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Tethered libraries: Solid-phase synthesis of substituted urea-linked bicyclic guanidines
JOURNAL OF COMBINATORIAL CHEMISTRY
Benzodiazepine receptor (BZR) ligands. 6 new 3-(2-,3- or 4-substituted benzyloxycarbonyl) derivatives of the 8-chloropyrazolo[5,1-c][1,2,4]benzotriazine 5-oxide: Receptor affinity and in vivo testing
MEDICINAL CHEMISTRY RESEARCH
A pyridone analogue of traditional cannabinoids. A new class of selective ligands for the CB2 receptor
BIOORGANIC & MEDICINAL CHEMISTRY
Recent developments in the synthesis, chemistry and applications of the fully unsaturated 1,2,4-oxadiazoles
JOURNAL OF CHEMICAL RESEARCH-S
Suppression of conditioned fear by administration of CCKB receptor antisense oligodeoxynucleotide into the lateral ventricle
PHARMACOPSYCHIATRY
2-Substituted 4-anilinopiperidines from 2H-thiopyran-2-thiones
TETRAHEDRON
Novel pyrazole cannabinoids: Insights into CB1 receptor recognition and activation
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Original 2-alkylamino-6-halogenoquinazolin-4(3H)-ones and K-ATP channel activity
JOURNAL OF MEDICINAL CHEMISTRY
Synthesis and characterization of a quinolinonic compound activating ATP-sensitive K+ channels in endocrine smooth muscle tissues
BRITISH JOURNAL OF PHARMACOLOGY
Synthesis of new fused heterocycles by annilation of pyridocinnolines
AFINIDAD
Tumor necrosis factor-alpha augments tumor effects in isolated hepatic perfusion with melphalan in a rat sarcoma model
JOURNAL OF IMMUNOTHERAPY
Role of NPYY1 receptors in cardiovascular control in the conscious rabbit
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY
Thermal behaviour of some spiro benzodiazepine derivatives
THERMOCHIMICA ACTA
Application of organolithium and related reagents in synthesis, part 24. Synthetic strategies based on aromatic metallation. A concise regiospecific conversion of benzoic acids into 2-(1-aryl-2-methoxycarbonylethyl)benzoic acids
SYNTHESIS-STUTTGART
Molecular docking reveals a novel binding site model for fentanyl at the mu-opioid receptor
JOURNAL OF MEDICINAL CHEMISTRY
Synthesis of 2-aminoquinazoline-4(3H)-one derivatives as potential potassium channel openers
JOURNAL OF HETEROCYCLIC CHEMISTRY
Antinociceptive effects of tetrahydrocannabinol side chain analogs: dependence upon route of administration
EUROPEAN JOURNAL OF PHARMACOLOGY
Intra-abdominal fibrosis after systemic and intraperitoneal therapy containing fluoropyrimidines
CANCER
Inhibition of H+,K+-ATPase by hinesol, a major component of So-jutsu, by interaction with enzyme in the E-1 state
BIOCHEMICAL PHARMACOLOGY
Stereoselective follow-up reactions of (S)-2-sulfanyl nitriles
TETRAHEDRON-ASYMMETRY
A convenient method for the N-acylation and esterification of hindered amino acids: Synthesis of ultra short acting opioid agonist, remifentanil
SYNLETT
Structure and receptor activity for classical cannabinoids
CURRENT MEDICINAL CHEMISTRY
The development of cannabinoid antagonists
CURRENT MEDICINAL CHEMISTRY
Norbornane compounds in pharmaceutical research
PHARMAZIE
beta-adrenoceptor subtype activities of trimetoquinol derivatives: Biochemical studies on human beta-adrenoceptors expressed in Chinese hamster ovarycells
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Manipulation of the tetrahydrocannabinol side chain delineates agonists, partial agonists, and antagonists
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Guanidine derivatives as combined thromboxane A(2) receptor antagonists and synthase inhibitors
JOURNAL OF MEDICINAL CHEMISTRY
The role of nitric oxide in sepsis - an overview
ACTA ANAESTHESIOLOGICA SCANDINAVICA
Cannabinoid transmission and pain perception
NEUROBIOLOGY OF DISEASE
ANTIPLATELET AND VASORELAXING ACTIONS OF APORPHINOIDS FROM CASSYTHA-FILIFORMIS
PTR. Phytotherapy research
ANTIPROLIFERATIVE AND CYTOTOXIC EFFECTS OF GELDANAMYCIN, CYTOCHALASIN-E, SURAMIN AND THIACETAZONE IN HUMAN PROSTATE XENOGRAFT TUMOR HISTOCULTURES
Pharmaceutical research
AUGMENTATION OF HEPATIC DOXORUBICIN EXTRACTION WITH EXTRACORPOREAL FILTRATION AVOIDS THE DOSE-DEPENDENT, NONLINEAR INCREASE IN AUC OBSERVEDWITH SYSTEMIC ADMINISTRATION
Cancer chemotherapy and pharmacology
HOMOLOGOUS DESENSITIZATION OF THE D-1A DOPAMINE-RECEPTOR - EFFICACY IN CAUSING DESENSITIZATION DISSOCIATES FROM BOTH RECEPTOR OCCUPANCY ANDFUNCTIONAL POTENCY
The Journal of pharmacology and experimental therapeutics
QUANTITATIVE-ANALYSIS OF THE STRUCTURAL REQUIREMENTS FOR BLOCKADE OF THE N-METHYL-D-ASPARTATE RECEPTOR AT THE PHENCYCLIDINE BINDING-SITE
Journal of medicinal chemistry
REGIONAL PHARMACOKINETICS OF DOXORUBICIN FOLLOWING HEPATIC ARTERIAL AND PORTAL VENOUS ADMINISTRATION - EVALUATION WITH HEPATIC VENOUS ISOLATION AND CHARCOAL HEMOPERFUSION
Cancer research
NEW HETEROCYCLES FROM THIENOPYRIDOCINNOLINES
Canadian journal of chemistry
LIVER-INJURY MODEL INDUCED IN MICE BY A CELLULAR IMMUNOLOGICAL MECHANISM - STUDY FOR USE IN IMMUNOPHARMACOLOGICAL EVALUATIONS
Pharmacological research
N,N-DIETHYLAMINO)-N-OCTYL-3,4,5-TRIMETHOXYBENZOATE ACTIONS ON CALCIUMDYNAMICS IN CULTURED VASCULAR SMOOTH-MUSCLE CELLS
Zhongguo yaoli xuebao
COMPARATIVE-STUDIES ON BETA-ADRENOLYTIC POTENCIES OF SOME NEW PHENOXYAMINOPROPANOL DERIVATIVES AND CELIPROLOL
Die Pharmazie
SYNTHESIS AND EVALUATION OF TRIMETOQUINOL DERIVATIVES - NOVEL THROMBOXANE A(2) PROSTAGLANDIN H-2 ANTAGONISTS WITH DIMINISHED BETA-ADRENERGIC AGONIST ACTIVITY
Journal of medicinal chemistry
POTENTIAL GABA(B) RECEPTOR ANTAGONISTS .8. THE SYNTHESIS OF 3-AMINO-N-ARYL-2-HYDROXY-PROPANE-1-SULFONAMIDES AND ANALOGS OF BACLOFEN CONTAINING NITRO-GROUPS
Australian Journal of Chemistry
OPEN TRIAL OF LAMOTRIGINE IN THE TREATMENT OF SELF-INJURIOUS-BEHAVIORIN AN ADOLESCENT WITH PROFOUND MENTAL-RETARDATION
Journal of child and adolescent psychopharmacology
THE SYNTHESIS OF LACTAM ANALOGS OF FENTANYL
Journal of the Chemical Society. Perkin transactions. I
PHARMACOKINETIC AND PHARMACODYNAMIC PROFILE OF TRIETHYLENE GLYCOL INDOMETHACIN ESTER AS A NEW ORAL PRODRUG
Journal of controlled release
EVALUATION OF AGONIST-ANTAGONIST PROPERTIES OF NITROGEN-MUSTARD AND CYANO DERIVATIVES OF DELTA(8)-TETRAHYDROCANNABINOL
Neuropharmacology
EFFECTS OF 8-(N-N-DIETHYLAMINO)OCTYL-3,4,5-TRIMETHOXYBENZOATE HYDROCHLORIDE (TMB-8) ON SKINNED MYOCARDIAL FIBERS OF THE RAT - REVERSIBLE INHIBITION OF CALCIUM-RELEASE FROM THE SARCOPLASMIC-RETICULUM
Naunyn-Schmiedeberg's archives of pharmacology
IN-VIVO CHARACTERIZATION OF A SPECIFIC CANNABINOID RECEPTOR ANTAGONIST (SR141716A) - INHIBITION OF DELTA(9)-TETRAHYDROCANNABINOL-INDUCED RESPONSES AND APPARENT AGONIST ACTIVITY
The Journal of pharmacology and experimental therapeutics
SYNTHESIS, RESOLUTION, AND PRELIMINARY EVALUATION OF AMINO-6(5)-HYDROXY-1-PHENYL-2,3-DIHYDRO-1H-INDENES AND RELATED DERIVATIVES AS DOPAMINE-RECEPTORS LIGANDS
Journal of medicinal chemistry
2-AMINO-4-METHYLPYRIDINE AS A POTENT INHIBITOR OF INDUCIBLE NO SYNTHASE ACTIVITY IN-VITRO AND IN-VIVO
British Journal of Pharmacology
NEW DIBENZAZEPINE DERIVATIVES WITH DISINHIBITORY AND OR ANTIDEPRESSANT POTENTIAL - NEUROCHEMICAL AND BEHAVIORAL-STUDY IN THE OPEN-FIELD ANDFORCED SWIMMING TESTS/
Behavioural pharmacology
PEROXIDASE-CATALYZED OXIDATION OF DIFFERENT DIBENZAZEPINE DERIVATIVES
Archiv der pharmazie
A COMPARISON OF THE EFFECTS OF TMB-8 AND NIFEDIPINE ON PRESSOR-RESPONSES TO ALPHA(1)-ADRENOCEPTOR AND ALPHA(2)-ADRENOCEPTOR AGONISTS IN PITHED RATS
Naunyn-Schmiedeberg's archives of pharmacology
THE CALCIUM-ANTAGONIST TMB-8 [3,4,5-TRIMETHOXYBENZOIC ACID 8-(DIETHYTAMINO)OCTYL ESTER] IS A POTENT, NONCOMPETITIVE, FUNCTIONAL ANTAGONIST AT DIVERSE NICOTINIC ACETYLCHOLINE-RECEPTOR SUBTYPES
The Journal of pharmacology and experimental therapeutics
PREVENTION AND REDUCTION OF NEURAL DAMAGE IN ISCHEMIC STROKES BY ,N'-DIETHYLAMINO)-N-ALKYL-3,4,5-TRIMETHOXYBENZOATE COMPOUNDS
The Journal of pharmacology and experimental therapeutics
DUAL-ACTING THROMBOXANE RECEPTOR ANTAGONIST SYNTHASE INHIBITORS - SYNTHESIS AND BIOLOGICAL PROPERTIES OF SUBSTITUTED-4-(3-PYRIDYL)-1,3-DIOXAN-5-YL]ALKENOIC ACIDS
Journal of medicinal chemistry
A NOVEL-APPROACH TO DUAL-ACTING THROMBOXANE RECEPTOR ANTAGONIST SYNTHASE INHIBITORS BASED ON THE LINK OF 1,3-DIOXANE-THROMBOXANE RECEPTOR ANTAGONISTS AND 1,3-DIOXANE-THROMBOXANE SYNTHASE INHIBITORS
Journal of medicinal chemistry
PENTATOMIC CYCLIC AGONISTS AND MUSCARINIC RECEPTORS - A 20 YEARS REVIEW
Il Farmaco
AN EVALUATION OF HEPATIC EXTRACTION AND CLEARANCE OF DOXORUBICIN
British Journal of Cancer
CLINICAL DRUG-RESISTANCE - THE ROLE OF FACTORS OTHER THAN P-GLYCOPROTEIN
The American journal of medicine
A PHARMACODYNAMIC MODEL TO INVESTIGATE THE STRUCTURE-ACTIVITY PROFILEOF A SERIES OF NOVEL OPIOID ANALGESICS
The Journal of pharmacology and experimental therapeutics
PYRIDOBENOZOXAZEPINE AND PYRIDOBENZOTHIAZEPINE DERIVATIVES AS POTENTIAL CENTRAL-NERVOUS-SYSTEM AGENTS - SYNTHESIS AND NEUROCHEMICAL STUDY
Journal of medicinal chemistry
AGENTS COMBINING THROMBOXANE RECEPTOR ANTAGONISM WITH THROMBOXANE SYNTHASE INHIBITION - [[[2-(1H-IMIDAZOL-1-YL)ETHYLIDENE]AMINO]OXY] ALKANOIC ACIDS
Journal of medicinal chemistry
6,6-DISUBSTITUTED HEX-5-ENOIC ACID-DERIVATIVES AS COMBINED THROMBOXANE A(2) RECEPTOR ANTAGONISTS AND SYNTHETASE INHIBITORS
Journal of medicinal chemistry
SYNTHESIS AND BIOLOGICAL EVALUATION OF 14-ALKOXYMORPHINANS .10. 14-O-METHYL DERIVATIVES OF 5-METHYLNALTREXONE AND 5-METHYLNALOXONE
Helvetica Chimica Acta
EFFECTS OF TMB-8, A PUTATIVE CALCIUM-ANTAGONIST, ON NEUROMUSCULAR-TRANSMISSION AND MUSCLE CONTRACTILITY IN THE MOUSE PHRENIC NERVE-HEMIDIAPHRAGM PREPARATION
Archives internationales de pharmacodynamie et de therapie
APPLICATION OF PHARMACOKINETICALLY GUIDED DOSE-ESCALATION WITH RESPECT TO CELL-CYCLE PHASE SPECIFICITY
Journal of the National Cancer Institute
INCREASED DOXORUBICIN LEVELS IN HEPATIC-TUMORS WITH REDUCED SYSTEMIC DRUG EXPOSURE ACHIEVED WITH COMPLETE HEPATIC VENOUS ISOLATION AND EXTRACORPOREAL CHEMOFILTRATION
Cancer chemotherapy and pharmacology
EFFECT OF TMB-8 ON ALPHA-ADRENOCEPTOR AGONIST AND KCL INDUCED-CONTRACTIONS IN ISOLATED RABBIT AORTA
General pharmacology
NEW APPROACHES IN PRECLINICAL AND CLINICAL PHARMACOKINETICS
Cancer surveys
IODODEOXYURIDINE UPTAKE AND RETENTION AS A MEASURE OF TUMOR-GROWTH
The Journal of nuclear medicine
ANANDAMIDE, AN ENDOGENOUS LIGAND OF THE CANNABINOID RECEPTOR, INDUCESHYPOMOTILITY AND HYPOTHERMIA IN-VIVO IN RODENTS
Pharmacology, biochemistry and behavior
THE SYNTHESIS OF A CONFORMATIONALLY RESTRAINED, COMBINED THROMBOXANE ANTAGONIST SYNTHASE INHIBITOR USING AN INTRAMOLECULAR STILLE-PALLADIUM-CATALYZED OR GRIGG-PALLADIUM-CATALYZED CYCLIZATION STRATEGY/
Tetrahedron letters
INTERACTIONS OF NONPROSTANOID TRIMETOQUINOL ANALOGS WITH THROMBOXANE A(2) PROSTAGLANDIN H-2 RECEPTORS IN HUMAN PLATELETS, RAT VASCULAR ENDOTHELIAL-CELLS AND RAT VASCULAR SMOOTH-MUSCLE CELLS/
The Journal of pharmacology and experimental therapeutics
CANNABINOID STRUCTURE-ACTIVITY-RELATIONSHIPS - CORRELATION OF RECEPTOR-BINDING AND INVIVO ACTIVITIES
The Journal of pharmacology and experimental therapeutics
NEW PYRIDOBENZODIAZEPINE DERIVATIVES AS POTENTIAL ANTIPSYCHOTICS - SYNTHESIS AND NEUROCHEMICAL STUDY
Journal of medicinal chemistry
NONSURGICAL MANAGEMENT OF RECURRENT COLORECTAL-CANCER
Cancer