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Parallel synthesis and pharmacological screening oi nonpeptide ligands of the neuropeptide Y receptor subtype Y-5
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Spatial requirements of the antagonist binding site of the NK2 receptor
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Neuropeptide receptor status in human tumor cell lines
ANTI-CANCER DRUGS
Maintaining cell sensitivity to G-protein coupled receptor agonists: Neurotensin and the role of receptor gene activation
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CURRENT MEDICINAL CHEMISTRY
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ANNUAL REVIEW OF PHARMACOLOGY AND TOXICOLOGY
Arginine mimetics
TETRAHEDRON
Stepwise modulation of neurokinin-3 and neurokinin-2 receptor affinity andselectivity in quinoline tachykinin receptor antagonists
JOURNAL OF MEDICINAL CHEMISTRY
Interaction of Met(297) in the seventh transmembrane segment of the tachykinin NK2 receptor with neurokinin A
JOURNAL OF BIOLOGICAL CHEMISTRY
Molecular and pharmacological characterization of the murine tachykinin NK3 receptor
EUROPEAN JOURNAL OF PHARMACOLOGY
Central AT(1) and AT(2) receptors mediate chronic intracerebroventricular angiotensin II-induced drinking in rats fed high sodium chloride diet from weaning
ACTA PHYSIOLOGICA SCANDINAVICA
Vitronectin receptor antagonists: Purine-based peptidomimetics
ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
Neurokinin receptor antagonists
EXPERT OPINION ON INVESTIGATIONAL DRUGS
Recent advances in neurokinin-3 receptor antagonists
EXPERT OPINION ON THERAPEUTIC PATENTS
Angiotensin antagonists (Reprinted from Receptor-Based Drug Design, pg 207-230, 1998)
JOURNAL OF RECEPTOR AND SIGNAL TRANSDUCTION RESEARCH
RGD mimetics containing a central hydantoin scaffold: alpha(v)beta(3) vs alpha(IIb)beta(3) selectivity requirements
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
NK1, NK2 and NK3 tachykinin receptor localization and tachykinin distribution in the ileum of the mouse
ANATOMY AND EMBRYOLOGY
The psychopharmacology of tachykinin NK-3 receptors in laboratory animals
PEPTIDES
Uncovering molecular mechanisms involved in activation of G protein-coupled receptors
ENDOCRINE REVIEWS
Privileged structures - An update
ANNUAL REPORTS IN MEDICINAL CHEMISTRY, VOL 35
Synthesis of a substance P antagonist with a somatostatin scaffold: Factors affecting agonism/antagonism at GPCRs and the role of pseudosymmetry
JOURNAL OF MEDICINAL CHEMISTRY
Respiratory actions of tachykinins in the nucleus of the solitary tract: characterization of receptors using selective agonists and antagonists
BRITISH JOURNAL OF PHARMACOLOGY
MEGA-SQ: A method using the SQuEAL function to find the optimal superposition of several quasi-flexible molecules
MEDICINAL CHEMISTRY RESEARCH
Nonpeptide vasopressin antagonists: A new group of hormone blockers entering the scene
EXPERIMENTAL AND CLINICAL ENDOCRINOLOGY & DIABETES
Effect of LF 16-0687MS, a new nonpeptide bradykinin B-2 receptor antagonist, in a rat model of closed head trauma
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Tachykinins stimulate release of peptide hormones (glucagon-like peptide-1) and paracrine (somatostatin) and neurotransmitter (vasoactive intestinal polypeptide) from porcine ileum through NK-1 receptors
DIGESTIVE DISEASES AND SCIENCES
Valsartan and the kidney: Present and future
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Agonists and inverse agonists for the herpesvirus 8-encoded constitutivelyactive seven-transmembrane oncogene product, ORF-74
JOURNAL OF BIOLOGICAL CHEMISTRY
CORTICOTROPIN-RELEASING FACTOR-RECEPTOR ANTAGONISTS
Expert opinion on therapeutic patents
HPLC ASSAYS TO SIMULTANEOUSLY DETERMINE THE ANGIOTENSIN-AT(1) ANTAGONIST LOSARTAN AS WELL AS ITS MAIN AND ACTIVE METABOLITE EXP3174 IN BIOLOGICAL-MATERIAL OF HUMANS AND RATS
Journal of pharmaceutical and biomedical analysis
HYPOTHALAMIC ANGIOTENSIN RECEPTOR SUBTYPES IN NORMOTENSIVE AND HYPERTENSIVE RATS
American journal of physiology. Heart and circulatory physiology
STERIC HINDRANCE MUTAGENESIS VERSUS ALANINE SCAN IN MAPPING OF LIGAND-BINDING SITES IN THE TACHYKININ NK1 RECEPTOR
Molecular pharmacology
SHARED DETERMINANTS OF RECEPTOR-BINDING FOR SUBTYPE-SELECTIVE, AND DUAL ENDOTHELIN-ANGIOTENSIN ANTAGONISTS ON THE AT(1) ANGIOTENSIN-II RECEPTOR
FEBS letters
PROBING OF THE NEUROPEPTIDE Y-Y-1-RECEPTORS INTERACTION WITH ANTIRECEPTOR ANTIBODIES
European journal of biochemistry
NONPEPTIDE ANGIOTENSIN-II RECEPTOR ANTAGO NISTS - POTENTIAL-DRUGS AGAINST HYPERTENSION
Chemicke listy
A STRUCTURAL RATIONALE FOR THE DESIGN OF WATER-SOLUBLE PEPTIDE-DERIVED NEUROKININ-1 ANTAGONISTS
Journal of receptor and signal transduction research
PHARMACOLOGICAL PROFILE OF TH-142177, NOVEL ORALLY-ACTIVE AT(1)-RECEPTOR ANTAGONIST
Fundamental and clinical pharmacology
TACHYKININ RECEPTORS MEDIATING NONCHOLINERGIC CONTRACTION OF THE GUINEA-PIG ISOLATED MAIN BRONCHUS IN RESPONSE TO FIELD STIMULATION
Clinical and experimental pharmacology and physiology
TACHYKININS MAY MEDIATE CAPSAICIN-INDUCED, BUT NOT VAGALLY INDUCED MOTILITY IN PORCINE ANTRUM
Peptides
THE TACHYKININ NK1 RECEPTOR - PART I - LIGANDS AND MECHANISMS OF CELLULAR ACTIVATION
Neuropeptides
THE CONFORMATIONAL CHANGE RESPONSIBLE FOR AT(1) RECEPTOR ACTIVATION IS DEPENDENT UPON 2 JUXTAPOSED ASPARAGINE RESIDUES ON TRANSMEMBRANE-HELICES-III AND TRANSMEMBRANE-HELICES-VII
The Journal of biological chemistry
NEUROKININ RECEPTOR INHIBITORS - FERMENTATION, ISOLATION, PHYSICOCHEMICAL PROPERTIES, STRUCTURE AND BIOLOGICAL-ACTIVITY
Journal of antibiotics
EFFECT OF SINGLE-POINT MUTATIONS OF THE HUMAN TACHYKININ NK1 RECEPTORON ANTAGONIST AFFINITY
European journal of pharmacology
THE EFFECT OF ANGIOTENSIN-II RECEPTOR ANTAGONISTS ON KIDNEY-FUNCTION IN 2-KIDNEY, 2-CLIP GOLDBLATT HYPERTENSIVE RATS
European journal of pharmacology
P-(4-HYDROXYBENZOYL)PHENYLALANINE - A PHOTOREACTIVE AMINO-ACID ANALOGAMENABLE TO RADIOIODINATION FOR ELUCIDATION OF PEPTIDE-PROTEIN INTERACTION APPLICATION TO SUBSTANCE-P RECEPTOR
Biochemistry
EFFECT OF THE TACHYKININ RECEPTOR ANTAGONISTS, SR-140333, PK-888, ANDSR-142801, ON CAPSAICIN-INDUCED MOUSE EAR EDEMA
Inflammation research
CONNECTIVITY AND ORIENTATION OF THE 7 HELICAL BUNDLE IN THE TACHYKININ NK-1 RECEPTOR PROBED BY ZINC SITE ENGINEERING
EMBO journal
EFFECT OF BRAIN ANGIOTENSIN-II AT(1), AT(2), AND CHOLINERGIC RECEPTORANTAGONISM ON DRINKING IN WATER-DEPRIVED RATS
Regulatory peptides
ANGIOTENSIN-II RECEPTOR SUBTYPE ANTAGONISTS CAN BOTH STIMULATE AND INHIBIT SALT APPETITE IN RATS
Regulatory peptides
THE INFLUENCE OF GUANYL NUCLEOTIDE ON AGONIST AND ANTAGONIST AFFINITYAT GUINEA-PIG CCK-B GASTRIN RECEPTORS - BINDING-STUDIES USING [H-3] PD140376/
Regulatory peptides
TARGETED MOLECULAR DIVERSITY - DESIGN AND DEVELOPMENT OF NONPEPTIDE ANTAGONISTS FOR CHOLECYSTOKININ AND TACHYKININ RECEPTORS
Immunopharmacology
INTERACTIONS OF NONPEPTIDE ANGIOTENSIN-II RECEPTOR ANTAGONISTS AT IMIDAZOLINE GUANIDINIUM RECEPTOR-SITES IN RAT FOREBRAIN/
Journal of cardiovascular pharmacology
CHARACTERIZATION OF CCKA RECEPTOR-MEDIATED PEPSINOGEN SECRETION IN PORCINE CHIEF CELLS
Pharmacology
RADIOLIGAND-DEPENDENT DISCREPANCY IN AGONIST AFFINITIES ENHANCED BY MUTATIONS IN THE KAPPA-OPIOID RECEPTOR
Molecular pharmacology
STRUCTURAL MOTIFS ENCODED BY INDIVIDUAL EXONS OF THE HUMAN NEUROKININ-1 RECEPTOR GENE INTERACT DIFFERENTIALLY WITH SELECTIVE AGONISTS AND ANTAGONISTS
Journal of neurochemistry
THE USE OF PHOTOLABELED PEPTIDES TO LOCALIZE THE SUBSTANCE-P-BINDING SITE IN THE HUMAN NEUROKININ-1 TACHYKININ RECEPTOR
European journal of biochemistry
INTERACTION OF BIPHENYLIMIDAZOLE AND IMIDAZOLEACRYLIC ACID NONPEPTIDEANTAGONISTS WITH VALINE-108 IN TM-III OF THE AT(1) ANGIOTENSIN RECEPTOR
British Journal of Pharmacology
THE NEURONAL ROLE OF ANGIOTENSIN-II IN THIRST, SODIUM APPETITE, COGNITION AND MEMORY
Biological Reviews of the Cambridge Philosophical Society
EFFECTS OF HCGRP-8-37 AND THE NK1-RECEPTOR ANTAGONIST SR-140.333 ON CAPSAICIN-EVOKED VASODILATION IN THE PIG NASAL-MUCOSA IN-VIVO
Acta Physiologica Scandinavica
PHARMACOLOGICAL CHARACTERIZATION OF ANGIOTENSIN-II AT(2) RECEPTOR SUBTYPE HETEROGENEITY IN THE RAT ADRENAL-CORTEX AND MEDULLA
Endocrine
NEUROPHARMACOLOGICAL PROFILE OF NONPEPTIDE NEUROTENSIN ANTAGONISTS
Fundamental and clinical pharmacology
A COMPUTER MODELING POSTULATED MECHANISM FOR ANGIOTENSIN-II RECEPTOR ACTIVATION
Journal of protein chemistry
NEW POTENT AND SELECTIVE NONPEPTIDE ANTAGONISTS OF NEUROTENSIN RECEPTORS
European journal of medicinal chemistry
HETEROGENEITY OF NEUROKININ, BINDING-SITES IN PORCINE RESPIRATORY-TRACT
Peptides
NONPEPTIDE ANGIOTENSIN-II RECEPTOR ANTAGO NISTS
Yuki Gosei Kagaku Kyokaishi
2 CLASSES OF STRUCTURALLY DIFFERENT ANTAGONISTS DISPLAY SIMILAR SPECIES PREFERENCE FOR THE HUMAN TACHYKININ NEUROKININ(3) RECEPTOR
Molecular pharmacology
NOVEL ANGIOTENSIN-II RECEPTOR ANTAGONISTS - DESIGN, SYNTHESIS, AND IN-VITRO EVALUATION OF DIBENZO[A,D]CYCLOHEPTENE AND DIBENZO[B,F]OXEPIN DERIVATIVES - SEARCHING FOR BIOISOSTERES OF BIPHENYLYLTETRAZOLE USING A3-DIMENSIONAL SEARCH TECHNIQUE
Journal of medicinal chemistry
HUMAN INTERNAL MAMMARY ARTERY RESPONSES TO NONPEPTIDE VASOPRESSIN ANTAGONISTS
Clinical and experimental pharmacology and physiology
THE MARKED DISPARITY BETWEEN THE SIZES OF ANGIOTENSIN TYPE-2 RECEPTORS FROM DIFFERENT TISSUES IS RELATED TO DIFFERENT DEGREES OF N-GLYCOSYLATION
Molecular pharmacology
PHARMACOLOGICAL PROFILE OF FK480, A NOVEL CHOLECYSTOKININ TYPE-A RECEPTOR ANTAGONIST - COMPARISON TO LOXIGLUMIDE
The Journal of pharmacology and experimental therapeutics
MOLECULAR-CLONING OF THE CANINE ANGIOTENSIN-II RECEPTOR - AN AT1-LIKERECEPTOR WITH REDUCED AFFINITY FOR DUP753
FEBS letters
COMPARISON OF TACHYKININ NK(1) RECEPTORS IN HUMAN IM9 AND U373-MG CELLS, USING ANTAGONIST (FK888, (PLUS-OR-MINUS)-CP-96,345, AND RP-67580) BINDING
European journal of pharmacology
CORTICOTROPIN-RELEASING FACTOR RECEPTORS IN HUMAN SMALL-CELL LUNG-CARCINOMA CELLS - RADIOLIGAND BINDING, 2ND-MESSENGER, AND NORTHERN BLOT ANALYSIS DATA
Endocrinology
EFFECTS OF RP-67580, A TACHYKININ NK1 RECEPTOR ANTAGONIST, ON A PRIMARY AFFERENT-EVOKED RESPONSE OF VENTRAL ROOTS IN THE NEONATAL RAT SPINAL-CORD
British Journal of Pharmacology
MUTATIONS IN TRANSMEMBRANE SEGMENT-VII OF THE AT(1) RECEPTOR DIFFERENTIATE BETWEEN CLOSELY-RELATED INSURMOUNTABLE AND COMPETITIVE ANGIOTENSIN ANTAGONISTS
British Journal of Pharmacology
EFFECT OF THE TACHYKININ NK1 RECEPTOR ANTAGONISTS, RP-67580 AND SR-140333, ON ELECTRICALLY-EVOKED SUBSTANCE-P RELEASE FROM RAT SPINAL-CORD
British Journal of Pharmacology
COMPARISON OF TACHYKININ NK1 AND NK2 RECEPTORS IN THE CIRCULAR MUSCLEOF THE GUINEA-PIG ILEUM AND PROXIMAL COLON
British Journal of Pharmacology
COMPARATIVE PHARMACOLOGY OF RECOMBINANT RAT AT(1A), AT(1B) AND HUMAN AT(1) RECEPTORS EXPRESSED BY TRANSFECTED COS-M6 CELLS
British Journal of Pharmacology
NONSPECIFIC ACTIONS OF THE NONPEPTIDE TACHYKININ RECEPTOR ANTAGONISTS, CP-96,345, RP-67580 AND SR-48968, ON NEUROTRANSMISSION
British Journal of Pharmacology
INHIBITORY EFFECT OF THE NONPEPTIDE ANGIOTENSIN-II RECEPTOR ANTAGONIST LOSARTAN AND ITS ACTIVE METABOLITE, E-3174, ON CAMP-PHOSPHODIESTERASE - ADDITIONAL ACTION OF THE ANTAGONISTS
Biochemical pharmacology
ESTABLISHMENT OF A CELLULAR-ASSAY SYSTEM FOR G-PROTEIN-LINKED RECEPTORS - COUPLING OF HUMAN NK2 AND 5-HT(2) RECEPTORS TO PHOSPHOLIPASE-C ACTIVATES A LUCIFERASE REPORTER GENE
Receptors & channels
DIFFERENTIAL EFFECT OF DITHIOTHREITOL AND DUP-753 ON ANGIOTENSIN-II RECEPTOR SUBTYPES IN BOVINE CEREBELLAR CORTEX
Peptides
ANGIOTENSIN-II RECEPTOR BLOCKADE - AN INNOVATIVE APPROACH TO CARDIOVASCULAR PHARMACOTHERAPY
Journal of clinical pharmacology
ANGIOTENSIN-II RECEPTORS AND ANGIOTENSIN-II RECEPTOR ANTAGONISTS
Pharmacological reviews
DIFFERENCES IN THE EFFECTS OF TACHYKININ NK(1) RECEPTOR ANTAGONISTS -NEURONAL VERSUS SMOOTH-MUSCLE TISSUES
European journal of pharmacology
A NONPEPTIDE NK1-RECEPTOR ANTAGONIST, RP-67580, INHIBITS NEUROGENIC INFLAMMATION POSTSYNAPTICALLY
British Journal of Pharmacology
ANGIOTENSIN RECEPTOR-SITES IN RENAL VASCULATURE OF RATS DEVELOPING GENETIC-HYPERTENSION
The American journal of physiology
ANGIOTENSIN-II TYPE-2 RECEPTOR-MODULATED CHANGES IN POTASSIUM CURRENTS IN CULTURED NEURONS
The American journal of physiology