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The amide hydrogen of (-)-indolactam-V and benzolactam-V8's plays a critical role in protein kinase C binding and tumor-promoting activities
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Protein kinase C-delta C2-like domain is a binding site for actin and enables actin redistribution in neutrophils
BIOCHEMICAL JOURNAL
A Dictyostelium nuclear phosphatidylinositol phosphate kinase required fordevelopmental gene expression
EMBO JOURNAL
Structural basis of binding of high-affinity ligands to protein kinase C: Prediction of the binding modes through a new molecular dynamics method andevaluation by site-directed mutagenesis
JOURNAL OF MEDICINAL CHEMISTRY
Na+/K(+)ATPase activity inhibition and isoform-specific translocation of protein kinase C following angiotensin II administration in isolated eel enterocytes
JOURNAL OF ENDOCRINOLOGY
Membrane translocation of novel protein kinase Cs is regulated by phosphorylation of the C2 domain
JOURNAL OF BIOLOGICAL CHEMISTRY
Roles of ionic residues of the C1 domain in protein kinase C-alpha activation and the origin of phosphatidylserine specificity
JOURNAL OF BIOLOGICAL CHEMISTRY
Membrane targeting by C1 and C2 domains
JOURNAL OF BIOLOGICAL CHEMISTRY
Role of hydrophobic residues in the C1b domain of protein kinase C delta on ligand and phospholipid interactions
JOURNAL OF BIOLOGICAL CHEMISTRY
The C1 domain of protein kinase C as a lipid bilayer surface sensing module
BIOCHEMISTRY
Signaling and subcellular targeting by membrane-binding domains
ANNUAL REVIEW OF BIOPHYSICS AND BIOMOLECULAR STRUCTURE
Chemistry and clinical biology of the bryostatins
BIOORGANIC & MEDICINAL CHEMISTRY
Synthesis and PKC isozyme surrogate binding of indothiolactam-V, a new thioamide analogue of tumor promoting indolactam-V
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Reversible protein kinase C activation in PC12 cells: effect of NGF treatment
EUROPEAN JOURNAL OF NEUROSCIENCE
Synthesis and tumor-promoting activities of 12-epi-phorbol-12, 13-dibutyrate
BIOSCIENCE BIOTECHNOLOGY AND BIOCHEMISTRY
Properties and functions of diacylglycerol kinases
CELLULAR SIGNALLING
Protein kinase C signaling and oxidative stress
FREE RADICAL BIOLOGY AND MEDICINE
Conformationally constrained analogues of diacylglycerol (DAG). 17. Contrast between sn-1 and sn-2 DAG lactones in binding to protein kinase C
JOURNAL OF MEDICINAL CHEMISTRY
The cysteine-rich regions of the regulatory domains of Raf and protein kinase C as retinoid receptors
JOURNAL OF EXPERIMENTAL MEDICINE
Subtype-specific translocation of diacylglycerol kinase alpha and gamma and its correlation with protein kinase C
JOURNAL OF BIOLOGICAL CHEMISTRY
Recombinant Clb domain of PKC delta triggers meiotic maturation upon microinjection in Xenopus laevis oocytes
FEBS LETTERS
The C1 and C2 domains of protein kinase C are independent membrane targeting modules, with specificity for phosphatidylserine conferred by the C1 domain
BIOCHEMISTRY
1,2-sn-Diacylglycerol in plant cells: Product, substrate and regulator
PLANT PHYSIOLOGY AND BIOCHEMISTRY
Selective binding of bryostatin analogues to the cysteine rich domains of protein kinase C isozymes
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Role of the membrane in the modulation of the activity of protein kinase C
JOURNAL OF LIPOSOME RESEARCH
The rational design of potential chemotherapeutic agents: Synthesis of bryostatin analogues
MEDICINAL RESEARCH REVIEWS
beta 2-chimaerin is a novel target for diacylglycerol: Binding properties and changes in subcellular localization mediated by ligand binding to its C1 domain
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
Administration of dexamethasone up-regulates protein kinase C activity andthe expression of gamma and epsilon protein kinase C isozymes in the rat brain
JOURNAL OF NEUROCHEMISTRY
Probing the binding of indolactam-V to protein kinase C through site-directed mutagenesis and computational docking simulations
JOURNAL OF MEDICINAL CHEMISTRY
Interplay of C1 and C2 domains of protein kinase C-alpha in its membrane binding and activation
JOURNAL OF BIOLOGICAL CHEMISTRY
Protein kinase D activation by deletion of its cysteine-rich motifs
FEBS LETTERS
Protein kinase C delta
EUROPEAN JOURNAL OF BIOCHEMISTRY
Differential roles of the tandem C1 domains of protein kinase C delta in the biphasic down-regulation induced by bryostatin 1
CANCER RESEARCH
Stimulation of A(2A) adenosine receptor phosphorylation by protein kinase C activation: Evidence for regulation by-multiple protein kinase C isoforms
BIOCHEMISTRY
Rapid in vitro conformational changes of the catalytic site of PKC alpha assessed by FIM-1 fluorescence
BIOCHEMISTRY
Ca2+ and protein kinase C signaling for histamine and sulfidoleukotrienes released from human cultured mast cells (vol 257, pg 895, 1999)
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS
Ca2+ and protein kinase C signaling for histamine and sulfidoleukotrienes released from human cultured mast cells
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS
Tumor promoter benzoyl peroxide induces sulfhydryl oxidation in protein kinase C: Its reversibility is related to the cellular resistance to peroxide-induced cytotoxicity
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS
CONFORMATIONALLY CONSTRAINED ANALOGS OF DIACYLGLYCEROL (DAG) - 14 - DISSECTION OF THE ROLES OF THE SN-1 AND SN-2 CARBONYLS IN DAG MIMETICS BY ISOPHARMACOPHORE REPLACEMENT
Bioorganic & medicinal chemistry letters
UP-REGULATION OF A HYDRA-VULGARIS CPKC GENE IS TIGHTLY COUPLED TO THEDIFFERENTIATION OF HEAD STRUCTURES
Development, genes and evolution
Neuronal signaling systems and ethanol dependence
MOLECULAR NEUROBIOLOGY
SIGNAL-TRANSDUCTION IN ENVIRONMENTAL NEUROTOXICITY
Annual review of pharmacology and toxicology
PROTEIN-KINASE-C - A PARADIGM FOR REGULATION OF PROTEIN FUNCTION BY 2MEMBRANE-TARGETING MODULES
Biochimica et biophysica acta, MR. Reviews on biomembranes
SYMPOSIUM OVERVIEW - TOXICITY OF NONCOPLANAR PCBS
Fundamental and applied toxicology
CA2-UNSATURATED FATTY ACID-INDUCED MUTANT PROTEIN-KINASE-C ACTIVITY -INDICATION OF INHIBITORY CA2+-BINDING SITE IN PROTEIN-KINASE-C-ALPHA(MODULATION OF CIS)
Biochemical journal
CALPHOSTIN-C INDUCES SELECTIVE DISASSEMBLY OF THE GOLGI-COMPLEX BY A PROTEIN-KINASE C-INDEPENDENT MECHANISM
European journal of cell biology
THE NEUROTOXICITY OF POLYCHLORINATED-BIPHENYLS
Neurotoxicology
INTERACTIVE EFFECTS OF ENVIRONMENTALLY RELEVANT POLYCHLORINATED-BIPHENYLS AND DIOXINS ON [H-3]PHORBOL ESTER BINDING IN RAT CEREBELLAR GRANULE CELLS
Environmental health perspectives
ORTHO-SUBSTITUTED POLYCHLORINATED-BIPHENYLS ACTIVATE RESPIRATORY BURST MEASURED AS LUMINOL-AMPLIFIED CHEMOLUMINESCENCE IN HUMAN GRANULOCYTES
Toxicology and applied pharmacology
Repeated exposure of adult rats to Aroclor 1254 causes brain region-specific changes in intracellular Ca2+ buffering and protein kinase C activity inthe absence of changes in tyrosine hydroxylase
TOXICOLOGY AND APPLIED PHARMACOLOGY
SYNTHESIS AND BINDING-STUDIES OF THE 116-MER PEPTIDE-CONTAINING THE DOUBLE CYSTEINE-RICH MOTIFS OF PROTEIN-KINASE-C-GAMMA
Tetrahedron letters
GREEN FLUORESCENT PROTEIN (GFP)-TAGGED CYSTEINE-RICH DOMAINS FROM PROTEIN-KINASE-C AS FLUORESCENT INDICATORS FOR DIACYLGLYCEROL SIGNALING IN LIVING CELLS
The Journal of cell biology
THE ROLE OF C2 DOMAINS IN CA2-ACTIVATED AND CA2+ INDEPENDENT PROTEIN-KINASE CS IN APLYSIA()
The Journal of biological chemistry
INHIBITORY PROPERTIES OF THE REGULATORY DOMAINS OF HUMAN PROTEIN-KINASE-C-ALPHA AND MOUSE PROTEIN-KINASE C-EPSILON
The Journal of biological chemistry
MGCRACGAP, A NEW HUMAN GTPASE-ACTIVATING PROTEIN FOR RAC AND CDC42 SIMILAR TO DROSOPHILA ROTUNDRACGAP GENE-PRODUCT, IS EXPRESSED IN MALE GERM-CELLS
The Journal of biological chemistry
Contributions to maxima in protein kinase C activation
JOURNAL OF BIOLOGICAL CHEMISTRY
DELETION ANALYSIS OF PROTEIN-KINASE-C-ALPHA REVEALS A NOVEL REGULATORY SEGMENT
Journal of Biochemistry (Tokyo)
DISSIMILAR PHORBOL ESTER BINDING-PROPERTIES OF THE INDIVIDUAL CYSTEINE-RICH MOTIFS OF PROTEIN-KINASE-D
FEBS letters
VERAPAMIL INHIBITS PROLIFERATION, MIGRATION AND PROTEIN-KINASE-C ACTIVITY IN HUMAN RETINAL-PIGMENT EPITHELIAL-CELLS
Experimental Eye Research
ESTRADIOL ELEVATES PROTEIN-KINASE-C CATALYTIC ACTIVITY IN THE PREOPTIC AREA OF FEMALE RATS
Endocrinology
ROLE OF PROTEIN-KINASE-C AS A CELLULAR MEDIATOR OF ISCHEMIC PRECONDITIONING - A CRITICAL-REVIEW
Cardiovascular Research
Mechanism of the apparent cooperativity in the interaction of protein kinase C with phosphatidylserine
BIOCHEMISTRY
RATIONAL DESIGN, SYNTHESIS, AND EVALUATION OF A NEW-TYPE OF PKC INHIBITOR
Journal of the American Chemical Society
CGP-41251 AND TAMOXIFEN SELECTIVELY INHIBIT MITOGEN-ACTIVATED PROTEIN-KINASE ACTIVATION AND C-FOS PHOSPHOPROTEIN INDUCTION BY SUBSTANCE-P IN HUMAN ASTROCYTOMA-CELLS
Cell growth & differentiation
COMPARISON OF CHEMICAL CHARACTERISTICS OF THE FIRST AND THE 2ND CYSTEINE-RICH DOMAINS OF PROTEIN-KINASE C-GAMMA
Bioorganic & medicinal chemistry
TAXONOMY AND FUNCTION OF C1 PROTEIN-KINASE-C HOMOLOGY DOMAINS
Protein science
SYNTHESIS AND CHARACTERIZATION OF THE FIRST CYSTEINE-RICH DOMAIN OF NOVEL PROTEIN-KINASE-C
Bioorganic & medicinal chemistry letters
PROTEIN-KINASE-C AND PHOSPHOLIPASE-C - BILAYER INTERACTIONS AND REGULATION
Current opinion in structural biology
IN-VITRO ADDITION OF GLUTATHIONE TO BLOOD FROM ZINC-DEFICIENT RATS CORRECTS PLATELET DEFECTS - IMPAIRED AGGREGATION AND CALCIUM UP TAKE
Journal of nutritional biochemistry
LIPID BIOCHEMISTRY - FUNCTIONS OF GLYCEROLIPIDS AND SPHINGOLIPIDS IN CELLULAR SIGNALING
The FASEB journal
DEVELOPMENTAL-CHANGES IN THE INHIBITORY ACTIONS OF ETHANOL ON GLUTAMATE-INDUCED TRANSLOCATION OF PROTEIN-KINASE-C IN CEREBELLAR GRANULE NEURONS
Alcohol
REGULATION OF RAF-1 KINASE BY INTERACTION WITH THE LIPID 2ND-MESSENGER, PHOSPHATIDIC-ACID
Biochemical Society transactions
A CCHC METAL-BINDING DOMAIN IN NANOS IS ESSENTIAL FOR TRANSLATIONAL REGULATION
EMBO journal
STRUCTURE-ACTIVITY-RELATIONSHIPS OF POTENTIALLY NEUROTOXIC PCB CONGENERS IN THE RAT
Neurotoxicology
EMPIRICAL MODELING OF AN IN-VITRO ACTIVITY OF POLYCHLORINATED BIPHENYL CONGENERS AND MIXTURES
Environmental health perspectives
CHARACTERIZATION OF PROTEIN-KINASE-C IN PHOTORECEPTOR OUTER SEGMENTS
Journal of neurochemistry
A NOVEL GTPASE-ACTIVATING PROTEIN FOR RHO INTERACTS WITH A PDZ DOMAINOF THE PROTEIN-TYROSINE-PHOSPHATASE PTPL1
The Journal of biological chemistry
INTERACTION OF ALCOHOLS AND ANESTHETICS WITH PROTEIN-KINASE C-ALPHA
The Journal of biological chemistry
CYSTEINE-RICH REGIONS OF PROTEIN-KINASE C-DELTA ARE FUNCTIONALLY NONEQUIVALENT - DIFFERENCES BETWEEN CYSTEINE-RICH REGIONS OF NON-CALCIUM-DEPENDENT PROTEIN-KINASE C-DELTA AND CALCIUM-DEPENDENT PROTEIN-KINASE C-GAMMA
FEBS letters
CANCER-PREVENTIVE SELENOCOMPOUNDS INDUCE A SPECIFIC REDOX MODIFICATION OF CYSTEINE-RICH REGIONS IN CA2-DEPENDENT ISOENZYMES OF PROTEIN-KINASE-C()
Archives of biochemistry and biophysics
PROTEIN-KINASE-C INACTIVATION BY FENTONS-REACTION AT DISCRETE CU-SITES(+ BINDING)
Biochemistry and molecular biology international
REGULATION OF PROTEIN-KINASE-C - A TALE OF LIPIDS AND PROTEINS
Enzyme & protein
DEVELOPMENTALLY EXPRESSED MYOSIN HEAVY-CHAIN KINASE POSSESSES A DIACYLGLYCEROL KINASE DOMAIN
Protein science
SYNTHESIS AND CHARACTERIZATION OF THE 2ND CYSTEINE-RICH REGION OF MOUSE SKIN PKC-ETA
Bioorganic & medicinal chemistry letters
EFFECTS OF REPEATED ADMINISTRATION OF A K-OPIOID AGONIST ON PHORBOL ESTER BINDING TO MEMBRANE-BOUND PROTEIN-KINASE-C IN RAT-BRAIN
Biological & pharmaceutical bulletin
STRUCTURAL ASPECTS OF THE FUNCTIONAL MODULES IN HUMAN PROTEIN KINASE-C-ALPHA DEDUCED FROM COMPARATIVE ANALYSES
Proteins
ACTIVATION OF CONVENTIONAL MAMMALIAN PROTEIN-KINASE-C ISOFORMS EXPRESSED IN BUDDING YEAST MODULATES THE CELL DOUBLING TIME - POTENTIAL IN-VIVO SCREEN FOR PROTEIN-KINASE-C ACTIVATORS
Cancer detection and prevention
CALCIUM-BINDING AND ZINC-BINDING PROTEINS IN INTRACELLULAR-TRANSPORT
Biocell
ROLE OF THE RAB3A-BINDING DOMAIN IN TARGETING OF RABPHILIN-3A TO VESICLE MEMBRANES OF PC12 CELLS
Molecular and cellular biology
THE C-TERMINAL PART OF DIACYLGLYCEROL KINASE-ALPHA LACKING TINT - FINGERS SERVES AS A CATALYTIC DOMAIN
Biochemical journal
PHOSPHORYLATION OF MEMBRANE-PROTEINS IN ERYTHROCYTES TREATED WITH LEAD
Biochemical journal
PROTEIN-KINASE-D (PKD) ACTIVATION IN INTACT-CELLS THROUGH A PROTEIN-KINASE C-DEPENDENT SIGNAL-TRANSDUCTION PATHWAY
EMBO journal
PROTEIN-KINASE-C ISOENZYMES - REGULATION AND FUNCTION
Cancer surveys
DEVELOPMENTAL-CHANGES IN GLUTAMATE RECEPTOR-ACTIVATED TRANSLOCATION OF PROTEIN-KINASE-C IN CEREBELLAR GRANULE NEURONS
Developmental brain research
PROTEIN-KINASE-C - MOLECULAR AND CELLULAR TARGETS FOR THE ACTION OF ETHANOL
Alcoholism, clinical and experimental research
THE SOLUTION STRUCTURE OF THE RAF-1 CYSTEINE-RICH DOMAIN - A NOVEL RAS AND PHOSPHOLIPID-BINDING SITE
Proceedings of the National Academy of Sciences of the United Statesof America
ETHANOL ENHANCES THE IN-SITU PHOSPHORYLATION OF MARCKS AND PROTEIN-KINASE-C ACTIVITY IN PRIMARY CULTURES OF ASTROCYTES
Life sciences
THE PRODUCTION OF POST-GOLGI VESICLES REQUIRES A PROTEIN-KINASE C-LIKE MOLECULE, BUT NOT ITS PHOSPHORYLATING ACTIVITY
The Journal of cell biology
CLONING AND CHARACTERIZATION OF A GLUCOCORTICOID-INDUCED DIACYLGLYCEROL KINASE
The Journal of biological chemistry
IN-VITRO ACTIVATION AND SUBSTRATES OF RECOMBINANT, BACULOVIRUS-EXPRESSED HUMAN PROTEIN-KINASE C-MU
FEBS letters