4-DICHLOROISOCOUMARIN WITH SUBUNITS OF PITUITARY AND SPLEEN MULTICATALYTIC PROTEINASE COMPLEXES (PROTEASOMES)

      Biochemistry
    51. BONNEAU PR; GRANDMAITRE C; GREENWOOD DJ; LAGACE L; LAPLANTE SR; MASSARIOL MJ; OGILVIE WW; OMEARA JA; KAWAI SH
      EVIDENCE OF A CONFORMATIONAL CHANGE IN THE HUMAN CYTOMEGALOVIRUS PROTEASE UPON BINDING OF PEPTIDYL-ACTIVATED CARBONYL INHIBITORS

      Biochemistry
    52. GROUTAS WC; KUANG RZ; VENKATARAMAN R; EPP JB; RUAN SM; PRAKASH O
      STRUCTURE-BASED DESIGN OF A GENERAL-CLASS OF MECHANISM-BASED INHIBITORS OF THE SERINE PROTEINASES EMPLOYING A NOVEL AMINO ACID-DERIVED HETEROCYCLIC SCAFFOLD

      Biochemistry
    53. FRUH H; KOSTOULAS G; MICHEL BA; BAICI A
      HUMAN MYELOBLASTIN (LEUKOCYTE PROTEINASE-3) - REACTIONS WITH SUBSTRATES, INACTIVATORS AND ACTIVATORS IN COMPARISON WITH LEUKOCYTE ELASTASE

      Biological chemistry
    54. BETSUYAKU T; NISHIMURA M; YOSHIOKA A; TAKEYABU K; MIYAMOTO K; KAWAKAMI Y
      ELASTIN-DERIVED PEPTIDES AND NEUTROPHIL ELASTASE IN BRONCHOALVEOLAR LAVAGE FLUID

      American journal of respiratory and critical care medicine
    55. YING QL; KEMME M; SIMON SR
      ALGINATE, THE SLIME EXOPOLYSACCHARIDE OF PSEUDOMONAS-AERUGINOSA, BINDS HUMAN-LEUKOCYTE ELASTASE, RETARDS INHIBITION BY ALPHA(1)-PROTEINASE INHIBITOR, AND ACCELERATES INHIBITION BY SECRETORY LEUKOPROTEASE INHIBITOR

      American journal of respiratory cell and molecular biology
    56. JARVEST RL; PARRATT MJ; DEBOUCK CM; GORNIAK JG; JENNINGS LJ; SERAFINOWSKA HT; STRICKLER JE
      INHIBITION OF HSV-1 PROTEASE BY BENZOXAZINONES

      Bioorganic & medicinal chemistry letters
    57. LABARRE S; LONGEON A; BARTHELEMY M; GUYOT M; LECAER JP; BARGIBANT G
      CHARACTERIZATION OF A NOVEL ELASTASE INHIBITOR FROM A FAN CORAL

      Comptes rendus de l'Academie des sciences. Serie 3, Sciences de la vie
    58. YAVIN EJ; YAN L; DESIDERIO D; FRIDKIN M
      SYNTHETIC PEPTIDES DERIVED FROM THE SEQUENCE OF HUMAN C-REACTIVE PROTEIN INHIBIT THE ENZYMATIC-ACTIVITIES OF HUMAN-LEUKOCYTE ELASTASE AND HUMAN-LEUKOCYTE CATHEPSIN-G

      International journal of peptide & protein research
    59. ZEMBOWER DE; NEUDAUER CL; WICK MJ; AMES MM
      PEPTIDE BORONIC ACIDS - VERSATILE SYNTHETIC LIGANDS FOR AFFINITY-CHROMATOGRAPHY OF SERINE PROTEINASES

      International journal of peptide & protein research
    60. KLINE T; MUELLER L; SIEBERMCMASTER E; LAU WF; MEYERS CA
      A PSEUDOPEPTIDE INCORPORATING THE TETRAHYDROPHTHALAZINE NUCLEUS, A CONSTRAINED AZA ANALOG OF PHENYLALANINE

      International journal of peptide & protein research
    61. VERGELY I; LAUGAA P; REBOUDRAVAUX M
      INTERACTION OF HUMAN-LEUKOCYTE ELASTASE WITH A N-ARYL AZETIDINONE SUICIDE SUBSTRATE - CONFORMATIONAL-ANALYSES BASED ON THE MECHANISM OF ACTION OF SERINE PROTEINASES

      Journal of molecular graphics
    62. WINKLER U; ALLISON NJ; WOODARD SL; GAULT RA; EWOLDT GR; KAM CM; ABUELYAMAN A; POWERS JC; HUDIG D
      CHARACTERIZATION, APPLICATION AND POTENTIAL USES OF BIOTIN-TAGGED INHIBITORS FOR LYMPHOCYTE SERINE PROTEASES (GRANZYMES)

      Molecular immunology
    63. LABOW RS; ERFLE DJ; SANTERRE JP
      ELASTASE-INDUCED HYDROLYSIS OF SYNTHETIC SOLID SUBSTRATES - POLY(ESTER-UREA-URETHANE) AND POLY(ETHER-UREA-URETHANE)

      Biomaterials
    64. ALLEN KN; BELLAMACINA CR; DING XC; JEFFERY CJ; MATTOS C; PETSKO GA; RINGE D
      AN EXPERIMENTAL APPROACH TO MAPPING THE BINDING SURFACES OF CRYSTALLINE PROTEINS

      Journal of physical chemistry
    65. EDWARDS PD; ANDISIK DW; STRIMPLER AM; GOMES B; TUTHILL PA
      NONPEPTIDIC INHIBITORS OF HUMAN NEUTROPHIL ELASTASE .7. DESIGN, SYNTHESIS, AND IN-VITRO ACTIVITY OF A SERIES OF PYRIDOPYRIMIDINE TRIFLUOROMETHYL KETONES

      Journal of medicinal chemistry
    66. PATTERSON JE; OLLMANN IR; CRAVATT BF; BOGER DL; WONG CH; LERNER RA
      INHIBITION OF OLEAMIDE HYDROLASE CATALYZED-HYDROLYSIS OF THE ENDOGENOUS SLEEP-INDUCING LIPID CIS-9-OCTADECENAMIDE

      Journal of the American Chemical Society
    67. SCHILTZ M; FOURME R; BROUTIN I; PRANGE T
      THE CATALYTIC SITE OF SERINE PROTEINASES AS A SPECIFIC BINDING CAVITYFOR XENON

      Structure
    68. MEYER EF; BOTOS I; SCAPOZZA L; ZHANG DC
      BACKWARD BINDING AND OTHER STRUCTURAL SURPRISES

      Perspectives in drug discovery and design
    69. BERGLUND GI; SMALAS AO; HANSEN LK; WILLASSEN NP
      CRYSTALLIZATION AND PRELIMINARY-X-RAY CRYSTALLOGRAPHIC STUDIES OF NATIVE ELASTASE FROM NORTH-ATLANTIC SALMON (SALMO-SALAR)

      Acta crystallographica. Section D, Biological crystallography
    70. TOTH I; CHRISTODOULOU M; BANKOWSKY K; FLINN N; GIBBONS WA; GODEAU G; MOCZAR E; HORNEBECK W
      DESIGN OF POTENT LIPOPHILIC-PEPTIDE INHIBITORS OF HUMAN NEUTROPHIL ELASTASE - IN-VITRO AND IN-VIVO STUDIES

      International journal of pharmaceutics
    71. HOFFMAN RV; KIM HO
      THE STEREOSELECTIVE SYNTHESIS OF 2-ALKYL GAMMA-KETO ACID AND HETEROCYCLIC KETOMETHYLENE PEPTIDE ISOSTERE CORE UNITS USING CHIRAL ALKYLATIONBY 2-TRIFLYLOXY ESTERS

      Journal of organic chemistry
    72. PARISI MF; GATTUSO G; NOTTI A; RAYMO FM; ABELES RH
      CONVERSION OF ALPHA-KETO ESTERS INTO BETA,BETA-DIFLUORO-ALPHA-KETO ESTERS AND CORRESPONDING ACIDS - A SIMPLE ROUTE TO A NOVEL CLASS OF SERINE-PROTEASE INHIBITORS

      Journal of organic chemistry
    73. KERRIGAN JE; OLEKSYSZYN J; KAM CM; SELZLER J; POWERS JC
      MECHANISM-BASED ISOCOUMARIN INHIBITORS FOR HUMAN-LEUKOCYTE ELASTASE -EFFECT OF THE 7-AMINO SUBSTITUENT AND 3-ALKOXY GROUP IN 3-ALKOXY-7-AMINO-4-CHLOROISOCOUMARINS ON INHIBITORY POTENCY

      Journal of medicinal chemistry
    74. VEALE CA; DAMEWOOD JR; STEELMAN GB; BRYANT C; GOMES B; WILLIAMS J
      NONPEPTIDIC INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE .4. DESIGN, SYNTHESIS, AND IN-VITRO AND IN-VIVO ACTIVITY OF A SERIES OF BETA-CARBOLINONE-CONTAINING TRIFLUOROMETHYL KETONES

      Journal of medicinal chemistry
    75. VEALE CA; BERNSTEIN PR; BRYANT C; CECCARELLI C; DAMEWOOD JR; EARLEY R; FEENEY SW; GOMES B; KOSMIDER BJ; STEELMAN GB; THOMAS RM; VACEK EP; WILLIAMS JC; WOLANIN DJ; WOOLSON S
      NONPEPTIDIC INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE .5. DESIGN, SYNTHESIS, AND X-RAY CRYSTALLOGRAPHY OF A SERIES OF ORALLY-ACTIVE 5-AMINOPYRIMIDIN-6-ONE-CONTAINING TRIFLUOROMETHYL KETONES

      Journal of medicinal chemistry
    76. TAIPALE J; LOHI J; SAARINEN J; KOVANEN PT; KESKIOJA J
      HUMAN MAST-CELL CHYMASE AND LEUKOCYTE ELASTASE RELEASE LATENT TRANSFORMING GROWTH FACTOR-B1 FROM THE EXTRACELLULAR-MATRIX OF CULTURED HUMANEPITHELIAL AND ENDOTHELIAL-CELLS

      The Journal of biological chemistry
    77. TOMOMURA A; TOMOMURA M; FUKUSHIGE T; AKIYAMA M; KUBOTA N; KUMAKI K; NISHII Y; NOIKURA T; SAHEKI T
      MOLECULAR-CLONING AND EXPRESSION OF SERUM CALCIUM-DECREASING FACTOR (CALDECRIN)

      The Journal of biological chemistry
    78. KELLENBERGER C; BOUDIER C; BERMUDEZ I; BIETH JG; LUU B; HIETTER H
      SERINE-PROTEASE INHIBITION BY INSECT PEPTIDES CONTAINING A CYSTEINE KNOT AND A TRIPLE-STRANDED BETA-SHEET

      The Journal of biological chemistry
    79. CADENE M; BOUDIER C; DEMARCILLAC GD; BIETH JG
      INFLUENCE OF LOW-MOLECULAR-MASS HEPARIN ON THE KINETICS OF NEUTROPHILELASTASE INHIBITION BY MUCUS PROTEINASE-INHIBITOR

      The Journal of biological chemistry
    80. YAMANE T; IWASAKI A; SUZUKI A; ASHIDA T; KAWATA Y; SAKIYAMA F
      CRYSTAL-STRUCTURE OF STREPTOMYCES-ERYTHRAEUS TRYPSIN AT 1.9-ANGSTROM RESOLUTION

      Journal of Biochemistry
    81. DING XC; RASMUSSEN BF; DEMUTH HU; RINGE D; STEINMETZ ACU
      NATURE OF THE INACTIVATION OF ELASTASE BY N-PEPTIDYL-O-AROYL HYDROXYLAMINE AS A FUNCTION OF PH

      Biochemistry
    82. JACKSON DS; BROWN AD; SCHAEPER RJ; POWERS JC
      A KINETIC-STUDY OF THE HYDROLYSIS OF THE N-TOSYLALANINE ESTER OF 3-HYDROXY-5-PHENYLPYRROLE AND RELATED-COMPOUNDS BY HUMAN-LEUKOCYTE ELASTASE

      Archives of biochemistry and biophysics
    83. MATTOS C; RASMUSSEN B; DING XC; PETSKO GA; RINGE D
      ANALOGOUS INHIBITORS OF ELASTASE DO NOT ALWAYS BIND ANALOGOUSLY

      Nature structural biology
    84. BERNSTEIN PR; KOSMIDER BJ; VACEK EP; VEALE CA; GOMES BC
      EXAMINATION OF PEPTIDIC ALPHA',BETA-DIAMINO-ALPHA,ALPHA-DIFLUOROKETONES AS INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE

      Bioorganic & medicinal chemistry letters
    85. HLASTA DJ; BELL MR; BOAZ NW; COURT JJ; DESAI RC; FRANKE CA; MURA AJ; SUBRAMANYAM C; DUNLAP RP
      A BENZISOTHIAZOLONE CLASS OF POTENT, SELECTIVE MECHANISM-BASED INHIBITORS OF HUMAN-LEUKOCYTE ELASTASE

      Bioorganic & medicinal chemistry letters
    86. SATO S; KATO S; ARISAKA Y; TAKAHASHI H; TOMOIKE H
      PULMONARY HEMODYNAMICS IN AWAKE RATS FOLLOWING TREATMENT WITH ENDOTRACHEAL PANCREATIC ELASTASE

      The European respiratory journal
    87. SMALAS AO; HEIMSTAD ES; HORDVIK A; WILLASSEN NP; MALE R
      COLD ADAPTION OF ENZYMES - STRUCTURAL COMPARISON BETWEEN SALMON AND BOVINE TRYPSINS

      Proteins
    88. AMOUR A; COLLET A; DUBAR C; REBOUDRAVAUX M
      SYNTHESIS AND PROTEASE-CATALYZED HYDROLYSIS OF A NOVEL HYDRAZINOPEPTIDE

      International journal of peptide & protein research
    89. EDWARDS PD; BERNSTEIN PR
      SYNTHETIC INHIBITORS OF ELASTASE

      Medicinal research reviews
    90. NEDER KM; FRENCH SA; MILLER SPF
      SYNTHESIS AND INHIBITORY ACTIVITY OF DIFLUOROKETONE SUBSTRATE-ANALOGSOF N-MYRISTOYLTRANSFERASE

      Tetrahedron
    91. APLIN RT; ROBINSON CV; SCHOFIELD CJ; WESTWOOD NJ
      DOES THE OBSERVATION OF NONCOVALENT COMPLEXES BETWEEN BIOMOLECULES BYELECTROSPRAY-IONIZATION MASS-SPECTROMETRY NECESSARILY REFLECT SPECIFIC SOLUTION INTERACTIONS

      Journal of the Chemical Society, Chemical Communications
    92. DURHAM SL; HARE CM; ANGELASTRO MR; BURKHART JP; KOEHL JR; MARQUART AL; MEHDI S; FEET NP; JANUSZ MJ
      PHARMACOLOGY OF FLUORO-1-(1-METHYLETHYL)-2-OXOBUTYL]-L-PROLINAMIDE (MDL-101,146) - A POTENT ORALLY-ACTIVE INHIBITOR OF HUMAN NEUTROPHIL ELASTASE

      The Journal of pharmacology and experimental therapeutics
    93. ARTYMIUK PJ; POIRRETTE AR; GRINDLEY HM; RICE DW; WILLETT P
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ASDD Area Sistemi Dipartimentali e Documentali, Università di Bologna, Catalogo delle riviste ed altri periodici
Documento generato il 21/01/21 alle ore 04:21:49