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Synthesis and in-vitro evaluation of novel low molecular weight thiocarbamates as inhibitors of human leukocyte elastase
JOURNAL OF ENZYME INHIBITION
Covalent binding of acrylonitrile to specific rat liver glutathione S-transferases in vivo
CHEMICAL RESEARCH IN TOXICOLOGY
Crystal structure of isopentenyl diphosphate : dimethylallyl diphosphate isomerase
EMBO JOURNAL
Methylidene-imidazolone (MIO) from histidine and phenylalanine ammonia-lyase
ADVANCES IN PROTEIN CHEMISTRY, VOL 58
Synthesis of enantiomerically enriched beta,gamma-unsaturated-alpha-amino acids
TETRAHEDRON
Stereocontrolled synthesis of quaternary beta,gamma-unsaturated amino acids: chain extension of D- and L-alpha-(2-tributylstannyl)vinyl amino acids
TETRAHEDRON
Transporters in African trypanosomes: role in drug action and resistance
INTERNATIONAL JOURNAL FOR PARASITOLOGY
Polyamine depletion in human melanoma cells leads to G(1) arrest associated with induction of p21(,)(WAF1/CIP1/SDI1) changes in the expression of p21-regulated genes, and a senescence-like phenotype
CANCER RESEARCH
Inhibition of tissue-bound semicarbazide-sensitive amine oxidase by two haloamines, 2-bromoethylamine and 3-bromopropylamine
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS
The angiogenesis inhibitor SU5416 has long-lasting effects on vascular endothelial growth factor receptor phosphorylation and function
CLINICAL CANCER RESEARCH
Phase III randomized study of postradiotherapy chemotherapy with alpha-difluoromethylornithine-procarbazin N-(2-chloroethyl)-N '-cyclohexyl-N-nitrosurea, vincristine (DFMO-PCV) versus PCV for glioblastoma multiforme
CLINICAL CANCER RESEARCH
Protective effect of melatonin against the 1-methyl-4-phenylpyridinium-induced inhibition of Complex I of the mitochondrial respiratory chain
JOURNAL OF PINEAL RESEARCH
Long chain diamines inhibit growth of C6 glioma cells according to their hydrophobicity. An in vitro and molecular modeling study
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY
The endogenous amine 1-methyl-1,2,3,4-tetrahydroisoquinoline prevents the inhibition of complex I of the respiratory chain produced by MPP+
JOURNAL OF NEUROCHEMISTRY
Characterization of arginine decarboxylase in rat brain and liver: Distinction from ornithine decarboxylase
JOURNAL OF NEUROCHEMISTRY
Polyamines, and effects from reducing their synthesis during egg development in the yellow fever mosquito, Aedes aegypti
JOURNAL OF INSECT PHYSIOLOGY
Refinement of the pressure assay for milk urea nitrogen
JOURNAL OF DAIRY SCIENCE
Effects of conditional overexpression of spermidine/spermine N-1-acetyltransferase on polyamine pool dynamics, cell growth, and sensitivity to polyamine analogs
JOURNAL OF BIOLOGICAL CHEMISTRY
Asymmetric preference of serine proteases toward phosphonate and phosphinate esters
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS
The role of biotransformation in dietary (anti)carcinogenesis
MUTATION RESEARCH-GENETIC TOXICOLOGY AND ENVIRONMENTAL MUTAGENESIS
Ligand and active-site dependent P-O versus C-O bond cleavage in organophosphorus adducts of serine hydrolases
PHOSPHORUS SULFUR AND SILICON AND THE RELATED ELEMENTS
Isolation and characterization of the product of inactivation of gamma-aminobutyric acid aminotransferase by gabaculine
BIOORGANIC & MEDICINAL CHEMISTRY
Analysis of CD39/ATP diphosphohydrolase (ATPDase) expression in endothelial cells, platelets and leukocytes
THROMBOSIS AND HAEMOSTASIS
Interaction of 3-alkylpyridinium polymers from the sea sponge Reniera sarai with insect acetylcholinesterase
JOURNAL OF PROTEIN CHEMISTRY
The stereoselectivity of inhibition of rat liver mitochondrial MAO-A and MAO-B by the enantiomers of 2-phenylpropylamine and their derivatives
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Cloning and kinetic characterization of the Trypanosoma cruzi S-adenosylmethionine decarboxylase
MOLECULAR AND BIOCHEMICAL PARASITOLOGY
Arginine decarboxylase in Trypanosoma cruzi, characteristics and kinetic properties
CELLULAR AND MOLECULAR BIOLOGY
Role of cysteine-82 in the catalytic mechanism of human S-adenosylmethionine decarboxylase
BIOCHEMISTRY
Irreversible inhibition of plasma membrane (Ca2++Mg2+)-ATPase and Ca2+ transport by 4-OH-2,3-trans-nonenal
ARCHIVES OF BIOCHEMISTRY AND BIOPHYSICS
SYNTHESIS AND KINETIC-STUDIES OF AN AMIDINE-CONTAINING PHOSPHONOFLUORIDATE - A NOVEL POTENT INHIBITOR OF TRYPSIN-LIKE ENZYMES
Bioorganic & medicinal chemistry
SYNTHESIS AND PROTEINASE INHIBITORY PROPERTIES OF DIPHENYL PHOSPHONATE ANALOGS OF ASPARTIC AND GLUTAMIC ACIDS
Bioorganic & medicinal chemistry letters
INHIBITION OF GLUTATHIONE-S-TRANSFERASE ACTIVITY BY THE QUINOID METABOLITES OF EQUINE ESTROGENS
Chemical research in toxicology
STRATEGIES TO CHARACTERIZE THE MECHANISMS OF ACTION AND THE ACTIVE-SITES OF GLUTATHIONE S-TRANSFERASES - A REVIEW
Drug metabolism reviews
DIFFERENTIAL EFFECT ON POLYAMINE METABOLISM IN MITOGEN-ACTIVATED AND SUPERANTIGEN-ACTIVATED HUMAN T-CELLS
Biochimica et biophysica acta (G). General subjects
EPOXYALKANOYLS AS NOVEL ACE-INHIBITORS
Archives of pharmacal research
EFFECTS OF DEMO ON GLIOMA CELL-PROLIFERATION, MIGRATION AND INVASION IN-VITRO
Journal of neuro-oncology
MGBG analogues as potent inhibitors of S-adenosylmethionine decarboxylase of Onchocerca volvulus
MOLECULAR AND BIOCHEMICAL PARASITOLOGY
METABOLISM-BASED INACTIVATION OF PENILE NITRIC-OXIDE SYNTHASE ACTIVITY BY GUANABENZ
Drug metabolism and disposition
IRREVERSIBLE INHIBITION OF THE HIV-1 PROTEASE - A THEORETICAL-STUDY
International journal of quantum chemistry
KINETIC-STUDY OF IRREVERSIBLE INHIBITION OF AN ENZYME CONSUMED IN THEREACTION IT CATALYZES - APPLICATION TO THE INHIBITION OF THE PUROMYCIN REACTION BY SPIRAMYCIN AND HYDROXYLAMINE
Journal of enzyme inhibition
COMBINED ACTION OF INHIBITORS OF S-ADENOSYLMETHIONINE DECARBOXYLASE WITH AN ANTIMALARIAL DRUG, CHLOROQUINE, ON PLASMODIUM-FALCIPARUM
The Journal of eukaryotic microbiology
THE ESSENTIAL TRYPTOPHAN RESIDUES OF PIG-KIDNEY AMINOACYLASE
Biochemistry and molecular biology international
INHIBITION OF CAMEL LENS ZETA-CRYSTALLIN NADPH-QUINONE OXIDOREDUCTASEACTIVITY BY CHLORANILIC ACID/
Biochemistry and molecular biology international
STRUCTURE, CATALYTIC MECHANISM, AND EVOLUTION OF THE GLUTATHIONE TRANSFERASES
Chemical research in toxicology
CHEMICAL AND QUANTUM-MECHANICAL STUDIES OF THE FREE-RADICAL C-C BOND FORMATION IN THE LIPOXYGENASE-CATALYZED DIMERIZATION OF OCTADECA-9,12-DIYNOIC ACID
Free radical biology & medicine
INFLUENCE OF NONNUTRIENT PLANT-COMPONENTS ON BIOTRANSFORMATION ENZYMES
Biomedicine & pharmacotherapy
ISOPENTENYL DIPHOSPHATE ISOMERASE - A CORE ENZYME IN ISOPRENOID BIOSYNTHESIS - A REVIEW OF ITS BIOCHEMISTRY AND FUNCTION
Natural product reports
PEPTIDYL INVERSE ESTERS OF P-METHOXYBENZOIC ACID - A NOVEL CLASS OF POTENT INACTIVATOR OF THE SERINE PROTEASES
Biochemical journal
SIGNAL ANALYSIS OF FIBEROPTIC BIOSENSOR FOR THE DETECTION OF ORGANOPHOSPHORUS COMPOUNDS IN THE CONTAMINATED WATER
The Korean journal of chemical engineering
KINETICS OF IRREVERSIBLE INHIBITION OF YEAST ALCOHOL-DEHYDROGENASE DURING MODIFICATION BY 4,4'-DITHIODIPYRIDINE
International journal of biological macromolecules
A CONVENIENT SYNTHESIS OF L-ALPHA-VINYLGLYCINE FROM D-MANNITOL
Synthesis
CONTROL OF PLANT-DISEASE BY PERTURBATION OF FUNGAL POLYAMINE METABOLISM
Physiologia Plantarum
INTERFERENCE WITH DNA METHYLTRANSFERASE ACTIVITY AND GENOME METHYLATION DURING F9 TERATOCARCINOMA STEM-CELL DIFFERENTIATION-INDUCED BY POLYAMINE DEPLETION
The Journal of biological chemistry
CHARACTERIZATION OF SIMIAN MALARIAL PARASITE (PLASMODIUM KNOWLESI)-INDUCED PUTRESCINE TRANSPORT IN RHESUS-MONKEY ERYTHROCYTES - A NOVEL PUTRESCINE CONJUGATE ARRESTS IN-VITRO GROWTH OF SIMIAN MALARIAL PARASITE (PLASMODIUM-KNOWLESI) AND CURES MULTIDRUG-RESISTANT MURINE MALARIA (PLASMODIUM-YOELII) INFECTION IN-VIVO
The Journal of biological chemistry
MODULATION OF GLUTATHIONE CONJUGATION IN-VIVO - HOW TO DECREASE GLUTATHIONE CONJUGATION IN-VIVO OR IN INTACT CELLULAR-SYSTEMS IN-VITRO
Chemico-biological interactions
TREATMENT WITH INHIBITORS OF POLYAMINE BIOSYNTHESIS, WHICH SELECTIVELY LOWER INTRACELLULAR SPERMINE, DOES NOT AFFECT THE ACTIVITY OF ALKYLATING-AGENTS BUT ANTAGONIZES THE CYTOTOXICITY OF DNA TOPOISOMERASE-II INHIBITORS
British Journal of Cancer
MECHANISM OF INHIBITION OF E(1)-E(2) ATPASES BY MELITTIN
Biochemistry
SANGUINARINE AND CHELERYTHRINE AS INHIBITORS OF AROMATIC AMINO-ACID DECARBOXYLASE
Journal of enzyme inhibition
FACILE ANALYSIS OF RIBONUCLEOTIDES IN D,L-ALPHA-DIFLUOROMETHYLORNITHINE-TREATED MOUSE LYMPHOID-CELLS BY HIGH-PERFORMANCE ANION-EXCHANGE COLUMN CHROMATOGRAPHY
Journal of chromatography B. Biomedical applications
KINETICS OF IRREVERSIBLE INHIBITION OF AMINOACYLASE BY MNP
Progress in Natural Science
ALPHA-VINYLLYSINE AND ALPHA-VINYLARGININE ARE TIME-DEPENDENT INHIBITORS OF THEIR COGNATE DECARBOXYLASES
Bioorganic & medicinal chemistry letters
INACTIVATION OF SERINE-PROTEASE, ALPHA-CHYMOTRYPSIN BY FLUORINATED PHENYLALANINE ANALOGS
Bioorganic & medicinal chemistry letters
KINETICS OF MODIFICATION OF THE MITOCHONDRIAL SUCCINATE-UBIQUINONE REDUCTASE BY 5,5'-DITHIOBIS-(2-NITRO-BENZOIC ACID)
Journal of protein chemistry
PANAGRELLUS REDIVIVUS ORNITHINE DECARBOXYLASE - STRUCTURE OF THE GENE, EXPRESSION IN ESCHERICHIA-COLI AND CHARACTERIZATION OF THE RECOMBINANT PROTEIN
Biochemical journal
A CONVENIENT SYNTHESIS OF L-ALPHA-VINYLGLYCINE FROM L-HOMOSERINE LACTONE
Synthesis
THE AF64A MODEL OF CHOLINERGIC HYPOFUNCTION - AN UPDATE
Life sciences
(CARBOXYALKYL)BENZYL PROPARGYL ETHERS AS SELECTIVE INHIBITORS OF LEUKOCYTE-TYPE 12-LIPOXYGENASES
Journal of medicinal chemistry
MECHANISTIC STUDIES ON THE INACTIVATION OF PAPAIN BY EPOXYSUCCINYL INHIBITORS
Journal of medicinal chemistry
PEROXYNITRITE FORMED BY SIMULTANEOUS GENERATION OF NITRIC-OXIDE AND SUPEROXIDE SELECTIVELY INHIBITS BOVINE AORTIC PROSTACYCLIN SYNTHASE
FEBS letters
INHIBITION OF RAT, MOUSE, AND HUMAN GLUTATHIONE-S-TRANSFERASE BY EUGENOL AND ITS OXIDATION-PRODUCTS
Chemico-biological interactions
CHARACTERISTICS OF INHIBITION OF BUTYRYL CHOLINESTERASE AND CARBOXYL ESTERASE HYDROLYSIS BY BETA,BETA-DIPHENYLETHYLPHOSPHONIC ACID FLUOROANHYDRIDE ESTERS
Biochemistry
MECHANISM OF LIPOXYGENASE INACTIVATION BY THE LINOLEIC-ACID ANALOG OCTADECA-9,12-DIYNOIC ACID
Biochemistry
EFFECTS OF CATIONIC DIAMIDINES ON POLYAMINE CONTENT AND UPTAKE ON LEISHMANIA-INFANTUM IN IN-VITRO CULTURES
Biochemical pharmacology
ANALYSIS OF MICHAELIS-MENTEN KINETICS IN THE PRESENCE OF IRREVERSIBLEINHIBITORS THAT REACT WITH THE SUBSTRATE
International journal of biochemistry & cell biology
INHIBITION OF POLYAMINE BIOSYNTHESIS IN FUNGI
Mycological research
A PHOTOCHEMICAL ROUTE TO VINYLGLYCINE AND A VINYLGLYCINE DIPEPTIDE
Liebigs Annalen
LOCALIZATION OF S-ADENOSYLMETHIONINE DECARBOXYLASE IN MURINE TISSUES BY IMMUNOHISTOCHEMISTRY
European journal of oral sciences
MODULATION OF QUINOL QUINONE-THIOETHER TOXICITY BY INTRAMOLECULAR DETOXICATION/
Drug metabolism reviews
STUDIES ON THE INHIBITING ACTION OF PCMB TO ARGINASE USING MICROCALORIMETRY
Gaodeng xuexiao huaxue xuebao
POLYAMINE DEPLETION-MEDIATED EFFECTS ON MURINE ODONTOGENESIS ARE DEPENDENT ON TOOTH DEVELOPMENTAL STAGE AND CULTURE CONDITIONS
The International journal of developmental biology
AF64A-INDUCED CYTOTOXICITY AND CHANGES IN CHOLINE-ACETYLTRANSFERASE ACTIVITY IN THE LA-N-2 NEUROBLASTOMA CELL-LINE ARE MODULATED BY CHOLINEAND HEMICHOLINIUM-3
Journal of neuroscience methods
METABOLISM AS A DETERMINANT OF SPECIES SUSCEPTIBILITY TO 2,3,5-(TRIGLUTATHION-S-YL)HYDROQUINONE-MEDIATED NEPHROTOXICITY - THE ROLE OF N-ACETYLATION AND N-DEACETYLATION
Drug metabolism and disposition
THERMOKINETIC STUDIES OF THE IRREVERSIBLE INHIBITION OF SINGLE-SUBSTRATE, ENZYME-CATALYZED REACTIONS
Thermochimica acta
ENANTIOENRICHED N-(2-CHLOROALKYL)-3-ACETOXYPIPERIDINES AS POTENTIAL CHOLINOTOXIC AGENTS - SYNTHESIS AND PRELIMINARY EVIDENCE FOR SPIROCYCLIC AZIRIDINIUM FORMATION
Tetrahedron
A SIMPLE DISPOSABLE POTENTIOMETRIC BIOSENSOR FOR PESTICIDES
Chemia Analityczna
FE(III)-LIPOXYGENASE CONVERTS ITS SUICIDE-TYPE INHIBITOR OCTADECA-9, 12-DIYNOIC ACID INTO 11-OXOOCTADECA-9,12-DIYNOIC ACID
Biochemistry
S-METHYL N,N-DIETHYLTHIOCARBAMATE SULFONE, A POTENTIAL METABOLITE OF DISULFIRAM AND POTENT INHIBITOR OF LOW K-M MITOCHONDRIAL ALDEHYDE DEHYDROGENASE
Biochemical pharmacology
REACTIVE OXYGEN SPECIES AND DNA-DAMAGE IN 2-BROMO-(GLUTATHIONE-S-YL) HYDROQUINONE-MEDIATED CYTOTOXICITY
Archives of biochemistry and biophysics
ALPHA-AMINOALKYLPHOSPHONATE DI(CHLOROPHENYL) ESTERS AS INHIBITORS OF SERINE PROTEASES
Journal of enzyme inhibition
ABNORMAL DNA-SYNTHESIS IN POLYAMINE DEFICIENT CELLS REVEALED BY BROMODEOXYURIDINE-FLOW CYTOMETRY TECHNIQUE
Cell proliferation
OXIDATION AND ACETYLATION AS DETERMINANTS OF 2-BROMOCYSTEIN-S-YLHYDROQUINONE-MEDIATED NEPHROTOXICITY
Chemical research in toxicology
A NEW S-ADENOSYLMETHIONINE DECARBOXYLASE FROM SOYBEAN AXES
Biochimica et biophysica acta (G). General subjects
MODIFICATION OF GLUTATHIONE-S-TRANSFERASE-3-3 MUTANTS WITH -(S-GLUTATHIONYL)-3,5,6-TRICHLORO-1,4-BENZOQUINONE - IDENTIFICATION OF THE C-TERMINAL TRYPTIC FRAGMENT AS PART OF THE H-SITE AND EVIDENCE THAT -(S-GLUTATHIONYL)-3,5,6-TRICHLORO-1,4-BENZOQUINONE IS NOT SPECIFIC FOR CYSTEINE LABELING
Biochemical journal
THE ROLE OF HYPUSINE DEPLETION IN CYTOSTASIS INDUCED BY S-ADENOSYL-L-METHIONINE DECARBOXYLASE INHIBITION - NEW EVIDENCE PROVIDED BY 1-METHYLSPERMIDINE AND 1,12-DIMETHYLSPERMINE
Biochemical journal
INHIBITION OF IMMEDIATE-EARLY-GENE INDUCTION IN RENAL MESANGIAL CELLSBY DEPLETION OF INTRACELLULAR POLYAMINES
Biochemical journal
POLYAMINE DEPRIVATION - A NEW TOOL IN CANCER-TREATMENT
Anticancer research
FLOW CYTOMETRIC ANALYSIS OF THE CELL-CYCLE IN POLYAMINE-DEPLETED CELLS
Cytometry
FINAL PHASE OF ENZYME-REACTIONS FOLLOWING A MICHAELIS-MENTEN MECHANISM IN WHICH THE FREE ENZYME AND OR THE ENZYME-SUBSTRATE COMPLEX AVE UNSTABLE/
Biological chemistry Hoppe-Seyler
AROMATASE INHIBITORS - MECHANISMS OF STEROIDAL INHIBITORS
Breast cancer research and treatment
CHARACTERIZATION OF A COS CELL-LINE DEFICIENT IN POLYAMINE TRANSPORT
Biochimica et biophysica acta. Molecular cell research