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Recent advances in feeding suppressing agents: potential therapeutic strategy for the treatment of obesity
EXPERT OPINION ON THERAPEUTIC PATENTS
Origins of the many NPY-family receptors in mammals
PEPTIDES
NPY in invertebrates: molecular answers to altered functions during evolution
PEPTIDES
Food intake inhibition and reduction in body weight gain in rats treated with GI264879A, a non-selective NPY-Y1 receptor antagonist
PEPTIDES
KO's and organisation of peptidergic feeding behavior mechanisms
NEUROSCIENCE AND BIOBEHAVIORAL REVIEWS
Neuropeptide Y stimulates food consumption through multiple receptors in goldfish
PHYSIOLOGY & BEHAVIOR
Leptin activates anorexigenic POMC neurons through a neural network in thearcuate nucleus
NATURE
Increased expression of the neuropeptide Y receptor Y-1 gene in the medialamygdala of transgenic mice induced by long-term treatment with progesterone or allopregnanolone
JOURNAL OF NEUROCHEMISTRY
Neuropeptide YY5 receptor antagonist CGP71683A: the effects on food intakeand anxiety-related behavior in the rat
EUROPEAN JOURNAL OF PHARMACOLOGY
The role of NPY in metabolic homeostasis: implications for obesity therapy
EXPERT OPINION ON INVESTIGATIONAL DRUGS
Cloning and transcriptional expression of a leucokinin-like peptide receptor from the Southern cattle tick, Boophilus microplus (Acari : Ixodidae)
INSECT MOLECULAR BIOLOGY
Molecular manipulation of G-protein-coupled receptors: A new avenue into drug discovery
CURRENT MEDICINAL CHEMISTRY
Characterisation of G-protein-coupled receptors by antibodies
CURRENT MEDICINAL CHEMISTRY
Neuropeptide Y-Y1 receptor antisense oligodeoxynucleotide increases the infarct volume after middle cerebral artery occlusion ln rats
NEUROSCIENCE
[D-Trp(34)] neuropeptide Y is a potent and selective neuropeptide YY5 receptor agonist with dramatic effects on food intake
PEPTIDES
2-36[K-4,RYYSA(19-23)]PP a novel Y5-receptor preferring ligand with strongstimulatory effect on food intake
REGULATORY PEPTIDES
Behavioural neuroscience and child psychopathology: Insights from model systems
JOURNAL OF CHILD PSYCHOLOGY AND PSYCHIATRY AND ALLIED DISCIPLINES
Pharmacological characterization of the cloned neuropeptide Y y(6) receptor
EUROPEAN JOURNAL OF PHARMACOLOGY
Food intake regulation in rodents: Y-5 or Y1NPY receptors or both?
CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY
Molecular dynamics of NPYY1 receptor activation
BIOORGANIC & MEDICINAL CHEMISTRY
Neuropeptide Y receptor alterations in the hypothalamus of lactating rats
PEPTIDES
Differential regulation of mRNAs for neuropeptide Y and its receptor subtypes in widespread areas of the rat limbic system during kindling epileptogenesis
MOLECULAR BRAIN RESEARCH
The corticotropin-release inhibitory factor hypothesis: A review of the evidence for the existence of inhibitory as well as stimulatory hypophysiotropic regulation of adrenocorticotropin secretion and biosynthesis
ENDOCRINE REVIEWS
Antisense mRNA for NPY-Y-1 receptor in the medial preoptic area increases prolactin secretion
BRAZILIAN JOURNAL OF MEDICAL AND BIOLOGICAL RESEARCH
Differential modulation of agonist potency and receptor coupling by mutations of Ser388Tyr and Thr389Pro at the junction of transmembrane domain VI and the third extracellular loop of human M-1 muscarinic acetylcholine receptors
MOLECULAR PHARMACOLOGY
Phencyclidine and dizocilpine modulate dopamine release from rat nucleus accumbens via sigma receptors
EUROPEAN JOURNAL OF PHARMACOLOGY
Neuropeptide Y-induced contraction is mediated by neuropeptide YY2 and Y-4receptors in the rat colon
EUROPEAN JOURNAL OF PHARMACOLOGY
Amygdalar neuropeptide Y Y-1 receptors mediate the anxiolytic-like actionsof neuropeptide Y in the social interaction test
EUROPEAN JOURNAL OF PHARMACOLOGY
Gi-protein alpha-subunit mRNA antisense oligonucleotide inhibition of Gi-coupled receptor contractile activity in the epididymis of the guinea-pig
BRITISH JOURNAL OF PHARMACOLOGY
An immunohistochemical marker for Wallerian degeneration of fibers in the central and peripheral nervous system
BRAIN RESEARCH
Sequence and tissue distribution of a novel G-protein-coupled receptor expressed prominently in human placenta
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS
Decreased responsiveness of vascular postjunctional alpha(1)-, alpha(2)-adrenoceptors and neuropeptide Y1 receptors in rats with heart failure
ACTA PHYSIOLOGICA SCANDINAVICA
MOLECULAR MODELING OF THE NPY BINDING-SITE ON THE Y-1 RECEPTOR
JOURNAL OF MOLECULAR MODELING
MICROSATELLITE MARKER CONTENT MAPPING OF 12 CANDIDATE GENES FOR OBESITY - ASSEMBLY OF 7 OBESITY SCREENING PANELS FOR AUTOMATED GENOTYPING
PCR methods and applications
DOWN-REGULATED NPY RECEPTOR SUBTYPE-5 MESSENGER-RNA EXPRESSION IN GENETICALLY-OBESE MOUSE-BRAIN
NeuroReport
THE MURINE Y-1 RECEPTOR 5' UPSTREAM SEQUENCE DIRECTS CELL-SPECIFIC AND DEVELOPMENTALLY-REGULATED LACZ EXPRESSION IN TRANSGENIC MICE CNS
European journal of neuroscience
NEUROPEPTIDE-Y INHIBITS CILIARY BEAT FREQUENCY IN HUMAN CILIATED CELLS VIA NPKC, INDEPENDENTLY OF PKA
American journal of physiology. Cell physiology
REGIONAL DISTRIBUTION OF NEUROPEPTIDE-Y Y2 RECEPTOR MESSENGER-RNA IN THE HUMAN POST-MORTEM BRAIN
Neuroscience
THE LIGAND-BINDING SITE OF NPY AT THE RAT Y-1 RECEPTOR INVESTIGATED BY SITE-DIRECTED MUTAGENESIS AND MOLECULAR MODELING
Molecular and cellular endocrinology
ALTERATIONS IN NEUROPEPTIDE-Y AND Y1 RECEPTOR MESSENGER-RNA EXPRESSION IN BRAINS FROM AN ANIMAL-MODEL OF DEPRESSION - REGION-SPECIFIC ADAPTATION AFTER FLUOXETINE TREATMENT
Molecular brain research
MOLECULAR-BIOLOGY AND PHARMACOLOGY OF MULTIPLE NPY Y-5 RECEPTOR SPECIES HOMOLOGS
Regulatory peptides
SUPPRESSION OF SENSORY-C FIBER-MEDIATED CONTRACTIONS BY NEUROPEPTIDE-Y Y1-RECEPTORS IN THE GUINEA-PIG BRONCHI
Regulatory peptides
NPY-INDUCED FEEDING INVOLVES THE ACTION OF A Y1-LIKE RECEPTOR IN RODENTS
Regulatory peptides
MULTIPLE RECEPTORS FOR THE PANCREATIC-POLYPEPTIDE (PP-FOLD) FAMILY - PHYSIOLOGICAL IMPLICATIONS
Proceedings of the Society for Experimental Biology and Medicine
HUMAN PLACENTA AND FETAL MEMBRANES CONTAIN PEPTIDE YY1-36 AND PEPTIDEYY3-36
Journal of Endocrinology
NEUROPEPTIDE-Y Y-1 RECEPTORS IN VASCULAR PHARMACOLOGY
European journal of pharmacology
GR231118 (1229U91) AND OTHER ANALOGS OF THE C-TERMINUS OF NEUROPEPTIDE-Y ARE POTENT NEUROPEPTIDE-Y Y-1 RECEPTOR ANTAGONISTS AND NEUROPEPTIDE-Y Y-4 RECEPTOR AGONISTS
European journal of pharmacology
CONCOMITANT REGULATION OF CA2-CELLS( MOBILIZATION AND G(13) EXPRESSION IN HUMAN ERYTHROLEUKEMIA)
European journal of pharmacology
Pharmacological profile of the rat intestinal crypt peptide YY receptor vs. the recombinant rat Y5 receptor
EUROPEAN JOURNAL OF PHARMACOLOGY
CLONING AND CHARACTERIZATION OF A NEW SUBTYPE OF THYROTROPIN-RELEASING-HORMONE RECEPTORS
Biochemical and biophysical research communications (Print)
LOCALIZATION OF NEUROPEPTIDE-Y Y-1 RECEPTOR MESSENGER-RNA HUMAN TOOTH-PULP
Archives of oral biology
MOLECULAR APPROACHES TO THE DISCOVERY OF NEW TREATMENTS FOR OBESITY
CURRENT OPINION IN CHEMICAL BIOLOGY
ALPHA-HELICAL CRF9-41 PREVENTS ANXIOGENIC-LIKE EFFECT OF NPY Y-1 RECEPTOR ANTAGONIST BIBP3226 IN RATS
NeuroReport
NPY OPPOSES PACAP PHASE-SHIFTS VIA RECEPTORS DIFFERENT FROM THOSE INVOLVED IN NPY PHASE-SHIFTS
NeuroReport
LOCALIZATION OF NEUROPEPTIDE-Y Y1 MESSENGER-RNA IN THE HUMAN BRAIN - ABUNDANT EXPRESSION IN CEREBRAL-CORTEX AND STRIATUM
European journal of neuroscience
CDNA CLONING AND TISSUE-SPECIFIC GENE-EXPRESSION OF OVINE LEPTIN, NPY-Y1 RECEPTOR, AND NPY-Y2 RECEPTOR
Domestic animal endocrinology
MODES OF PEPTIDE BINDING IN G-PROTEIN-COUPLED RECEPTORS
Neurochemical research
ANALYSIS OF NPY RECEPTOR SUBTYPES IN THE HUMAN FRONTAL-CORTEX REVEALSABUNDANT Y-1 MESSENGER-RNA AND BINDING-SITES
Peptides
DISTRIBUTION OF THE NEUROPEPTIDE-Y Y2 RECEPTOR MESSENGER-RNA IN RAT CENTRAL-NERVOUS-SYSTEM
Molecular brain research
PHARMACOLOGICAL CHARACTERIZATION AND SELECTIVITY OF THE NPY ANTAGONIST GR231118 (1229U91) FOR DIFFERENT NPY RECEPTORS
Regulatory peptides
CHARACTERIZATION OF THE RECEPTOR RESPONSE FOR THE NEUROPEPTIDE Y-EVOKED SUPPRESSION OF PARASYMPATHETICALLY-MEDIATED CONTRACTIONS IN THE GUINEA-PIG TRACHEA
Regulatory peptides
EVIDENCE FOR A ROLE OF THE GUT HORMONE PYY IN THE REGULATION OF INTESTINAL FATTY-ACID-BINDING PROTEIN TRANSCRIPTS IN DIFFERENTIATED SUBPOPULATIONS OF INTESTINAL EPITHELIAL-CELL HYBRIDS
The Journal of biological chemistry
NEUROPEPTIDE-Y Y-1 RECEPTOR BLOCKADE DOES NOT ALTER ADRENERGIC-NERVE RESPONSES OF THE RAT TAIL ARTERY
European journal of pharmacology
THE RABBIT ILEUM - A SENSITIVE AND SELECTIVE PREPARATION FOR THE NEUROPEPTIDE-Y Y-5 RECEPTOR
European journal of pharmacology
IDENTIFICATION OF MULTIPLE NEUROPEPTIDE-Y RECEPTOR SUBTYPES IN THE HUMAN FRONTAL-CORTEX
European journal of pharmacology
NONCOMPETITIVE BINDING OF THE NONPEPTIDE ANTAGONIST BIBP3226 TO RAT FOREBRAIN NEUROPEPTIDE Y-1 RECEPTORS
European journal of pharmacology
MONITORING OF ANTISENSE EFFECTS OF OLIGONUCLEOTIDES TARGETED TO THE NEUROPEPTIDE-Y Y-1 RECEPTOR GENE
European journal of pharmacology
NEUROPEPTIDE-Y Y-1 RECEPTORS ARE INVOLVED IN THE VASOCONSTRICTION CAUSED BY HUMAN SYMPATHETIC-NERVE STIMULATION
European journal of pharmacology
THE DOG SAPHENOUS-VEIN - A SENSITIVE AND SELECTIVE PREPARATION FOR THE Y-2 RECEPTOR OF NEUROPEPTIDE-Y
European journal of pharmacology
GW1229, A NOVEL NEUROPEPTIDE-Y Y-1 RECEPTOR ANTAGONIST, INHIBITS THE VASOCONSTRICTOR EFFECT OF NEUROPEPTIDE-Y IN THE HAMSTER MICROCIRCULATION
European journal of pharmacology
DISTRIBUTION OF [LEU(31),PRO(34)]NPY-SENSITIVE, BIBP3226-INSENSITIVE [I-125] PYY(3-36) BINDING-SITES IN RAT-BRAIN - POSSIBLE RELATIONSHIP TO Y-5 NPY RECEPTORS
Brain research
REDUCTION OF NEUROPEPTIDE-Y BINDING-SITES IN THE RAT HIPPOCAMPUS AFTER ELECTROCONVULSIVE STIMULATIONS
Brain research
GENE-EXPRESSION OF NEUROPEPTIDE-Y AND NEUROPEPTIDE-Y1 RECEPTOR IN RELATION TO PROTOONCOGENE TYROSINE KINASE-A, NERVE-GROWTH-FACTOR LOW-AFFINITY-RECEPTOR AND THE TRANSCRIPTION FACTOR N-MYC IN HUMAN NEUROBLASTOMAS
International journal of oncology
CELLULAR-LOCALIZATION OF NEUROPEPTIDE-Y RECEPTORS IN THE RAT HIPPOCAMPUS - LONG-TERM EFFECTS OF LIMBIC SEIZURES
NeuroReport
AUTORADIOGRAPHIC DISTRIBUTION OF [I-125] [LEU(31), PRO(34)]PYY AND [I-125] PYY3-36 BINDING-SITES IN THE RAT-BRAIN EVALUATED WITH 2 NEWLY DEVELOPED Y-1 AND Y-2 RECEPTOR RADIOLIGANDS
Synapse
MULTIPLE NPY RECEPTORS COEXIST IN PRESYNAPTIC AND POSTSYNAPTIC SITES - INHIBITION OF GABA RELEASE IN ISOLATED SELF-INNERVATING SCN NEURONS
The Journal of neuroscience
SYNTHESIS, STRUCTURE, AND ANTAGONISTIC PROPERTIES OF DES-ASN(29)[D-TRP(28,32)]NPY(27-36)
Peptides
LIGAND-BINDING AND FUNCTIONAL-EFFECTS OF SYSTEMATIC DOUBLE D-AMINO-ACID RESIDUE SUBSTITUTED NEUROPEPTIDE-Y ANALOGS ON Y1 AND Y2 RECEPTOR TYPES
Regulatory peptides
MOLECULAR CHARACTERIZATION OF A 2ND MOUSE PANCREATIC-POLYPEPTIDE RECEPTOR AND ITS INACTIVATED HUMAN HOMOLOG
The Journal of biological chemistry
HIGH-LEVELS OF SPECIFIC NEUROPEPTIDE Y PANCREATIC POLYPEPTIDE RECEPTORS IN THE RAT HYPOTHALAMUS AND BRAIN-STEM/
European journal of pharmacology
DIFFERENCES IN CATION SENSITIVITY OF LIGAND-BINDING TO Y-1 AND Y-2 SUBTYPE OF NEUROPEPTIDE-Y RECEPTOR OF RAT-BRAIN
European journal of pharmacology
ANXIOGENIC-LIKE EFFECT OF THE NEUROPEPTIDE-Y Y-1 RECEPTOR ANTAGONIST BIBP3226 - ANTAGONISM WITH DIAZEPAM
European journal of pharmacology
CYTOSKELETAL INHIBITORS IMPAIR CA2-Y AND OTHER G(I)-COUPLED RECEPTORS( ELEVATIONS VIA NEUROPEPTIDE)
European journal of pharmacology
SR 120107A ANTAGONIZES NEUROPEPTIDE-Y Y-1 RECEPTOR-MEDIATED SYMPATHETIC VASOCONSTRICTION IN PIGS IN-VIVO
European journal of pharmacology
ANTINOCICEPTIVE EFFECTS OF NEUROPEPTIDE-Y AND RELATED PEPTIDES IN MICE
Brain research
PEPTIDES AS NEUROTRANSMITTERS IN VASCULAR AUTONOMIC NEURONS
Clinical and experimental pharmacology and physiology
EXPRESSION OF THE NEUROPEPTIDE-Y Y-1 RECEPTOR IN HUMAN EMBRYONIC KIDNEY-293-CELLS - LIGAND-BINDING CHARACTERISTICS, IN-SITU HYBRIDIZATION AND RECEPTOR AUTORADIOGRAPHY
Molecular brain research
NEUROPEPTIDE Y-2-TYPE RECEPTOR-MEDIATED ACTIVATION OF LARGE-CONDUCTANCE CA2-SENSITIVE K+ CHANNELS IN A HUMAN NEUROBLASTOMA CELL-LINE()
Pflugers Archiv
NEUROPEPTIDE-Y RECEPTOR SUBTYPES
Life sciences
NEUROPEPTIDE-Y IS A VASOCONSTRICTOR AND ADRENERGIC MODULATOR IN THE HAMSTER MICROCIRCULATION BY ACTING ON NEUROPEPTIDE Y-1 AND Y-2 RECEPTORS
European journal of pharmacology
NEUROPEPTIDE-Y ACCOUNTS FOR SYMPATHETIC VASOCONSTRICTION IN GUINEA-PIG VENA-CAVA - EVIDENCE USING BIBP-3226 AND BIBP-3435
European journal of pharmacology
APPARENT AFFINITY AND POTENCY OF BIBP3226, A NONPEPTIDE NEUROPEPTIDE-Y RECEPTOR ANTAGONIST, ON PURPORTED NEUROPEPTIDE-Y Y-1, Y-2 AND Y-3 RECEPTORS
European journal of pharmacology
ROLES OF PEPTIDES AND OTHER SUBSTANCES IN COTRANSMISSION FROM VASCULAR AUTONOMIC AND SENSORY NEURONS
Canadian journal of physiology and pharmacology
REGIONAL INVOLVEMENT OF AN ENDOTHELIUM-DERIVED CONTRACTILE FACTOR IN THE VASOACTIVE ACTIONS OF NEUROPEPTIDE-Y IN BOVINE ISOLATED RETINAL ARTERIES
British Journal of Pharmacology
INCREASED VASOPRESSOR ACTIONS OF INTRAVENTRICULAR NEUROPEPTIDE Y-(13-36) IN SPONTANEOUSLY HYPERTENSIVE VERSUS NORMOTENSIVE WISTAR-KYOTO RATS - POSSIBLE RELATIONSHIP TO INCREASES IN Y-2 RECEPTOR-BINDING IN THE NUCLEUS-TRACTUS-SOLITARIUS
Brain research
REGULATION OF PROOPIOMELANOCORTIN GENE-EXPRESSION BY NEUROPEPTIDE-Y IN THE RAT ARCUATE NUCLEUS
Brain research
MODULATION OF VASCULAR CONTRACTILE RESPONSES TO ALPHA(1)-ADRENERGIC AND ALPHA(2)-ADRENERGIC AND NEUROPEPTIDE-Y RECEPTOR STIMULATION IN RATSWITH ISCHEMIC HEART-FAILURE
Acta Physiologica Scandinavica
RECEPTORS FOR GUT REGULATORY PEPTIDES
Bailliere's clinical endocrinology and metabolism
[PRO(34)]PEPTIDE YY IS A Y-1-SELECTIVE AGONIST AT PEPTIDE YY NEUROPEPTIDE-Y RECEPTORS
European journal of pharmacology. Molecular pharmacology section
A NOVEL NEUROPEPTIDE-Y ANALOG, N-ACETYL[LEU(28),LEU(31)]NEUROPEPTIDE Y-(24-36), WITH FUNCTIONAL SPECIFICITY FOR THE PRESYNAPTIC (Y-2) RECEPTOR
European journal of pharmacology. Molecular pharmacology section