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Synthesis and preliminary in vivo evaluation of 4-[I-123]iodo-N-{2-[4-(6-trifluoromethyl-2-pyridinyl)-1-piperazinyl]ethyl} benzamide, a potential SPECT radioligand for the 5-HT1A receptor
JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS
Visualisation of serotonin-1A (5-HT1A) receptors in the central nervous system
EUROPEAN JOURNAL OF NUCLEAR MEDICINE
The selective 5-HT1A receptor antagonist p-MPPI antagonizes sleep-waking and behavioural effects of 8-OH-DPAT in rats
BEHAVIOURAL BRAIN RESEARCH
Sleep and waking following microdialysis perfusion of the selective 5-HT1Areceptor antagonist p-MPPI into the dorsal raphe nucleus in the freely moving rat
BRAIN RESEARCH
Radioligands for the study of brain 5-HT1A receptors in vivo - Developmentof some new analogues of WAY
NUCLEAR MEDICINE AND BIOLOGY
Differential effects of 5-HT agonists and antagonists on the repeated acquisition and performance of response sequences in monkeys
BEHAVIOURAL PHARMACOLOGY
In vivo characterization of p-[F-18]MPPF, a fluoro analog of WAY-100635 for visualization of 5-HT1A receptors
SYNAPSE
Effect of alcohols on G-protein coupling of serotonin(1A) receptors from bovine hippocampus
BRAIN RESEARCH BULLETIN
Sleep-wake effects following the selective 5-HT1A receptor antagonist p-MPPI in the freely moving rat
BEHAVIOURAL BRAIN RESEARCH
The effects of compounds varying in selectivity as 5-HT1A receptor antagonists in three rat models of anxiety
NEUROPHARMACOLOGY
Reversal of morphine-induced apnea in the anesthetized rat by drugs that activate 5-hydroxytryptamine(1A) receptors
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Analogues of WAY 100635 as radiotracers for in vivo imaging of 5-HT1A receptors
JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS
Full and partial 5-HT1A receptor agonists disrupt learning and performancein rats
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Development of fluorine-18-labeled 5-HT1A antagonists
JOURNAL OF MEDICINAL CHEMISTRY
Differential discrimination of G-protein coupling of serotonin(1A) receptors from bovine hippocampus by an agonist and an antagonist
FEBS LETTERS
Partial antagonism of 8-OH-DPAT'S effects on male rat sexual behavior witha D-2, but not a 5-HMT1A, antagonist
BRAIN RESEARCH
Behavioural profiles in the mouse defence test battery suggest anxiolytic potential of 5-HT1A receptor antagonists
PSYCHOPHARMACOLOGY
DERIVATIVES OF WAY-100635 AS POTENTIAL IMAGING AGENTS FOR 5-HT1A RECEPTORS - SYNTHESES, RADIOSYNTHESES, AND IN-VITRO AND IN-VIVO EVALUATION
Nuclear medicine and biology
HIGH-YIELD RADIOSYNTHESIS AND PRELIMINARY IN-VIVO EVALUATION OF P-[F-18]MPPF, A FLUORO ANALOG OF WAY-100635
Nuclear medicine and biology
SEROTONIN(1B) RECEPTOR STIMULATION ENHANCES COCAINE REINFORCEMENT
The Journal of neuroscience
SYNTHESIS AND BIODISTRIBUTION OF ETRAHYDRO-1-NAPHTALENYL)PROPYL]-4-PHENYLPIPERAZINE (PNU-157760), A PUTATIVE RADIOLIGAND FOR 5-HT1A RECEPTORS
Bioorganic chemistry (Print)
MODULATION OF AGONIST AND ANTAGONIST INTERACTIONS IN SEROTONIN 1A RECEPTORS BY ALCOHOLS
FEBS letters
THE 5-HT1A RECEPTOR ANTAGONIST P-MPPI BLOCKS 5-HT1A AUTORECEPTORS ANDINCREASES DORSAL RAPHE UNIT-ACTIVITY IN AWAKE CATS
European journal of pharmacology
P-[F-18]-MPPF - A POTENTIAL RADIOLIGAND FOR PET STUDIES OF 5-HT1A RECEPTORS IN HUMANS
Synapse
THE 5-HT1A RECEPTOR ANTAGONIST P-MPPI BLOCKS RESPONSES MEDIATED BY POSTSYNAPTIC AND PRESYNAPTIC 5-HT1A RECEPTORS
Pharmacology, biochemistry and behavior
5-HYDROXYTRYPTAMINE(1A) RECEPTOR-MEDIATED INCREASES IN RECEPTOR EXPRESSION AND ACTIVATION OF NUCLEAR FACTOR-KAPPA-B IN TRANSFECTED CHINESE-HAMSTER OVARY CELLS
Molecular pharmacology
SEROTONIN 5-HT1A AND 5-HT2 1C RECEPTORS IN THE MIDBRAIN PERIAQUEDUCTAL GRAY DIFFERENTIALLY MODULATE DEFENSIVE RAGE BEHAVIOR ELICITED FROM THE MEDIAL HYPOTHALAMUS OF THE CAT/
Brain research
5-HT1A RECEPTORS IN LITHIUM-INDUCED CONDITIONED TASTE-AVERSION
Psychopharmacology
ANXIOLYTIC-LIKE PROFILE OF P-MPPI, A NOVEL 5HT(1A) RECEPTOR ANTAGONIST, IN THE MURINE ELEVATED PLUS-MAZE
Psychopharmacology
IN-VIVO SPECT IMAGING OF 5-HT1A RECEPTORS WITH [I-123] P-MPPI IN NONHUMAN-PRIMATES
Synapse
TIME-COURSE OF RECOVERY OF 5-HT1A RECEPTORS AND CHANGES IN 5-HT1A RECEPTOR MESSENGER-RNA AFTER IRREVERSIBLE INACTIVATION WITH EEDQ
Molecular brain research
A POTENTIAL 5-HT1A RECEPTOR ANTAGONIST - P-MPPI
Life sciences