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Molecular model of the Escherichia coli Na-1/H-1 antiporter NhaA
RECEPTORS & CHANNELS
Dopamine transporter in vitro binding and in vivo imaging in the brain
PHARMACOLOGY & TOXICOLOGY
Synthesis and preliminary characterization of a high-affinity novel radioligand for the dopamine transporter
SYNAPSE
Dopamine transporter imaging as an in vivo marker of dopaminergic neurons
DRUGS OF THE FUTURE
H-3-nicotine, H-3-flunitrazepam, and H-3-cocaine incorporation into melanin: A model for the examination of drug-melanin interactions
JOURNAL OF ANALYTICAL TOXICOLOGY
Amphetamine and N-acetylamphetamine incorporation into hair: An investigation of the potential role of drug basicity in hair color bias
JOURNAL OF ANALYTICAL TOXICOLOGY
Interactions of tryptamine derivatives with serotonin transporter species variants implicate transmembrane domain I in substrate recognition
MOLECULAR PHARMACOLOGY
Delineating structure-function relationships in the dopamine transporter from natural and engineered Zn2+ binding sites
LIFE SCIENCES
Functional role of critical stripe residues in transmembrane span 7 of theserotonin transporter - Effects of Na+, Li+, and methanethiosulfonate reagents
JOURNAL OF BIOLOGICAL CHEMISTRY
A conformationally sensitive residue on the cytoplasmic surface of serotonin transporter
JOURNAL OF BIOLOGICAL CHEMISTRY
Substrate-induced conformational changes of extracellular loop 1 in the glycine transporter GLYT2
JOURNAL OF BIOLOGICAL CHEMISTRY
Pharmacological properties of naturally occurring variants of the human norepinephrine transporter
PHARMACOGENETICS
Dopamine transporter function assessed by antisense knockdown in the rat: Protection from dopamine neurotoxicity
SYNAPSE
Evidence for bias in hair testing and procedures to correct bias
FORENSIC SCIENCE INTERNATIONAL
A comparison of sodium hydroxide and sodium sulfide digestion of mouse hair in the recovery of radioactivity following systemic administration of [H-3]-nicotine and [H-3]-flunitrazepam
JOURNAL OF ANALYTICAL TOXICOLOGY
Histologic localization of serum constituents, Ca-45(2+), Cl-36(-), [C-14]urea, and [S-35]cysteine in forming hair after systemic administration
DRUG METABOLISM AND DISPOSITION
Binding of uptake blockers to the neuronal dopamine transporter: further investigation about cationic and anionic requirements
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY
Importance of valine at position 152 for the substrate transport and 2 beta-carbomethoxy-3 beta-(4-fluorophenyl) tropane binding of dopamine transporter
MOLECULAR PHARMACOLOGY
Hair analysis for drugs of abuse XXI. Effect of para-substituents on benzene ring of methamphetamine on drug incorporation into rat hair
LIFE SCIENCES
Highly selective chiral N-substituted 3 alpha-[bis(4 '-fluorophenyl)methoxy]tropane analogues for the dopamine transporter: Synthesis and comparativemolecular field analysis
JOURNAL OF MEDICINAL CHEMISTRY
Novel conformationally constrained tropane analogues by 6-endo-trig radical cyclization and Stille coupling - Switch of activity toward the serotoninand/or norepinephrine transporter
JOURNAL OF MEDICINAL CHEMISTRY
Structure and function of the dopamine transporter
EUROPEAN JOURNAL OF PHARMACOLOGY
Structural probing of a microdomain in the dopamine transporter by engineering of artificial Zn2+ binding sites
BIOCHEMISTRY
Imaging of the dopaminergic neurotransmission system using single-photon emission tomography and positron emission tomography in patients with parkinsonism
EUROPEAN JOURNAL OF NUCLEAR MEDICINE
Transmembrane domain I contributes to the permeation pathway for serotoninand ions in the serotonin transporter
JOURNAL OF NEUROSCIENCE
Deposition of [H-3]cocaine, [H-3]nicotine, and [H-3]flunitrazepam in mousehair melanosomes after systemic administration
DRUG METABOLISM AND DISPOSITION
Comparison of the pharmacological properties of cloned rat, human, and bovine norepinephrine transporters
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Characteristics of drug interactions with recombinant biogenic amine transporters expressed in the same cell type
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Which form of dopamine is the substrate for the human dopamine transporter: The cationic or the uncharged species?
JOURNAL OF BIOLOGICAL CHEMISTRY
Defining proximity relationships in the tertiary structure of the dopaminetransporter - Identification of a conserved glutamic acid as a third coordinate in the endogenous Zn2+-binding site
JOURNAL OF BIOLOGICAL CHEMISTRY
NOVEL DOPAMINE TRANSPORTER LIGANDS - THE STATE-OF-THE-ART
Medicinal chemistry research
NEUROTRANSMITTER TRANSPORTERS AS MOLECULAR TARGETS FOR ADDICTIVE DRUGS
Drug and alcohol dependence
BRAIN DOPAMINE NEUROTOXICITY IN BABOONS TREATED WITH DOSES OF METHAMPHETAMINE COMPARABLE TO THOSE RECREATIONALLY ABUSED BY HUMANS - EVIDENCE FROM [C-11] WIN-35,428 POSITRON-EMISSION-TOMOGRAPHY STUDIES AND DIRECT IN-VITRO DETERMINATIONS
The Journal of neuroscience
DELINEATION OF AN ENDOGENOUS ZINC-BINDING SITE IN THE HUMAN DOPAMINE TRANSPORTER
EMBO journal (Print)
NOREPINEPHRINE TRANSPORTERS IN RAT PLACENTA LABELED WITH [H-3]NISOXETINE
The Journal of pharmacology and experimental therapeutics
RELATIONSHIPS BETWEEN THE CATECHOL SUBSTRATE-BINDING SITE AND AMPHETAMINE, COCAINE, AND MAZINDOL BINDING-SITES IN A KINETIC-MODEL OF THE STRIATAL TRANSPORTER OF DOPAMINE IN-VITRO
Journal of neurochemistry
CRITICAL AMINO-ACID-RESIDUES IN TRANSMEMBRANE SPAN-7 OF THE SEROTONINTRANSPORTER IDENTIFIED BY RANDOM MUTAGENESIS
The Journal of biological chemistry
HIGH-AFFINITY RECOGNITION OF SEROTONIN TRANSPORTER ANTAGONISTS DEFINED BY SPECIES-SCANNING MUTAGENESIS - AN AROMATIC RESIDUE IN TRANSMEMBRANE DOMAIN-I DICTATES SPECIES-SELECTIVE RECOGNITION OF CITALOPRAM AND MAZINDOL
The Journal of biological chemistry
Nature of methamphetamine-induced rapid and reversible changes in dopaminetransporters
EUROPEAN JOURNAL OF PHARMACOLOGY
SUBSTRATE TRANSPORT AND COCAINE BINDING OF HUMAN DOPAMINE TRANSPORTERIS REDUCED BY SUBSTITUTION OF CARBOXYL TAIL WITH THAT OF BOVINE DOPAMINE TRANSPORTER
NeuroReport
COMPARATIVE-EVALUATION OF [H-3] WIN-35428 AND [H-3] GBR-12935 AS MARKERS OF DOPAMINE INNERVATION DENSITY IN BRAIN
Synapse
DIFFERENTIAL REGULATION OF DOPAMINE TRANSPORTER AFTER CHRONIC SELF-ADMINISTRATION OF BUPROPION AND NOMIFENSINE
The Journal of pharmacology and experimental therapeutics
CATIONS AFFECT [H-3] MAZINDOL AND [H-3] WIN-35,428 BINDING TO THE HUMAN DOPAMINE TRANSPORTER IN A SIMILAR FASHION
Journal of neurochemistry
PHARMACOLOGY AND REGULATION OF THE NEURONAL DOPAMINE TRANSPORTER
European journal of pharmacology
SPECIES-DIFFERENCES IN FUNCTIONS OF DOPAMINE TRANSPORTER - PAUCITY OFMPP(+) UPTAKE AND COCAINE BINDING IN BOVINE DOPAMINE TRANSPORTER
Neuroscience letters
TRANSLOCATION OF DOPAMINE AND BINDING OF WIN-35,428 MEASURED UNDER IDENTICAL CONDITIONS IN CELLS EXPRESSING THE CLONED HUMAN DOPAMINE TRANSPORTER
Naunyn-Schmiedeberg's archives of pharmacology
SYNTHESIS AND TRANSPORTER BINDING-PROPERTIES OF 3-BETA-(4'-ALKYL)NORTROPANE-2-BETA-CARBOXYLIC ACID, 3-BETA-(4'-ALKENYL)NORTROPANE-2-BETA-CARBOXYLIC ACID, AND ETA-(4'-ALKYNYLPHENYL)NORTROPANE-2-BETA-CARBOXYLIC ACID METHYL-ESTERS - SEROTONIN TRANSPORTER SELECTIVE ANALOGS
Journal of medicinal chemistry
N-SUBSTITUTED ANALOGS OF 2-BETA-CARBOMETHOXY-3-BETA-(4'-IODOPHENYL)TROPANE (BETA-CIT) WITH SELECTIVE AFFINITY TO DOPAMINE OR SEROTONIN TRANSPORTERS IN RAT FOREBRAIN
Journal of medicinal chemistry
[H-3] WIN 35,428 BINDING IN THE HUMAN BRAIN
Brain research
BINDING DOMAINS FOR BLOCKERS AND SUBSTRATES ON THE CLONED HUMAN DOPAMINE TRANSPORTER STUDIED BY PROTECTION AGAINST N-ETHYLMALEIMIDE-INDUCEDREDUCTION OF A-CARBOMETHOXY-3-BETA-(4-FLUOROPHENYL)[H-3]TROPANE ([H-3]WIN-35,428) BINDING
Biochemical pharmacology
-BETA-CARBOMETHOXY-3-BETA-(4-FLUOROPHENYL)TROPANE] BINDING TO RAT-BRAIN MEMBRANES - COMPARING DOPAMINE CELL BODY AREAS WITH NERVE-TERMINAL REGIONS
Biochemical pharmacology
TEMPORAL RELATIONSHIPS BETWEEN THE PHARMACOKINETICS OF METHYLPHENIDATE IN THE HUMAN BRAIN AND ITS BEHAVIORAL AND CARDIOVASCULAR EFFECTS
Psychopharmacology
SYNTHESIS AND BINDING-PROPERTIES OF [H-3]NNC-12-0781, A NEW RADIOLIGAND FOR THE DOPAMINE REUPTAKE SYSTEM
Nuclear medicine and biology
RAT MESENCEPHALIC NEURONAL CELLS CULTURED FOR DIFFERENT PERIODS AS A MODEL OF DOPAMINE TRANSPORTER ONTOGENY
Molecular neurobiology
SENSITIVITY OF STRIATAL [C-11] COCAINE BINDING TO DECREASES IN SYNAPTIC DOPAMINE
Synapse
A NEW PET LIGAND FOR THE DOPAMINE TRANSPORTER - STUDIES IN THE HUMAN BRAIN
The Journal of nuclear medicine
STRIATAL DOPAMINE TRANSPORTER IMAGING IN NONHUMAN-PRIMATES WITH IODINE-123-IPT SPECT
The Journal of nuclear medicine
SELECTIVE LABELING OF THE DOPAMINE TRANSPORTER BY THE HIGH-AFFINITY LIGAND ETA-(4-[I-125]IODOPHENYL)TROPANE-2-BETA-CARBOXYLIC ACID ISOPROPYL ESTER
Molecular pharmacology
COMPARISON OF 2 PET RADIOLIGANDS FOR IMAGING EXTRASTRIATAL DOPAMINE TRANSPORTERS IN HUMAN BRAIN
Life sciences
LOCALIZATION AND QUANTIFICATION OF THE DOPAMINE TRANSPORTER - COMPARISON OF [H-3]WIN-35,428 AND [I-125]RTI-55
Brain research
MONOAMINE UPTAKE IN INSECT SYNAPTOSOMAL PREPARATIONS
Insect biochemistry and molecular biology
PHORBOL ESTERS ALTER FUNCTIONS OF THE EXPRESSED DOPAMINE TRANSPORTER
European journal of pharmacology. Molecular pharmacology section
PHARMACOKINETICS AND IN-VIVO SPECIFICITY OF [C-11] DL-THREO-METHYLPHENIDATE FOR THE PRESYNAPTIC DOPAMINERGIC NEURON
Synapse
MERCURIC-CHLORIDE AND P-CHLOROMERCURIPHENYLSULFONATE EXERT A BIPHASICEFFECT ON THE BINDING OF THE STIMULANT [H-3] METHYLPHENIDATE TO THE DOPAMINE TRANSPORTER
Synapse
STUDIES OF THE BIOGENIC-AMINE TRANSPORTERS .1. DOPAMINE REUPTAKE BLOCKERS INHIBIT [H-3] MAZINDOL BINDING TO THE DOPAMINE TRANSPORTER BY A COMPETITIVE MECHANISM - PRELIMINARY EVIDENCE FOR DIFFERENT BINDING DOMAINS
Neurochemical research
MOLECULAR, FUNCTIONAL AND BIOCHEMICAL CHARACTERISTICS OF THE DOPAMINETRANSPORTER - REGIONAL DIFFERENCES AND CLINICAL RELEVANCE
Clinical neuropharmacology
PREPARATION OF A POTENTIAL POSITRON EMISSION TOMOGRAPHIC RADIOLIGAND FOR THE DOPAMINE TRANSPORTER
European journal of nuclear medicine
PHARMACOLOGICAL HETEROGENEITY OF THE CLONED AND NATIVE HUMAN DOPAMINETRANSPORTER - DISASSOCIATION OF [H-3] WIN 35,428 AND [H-3] GBR 12,935BINDING
Molecular pharmacology
SYNTHESIS AND CHARACTERIZATION OF RADIOIODINATED -BETA-CARBOMETHOXY-3-BETA-(4-CHLOROPHENYL)TROPANES - POTENTIAL DOPAMINE REUPTAKE SITE IMAGING AGENTS
Journal of medicinal chemistry
EVALUATION OF THE MONOAMINE UPTAKE SITE LIGAND [I-123] METHYL 3-BETA-(4-IODOPHENYL)-TROPANE-2-BETA-CARBOXYLATE ([I-123)BETA-CIT) IN NONHUMAN-PRIMATES - PHARMACOKINETICS, BIODISTRIBUTION AND SPECT BRAIN IMAGINGCOREGISTERED WITH MRI
Nuclear medicine and biology
IN-VIVO IMAGING OF BABOON AND HUMAN DOPAMINE TRANSPORTERS BY POSITRONEMISSION TOMOGRAPHY USING [C-11] WIN-35,428
Synapse
COEXPRESSION OF DOPAMINE TRANSPORTER MESSENGER-RNA AND TYROSINE-HYDROXYLASE MESSENGER-RNA IN VENTRAL MESENCEPHALIC NEURONS
Molecular brain research
ALLOSTERIC REGULATION BY SODIUM OF THE BINDING OF [H-3] COCAINE AND [H-3] GBR-12935 TO RAT AND BOVINE STRIATA
Membrane biochemistry
QUANTITATIVE STRUCTURE-ACTIVITY-RELATIONSHIPS FOR SUBSTITUTED AMINOTETRALIN ANALOGS .2. INHIBITION OF DOPAMINE UPTAKE
Journal of pharmaceutical sciences