Per ulteriori informazioni selezionare i riferimenti di interesse.
Conformation of the tripeptide Cbz-Pro-Leu-Trp-OBzl(CF3)(2) deduced from two-dimensional H-1-NMR and conformational energy calculations is related toits affinity for NK1-receptor
JOURNAL OF PEPTIDE SCIENCE
Priming effects of substance P on calcium changes evoked by interleukin-8 in human neutrophils
JOURNAL OF LEUKOCYTE BIOLOGY
A flexible approach to the design of new potent substance P receptor ligands
JOURNAL OF PHARMACY AND PHARMACOLOGY
Molecular basis for selectivity of high affinity peptide antagonists for the gastrin-releasing peptide receptor
JOURNAL OF BIOLOGICAL CHEMISTRY
Tyrosine 220 in the 5th transmembrane domain of the neuromedin B receptor is critical for the high selectivity of the peptoid antagonist PD168368
JOURNAL OF BIOLOGICAL CHEMISTRY
Synthesis of a substance P antagonist with a somatostatin scaffold: Factors affecting agonism/antagonism at GPCRs and the role of pseudosymmetry
JOURNAL OF MEDICINAL CHEMISTRY
Substance P receptor antagonist I: Conversion of phosphoramidate prodrug after i.v. administration to rats and dogs
DRUG METABOLISM AND DISPOSITION
Axially chiral 1,7-naphthyridine-6-carboxamide derivatives as orally active tachykinin NK1 receptor antagonists: Synthesis, antagonistic activity, and effects on bladder functions
JOURNAL OF MEDICINAL CHEMISTRY
HUMAN SUBSTANCE-P RECEPTOR EXPRESSED IN SF9 CELLS COUPLES WITH MULTIPLE ENDOGENOUS G-PROTEINS
Journal of receptor and signal transduction research
HIGH-AFFINITY PHENYLGLYCINOL-BASED NK1 RECEPTOR ANTAGONISTS
Bioorganic & medicinal chemistry letters
Effect of temperature on recombinant protein expression in Semliki Forest virus infected mammalian cell lines growing in serum-free suspension cultures
CYTOTECHNOLOGY
Value of tachykinin receptor antagonists in the prevention of bronchial hyperresponsiveness, cough and bronchial inflammation.
REVUE FRANCAISE D ALLERGOLOGIE ET D IMMUNOLOGIE CLINIQUE
STERIC HINDRANCE MUTAGENESIS VERSUS ALANINE SCAN IN MAPPING OF LIGAND-BINDING SITES IN THE TACHYKININ NK1 RECEPTOR
Molecular pharmacology
STRUCTURAL OPTIMIZATION AFFORDING ENYL-4-(3-OXO-1,2,4-TRIAZOL-5-YL)METHYLMORPHOLINE, A POTENT, ORALLY-ACTIVE, LONG-ACTING MORPHOLINE ACETALHUMAN NK-1 RECEPTOR ANTAGONIST
Journal of medicinal chemistry
4,4-DISUBSTITUTED PIPERIDINE HIGH-AFFINITY NK1 ANTAGONISTS - STRUCTURE-ACTIVITY-RELATIONSHIPS AND IN-VIVO ACTIVITY
Journal of medicinal chemistry
SUBSTANCE-P DERIVATIVES WITH PHOTOACTIVATABLE LABELS IN THE N-TERMINAL PART OF THE MOLECULE
The journal of peptide research
THE TACHYKININ NK1 RECEPTOR - PART I - LIGANDS AND MECHANISMS OF CELLULAR ACTIVATION
Neuropeptides
ANTAGONISTS OF THE TACHYKININ RECEPTORS
Bioorganiceskaa himia
MAGNESIUM-DEFICIENCY-ENHANCED POSTISCHEMIC MYOCARDIAL INJURY IS REDUCED BY SUBSTANCE-P RECEPTOR BLOCKADE
Journal of Molecular and Cellular Cardiology
CHARACTERIZATION OF NONPEPTIDE ANTAGONIST AND PEPTIDE AGONIST BINDING-SITES OF THE NK1 RECEPTOR WITH FLUORESCENT LIGANDS
The Journal of biological chemistry
EFFECT OF SINGLE-POINT MUTATIONS OF THE HUMAN TACHYKININ NK1 RECEPTORON ANTAGONIST AFFINITY
European journal of pharmacology
CHARACTERIZATION OF THE BINDING AND ACTIVITY OF A HIGH-AFFINITY, PSEUDOIRREVERSIBLE MORPHOLINO TACHYKININ NK1 RECEPTOR ANTAGONIST
European journal of pharmacology
POTENT NK1 RECEPTOR ANTAGONISTS - SYNTHESIS AND ANTAGONISTIC ACTIVITYOF VARIOUS HETEROCYCLES WITH AN [3,5-BIS(TRIFLUOROMETHYL)BENZYL]-N-METHYLCARBAMOYL SUBSTITUENT
Chemical and Pharmaceutical Bulletin
P-(4-HYDROXYBENZOYL)PHENYLALANINE - A PHOTOREACTIVE AMINO-ACID ANALOGAMENABLE TO RADIOIODINATION FOR ELUCIDATION OF PEPTIDE-PROTEIN INTERACTION APPLICATION TO SUBSTANCE-P RECEPTOR
Biochemistry
SYSTEMATIC SEARCH STRATEGIES IN CONFORMATIONAL-ANALYSIS
Drug discovery today
LINEAR AMIDES AS SUBSTANCE-P ANTAGONISTS
Bioorganic & medicinal chemistry letters
NONPEPTIDE ANTAGONISTS OF THE NK1 TACHYKININ RECEPTOR
Medicinal research reviews
HETEROLOGOUS EXPRESSION OF G-PROTEIN-COUPLED RECEPTORS
Trends in biotechnology
DISSECTING PROCESSING AND APOPTOTIC ACTIVITY OF A CYSTEINE PROTEASE BY MUTANT ANALYSIS
The Journal of cell biology
IDENTIFICATION OF THE SITE IN THE SUBSTANCE-P (NK-1) RECEPTOR FOR MODULATION OF PEPTIDE BINDING BY SULFHYDRYL-REAGENTS
The Journal of biological chemistry
MOLECULAR CHARACTERIZATION OF A COMMON BINDING-SITE FOR SMALL MOLECULES WITHIN THE TRANSMEMBRANE DOMAIN OF G-PROTEIN COUPLED RECEPTORS
Journal of pharmacological and toxicological methods
PIPERIDINE-ETHER BASED HNK(1) ANTAGONISTS .2. INVESTIGATION OF THE EFFECT OF N-SUBSTITUTION
Bioorganic & medicinal chemistry letters
PHENYL-GLYCINOL BASED NK1 RECEPTOR ANTAGONISTS - TOWARDS THE MINIMUM PHARMACOPHORE
Bioorganic & medicinal chemistry letters
THE MAMMALIAN TACHYKININ RECEPTORS
General pharmacology
CHARACTERIZATION AND AUTORADIOGRAPHIC MAPPING OF [H-3] CP96,345, A NONPEPTIDE SELECTIVE NK1 RECEPTOR ANTAGONIST IN GUINEA-PIG LUNG
Peptides
4,4-DISUBSTITUTED PIPERIDINES - A NEW CLASS OF NK1 ANTAGONIST
Journal of medicinal chemistry
RADIOIODINATED L-703,606 - A POTENT, SELECTIVE ANTAGONIST TO THE HUMAN NK(1) RECEPTOR
Applied radiation and isotopes
GEM-DISUBSTITUTED AMINO-ETHER BASED SUBSTANCE-P ANTAGONISTS
Bioorganic & medicinal chemistry letters
PIPERIDINE-ETHER BASED HNK(1) ANTAGONISTS .1. DETERMINATION OF THE RELATIVE AND ABSOLUTE STEREOCHEMICAL REQUIREMENTS
Bioorganic & medicinal chemistry letters
FUNCTIONAL MAPPING OF THE LIGAND-BINDING SITES OF G-PROTEIN COUPLED RECEPTORS
Medicinal research reviews
STRUCTURE AND FUNCTION OF G-PROTEIN-COUPLED RECEPTORS
Annual review of biochemistry
TACHYKININ NK1 RECEPTOR SUBTYPES IN THE RAT URINARY-BLADDER
British Journal of Pharmacology
LYSINE-182 OF ENDOTHELIN-B RECEPTOR MODULATES AGONIST SELECTIVITY ANDANTAGONIST AFFINITY - EVIDENCE FOR THE OVER-LAP OF PEPTIDE AND NONPEPTIDE LIGAND-BINDING SITES
Biochemistry
QUINUCLIDINE BASED NK-1 ANTAGONISTS .2. DETERMINATION OF THE ABSOLUTESTEREOCHEMICAL REQUIREMENTS
Bioorganic & medicinal chemistry letters
MAPPING THE LIGAND-BINDING SITE OF THE NK-1 RECEPTOR
Regulatory peptides