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Intracellular levels of two cyclosporin derivatives valspodar (PSC 833) and cyclosporin a closely associated with multidrug resistance-modulating activity in sublines of human colorectal adenocarcinoma HCT-15
JAPANESE JOURNAL OF CANCER RESEARCH
Type-specific epitope locations revealed by X-ray crystallographic study of adenovirus type 5 hexon
MOLECULAR THERAPY
BBR 3464: A novel triplatinum complex, exhibiting a preclinical profile ofantitumor efficacy different from cisplatin
CLINICAL CANCER RESEARCH
Neutralisation of adenovirus infectivity by ascitic fluid from ovarian cancer patients
GENE THERAPY
Mechanisms of drug resistance to the platinum complex ZD0473 in ovarian cancer cell lines
EUROPEAN JOURNAL OF CANCER
Balanced and purposeful departures: Fixing a jurisprudence that underminesthe federal sentencing guidelines
NOTRE DAME LAW REVIEW
P-glycoprotein inhibitor valspodar (PSC 833) increases the intracellular concentrations of daunorubicin in vivo in patients with p-glycoprotein-positive acute myeloid leukemia
JOURNAL OF CLINICAL ONCOLOGY
Modulation of daunorubicin cellular resistance by combination of P-glycoprotein blockers acting on drug efflux and intracellular drug sequestration in golgi vesicles
CYTOMETRY
Effect of PSC 833 on the cytotoxicity and pharmacodynamics of mitoxantronein multidrug-resistant K562 cells
LEUKEMIA RESEARCH
Defensive use of a fecal thatch by a beetle larva (Hemisphaerota cyanea)
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
BCL-2 family protein expression and platinum drug resistance in ovarian carcinoma
BRITISH JOURNAL OF CANCER
Mini-review: discovery and development of platinum complexes designed to circumvent cisplatin resistance
JOURNAL OF INORGANIC BIOCHEMISTRY
Idarubicin overcomes P-glycoprotein-related multidrug resistance: comparison with doxorubicin and daunorubicin in human multiple myeloma cell lines
LEUKEMIA RESEARCH
The neutral cysteine protease bleomycin hydrolase is essential for epidermal integrity and bleomycin resistance
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
Cytotoxicity of 2,2 ': 6 ',2 ''-terpyridineplatinum(II) complexes against human ovarian carcinoma
JOURNAL OF MEDICINAL CHEMISTRY
Novel multidrug resistance reversal agents
JOURNAL OF MEDICINAL CHEMISTRY
In vivo efficacy of XR9051, a potent modulator of P-glycoprotein mediated multidrug resistance
BRITISH JOURNAL OF CANCER
Newly synthesized dihydropyridine derivatives as modulators of P-glycoprotein-mediated multidrug resistance
BIOORGANIC & MEDICINAL CHEMISTRY
ENHANCEMENT OF CHEMOTHERAPEUTIC DRUG TOXICITY TO HUMAN TUMOR-CELLS IN-VITRO BY A SUBSET OF NONSTEROIDAL ANTIINFLAMMATORY DRUGS (NSAIDS)
European journal of cancer
SYNTHESIS OF A HIGHLY FUNCTIONALIZED GAMMA-LACTONE AS A PRECURSOR OF 9-PENTYL ANTHRACYCLINES
Tetrahedron : asymmetry
OVARIAN-CANCER CISPLATIN-RESISTANT CELL-LINES - MULTIPLE CHANGES INCLUDING COLLATERAL SENSITIVITY TO TAXOL
Annals of oncology
INHIBITION OF P-GLYCOPROTEIN - RAPID ASSESSMENT OF ITS IMPLICATION INBLOOD-BRAIN-BARRIER INTEGRITY AND DRUG TRANSPORT TO THE BRAIN BY AN IN-VITRO MODEL OF THE BLOOD-BRAIN-BARRIER
Pharmaceutical research
CHEMICAL, BIOCHEMICAL AND PHARMACOLOGICAL ACTIVITY OF THE NOVEL STERICALLY HINDERED PLATINUM COORDINATION COMPLEX, CIS-[AMMINEDICHLORO(2-METHYLPYRIDINE)] PLATINUM(II) (AMD473)
Anti-cancer drug design
VILSMEIER AND MANNICH REACTIONS ON (4S)-N-2-SUBSTITUTED 4-DIHYDRO-1H-PYRAZINO[2,1-B]QUINAZOLINE-3,6-DIONES
Tetrahedron
CONSTRUCTION AND CHARACTERIZATION OF HEXON-CHIMERIC ADENOVIRUSES - SPECIFICATION OF ADENOVIRUS SEROTYPE
Journal of virology (Print)
REVERSAL OF P-GLYCOPROTEIN-MEDIATED MULTIDRUG-RESISTANCE BY XR9051, ANOVEL DIKETOPIPERAZINE DERIVATIVE
British Journal of Cancer
IN-VITRO CIRCUMVENTION OF CISPLATIN RESISTANCE BY THE NOVEL STERICALLY HINDERED PLATINUM COMPLEX AMD473
British Journal of Cancer
S9788 MODULATION OF P-GLYCOPROTEIN-RELATED AND MULTIDRUG-RELATED PROTEIN-MEDIATED MULTIDRUG-RESISTANCE BY SERVIER-9788 IN DOXORUBICIN-RESISTANT MCF7 CELLS
Biochemical pharmacology
INHIBITORY EFFECT OF ALKYLATING MODULATORS ON THE FUNCTION OF P-GLYCOPROTEIN
Oncology research
A NOVEL QUINOLINE DERIVATIVE, MS-209, OVERCOMES DRUG-RESISTANCE OF HUMAN LUNG-CANCER CELLS EXPRESSING THE MULTIDRUG RESISTANCE-ASSOCIATE PROTEIN (MRP) GENE
Cancer chemotherapy and pharmacology
SDZ-PSC-833 - A NEW MULTIDRUG-RESISTANCE MODULATOR
Tumori
THE REVERSAL OF MULTIDRUG-RESISTANCE IN MULTICELLULAR TUMOR SPHEROIDSBY SDZ PSC-833
Anticancer research
SECONDARY DRUG-RESISTANCE IN BREAST-CANCER - FAILURE TO REVERSE WITH ORAL NIFEDIPINE
International journal of cancer
PHASE IB STUDY OF DOXORUBICIN IN COMBINATION WITH THE MULTIDRUG-RESISTANCE REVERSING AGENT S9788 IN ADVANCED COLORECTAL AND RENAL-CELL CANCER
British Journal of Cancer
REGRESSION OF ESTABLISHED TUMORS EXPRESSING P-GLYCOPROTEIN BY COMBINATIONS OF ADRIAMYCIN, CYCLOSPORINE DERIVATIVES, AND MRK-16 ANTIBODIES
Journal of the National Cancer Institute
DEVELOPMENT AND PARTIAL CHARACTERIZATION OF A HUMAN T-LYMPHOBLASTIC LEUKEMIC (CCRF-CEM) CELL-LINE RESISTANT TO ETOPOSIDE - ANALYSIS OF POSSIBLE CIRCUMVENTING APPROACHES
Journal of chemotherapy
DOES VERAPAMIL HELP OVERCOME MULTIDRUG-RESISTANCE IN TUMOR-CELL LINESAND CANCER-PATIENTS
Journal of chemotherapy
SYNTHESIS AND BIOLOGICAL-ACTIVITY OF 4'-AZIDO-3'-CHLORO-3'-DEAMINO-4'-DEOXYDAUNORUBICIN AND CETAMIDO-3'-CHLORO-3'-DEAMINO-4'-DEOXYDAUNORUBICIN
Bioorganic & medicinal chemistry letters
CREMOPHOR EL REVERSED MULTIDRUG-RESISTANCE IN-VITRO BUT NOT IN TUMOR-BEARING MOUSE MODELS
Anti-cancer drugs
MODULATION OF MULTIDRUG-RESISTANCE BY SDZ PSC-833 IN LEUKEMIC AND SOLID-TUMOR-BEARING MOUSE MODELS
Japanese journal of cancer research
REVERSAL OF MULTIDRUG-RESISTANCE BY SDZ PSC-833, COMBINED WITH VAD (VINCRISTINE, DOXORUBICIN, DEXAMETHASONE) IN REFRACTORY MULTIPLE-MYELOMA- A PHASE-I STUDY
Leukemia
PHASE-I STUDY OF ETOPOSIDE WITH SDZ PSC 833 AS A MODULATOR OF MULTIDRUG-RESISTANCE IN PATIENTS WITH CANCER
Journal of clinical oncology
OVERCOMING PGP-RELATED MULTIDRUG-RESISTANCE - THE CYCLOSPORINE DERIVATIVE SDZ PSC-833 CAN ABOLISH THE RESISTANCE TO METHOXY-MORPHOLYNIL-DOXORUBICIN
Haematologica
POTENTIATION OF ANTITUMOR AND ANTIMETASTATIC ACTIVITIES OF ADRIAMYCINBY A NOVEL N-ALKYLATED DIHYDROPYRIDINE, AC394, AND ITS ENANTIOMERS INCOLON CANCER-BEARING MICE
Cancer chemotherapy and pharmacology
MOLECULAR MECHANISMS OF MULTIDRUG-RESISTANCE IN CANCER-CHEMOTHERAPY
Pathology research and practice
CHEMOSENSITIZATION AND DRUG ACCUMULATION ASSAYS AS COMPLEMENTARY METHODS FOR THE SCREENING OF MULTIDRUG-RESISTANCE REVERSAL AGENTS
Cancer letters
EFFECTS OF VERAPAMIL AND S9788 ON MDR-1 MESSENGER-RNA EXPRESSION STUDIED BY IN-SITU HYBRIDIZATION
Anticancer research
COMPARISON OF DRUG ACCUMULATION IN P-GLYCOPROTEIN-EXPRESSING AND MRP-EXPRESSING HUMAN LEUKEMIA-CELLS
Leukemia research
RELATION AMONG THE RESISTANCE FACTOR, KINETICS OF UPTAKE, AND KINETICS OF THE P-GLYCOPROTEIN-MEDIATED EFFLUX OF DOXORUBICIN, DAUNORUBICIN, 8-(S)-FLUOROIDARUBICIN, AND IDARUBICIN IN MULTIDRUG-RESISTANT K562 CELLS
Molecular pharmacology
EXPERIMENTAL-MODELS FOR THE STUDY OF DRUG-RESISTANCE IN OSTEOSARCOMA - P-GLYCOPROTEIN-POSITIVE, MURINE OSTEOSARCOMA CELL-LINES
Journal of bone and joint surgery. American volume
COMPETITIVE-INHIBITION OF PHOTOAFFINITY-LABELING OF P-GLYCOPROTEIN BYANTICANCER DRUGS AND MODULATORS INCLUDING S9788
European journal of pharmacology
REVERSAL OF P-GLYCOPROTEIN-MEDIATED MULTIDRUG-RESISTANCE BY A POTENT CYCLOPROPYLDIBENZOSUBERANE MODULATOR, LY335979
Cancer research
TRANSPORT OF CISPLATIN AND BIS-ACETATO-AMMINE-DICHLOROCYCLOHEXYL-AMINE PLATINUM(IV) (JM216) IN HUMAN OVARIAN-CARCINOMA CELL-LINES - IDENTIFICATION OF A PLASMA-MEMBRANE PROTEIN ASSOCIATED WITH CISPLATIN RESISTANCE
Clinical cancer research
METHANODIBENZOSUBERYLPIPERAZINES AS POTENT MULTIDRUG-RESISTANCE REVERSAL AGENTS
Bioorganic & medicinal chemistry letters
REVERSAL OF MULTIPLE-DRUG RESISTANCE IN-VITRO BY PHOSPHORATHIOATE OLIGONUCLEOTIDES AND RIBOZYMES
Anti-cancer drugs
IN-VITRO ACTIVITY OF S-9788 ON A MULTIDRUG-RESISTANT LEUKEMIC-CELL LINE AND ON NORMAL HEMATOPOIETIC CELLS-REVERSAL OF MULTIDRUG-RESISTANCE BY SERA FROM PHASE-I TREATED PATIENTS
Cancer chemotherapy and pharmacology
COMPARATIVE-STUDY ON REVERSAL EFFICACY OF SDZ PSC-833, CYCLOSPORINE-AAND VERAPAMIL ON MULTIDRUG-RESISTANCE IN-VITRO AND IN-VIVO
Acta oncologica
RESISTANCE TO CHEMOTHERAPY IN RENAL-CELL CANCER AND THERAPEUTIC PROSPECTIVES
Journal d'urologie
REVERSAL OF MULTIDRUG-RESISTANCE BY NOVEL CYCLOSPORINE-A ANALOGS AND THE CYCLOPEPTIDE SDZ-214-103 BIOSYNTHESIZED IN-VITRO
Journal of cancer research and clinical oncology
ACTIVITY OF THE MORPHOLINO ANTHRACYCLINE MINO-3'-MORPHOLINO-13-DEOXO-10-HYDROXYCARMINOMYCIN (MX2) AGAINST HUMAN TUMOR COLONY-FORMING-UNITS IN-VITRO
Investigational new drugs
EVALUATION OF RESISTANCE INDEX OF SEVERAL ANTICANCER AGENTS ON PARENTAL AND RESISTANT P-388 CELL-LINES
Leukemia research
NOVEL HEXAKIS(ARENEISONITRILE)TECHNETIUM(I) COMPLEXES AS RADIOLIGANDSTARGETED TO THE MULTIDRUG-RESISTANCE P-GLYCOPROTEIN
Journal of medicinal chemistry
ABSENCE OF THE MDR1A P-GLYCOPROTEIN IN MICE AFFECTS TISSUE DISTRIBUTION AND PHARMACOKINETICS OF DEXAMETHASONE, DIGOXIN, AND CYCLOSPORINE-A
The Journal of clinical investigation
SYNTHESIS AND ANTIPROLIFERATIVE EFFECTS OF A 4'-MORPHOLINO-9-METHYL ANTHRACYCLINE
Journal of antibiotics
DECREASED BIOTOLERABILITY FOR IVERMECTIN AND CYCLOSPORINE-A IN MICE EXPOSED TO POTENT P-GLYCOPROTEIN INHIBITORS
International journal of cancer
CARBOXYLATION OF KINETICALLY INERT PLATINUM(IV) HYDROXY COMPLEXES - AN ENTREE INTO ORALLY-ACTIVE PLATINUM(IV) ANTITUMOR AGENTS
Inorganic chemistry
N-ALKYLATED 1,4-DIHYDROPYRIDINES - NEW AGENTS TO OVERCOME MULTIDRUG-RESISTANCE
Chemical and Pharmaceutical Bulletin
A PHASE-III RANDOMIZED STUDY OF ORAL VERAPAMIL AS A CHEMOSENSITIZER TO REVERSE DRUG-RESISTANCE IN PATIENTS WITH REFRACTORY MYELOMA - A SOUTHWEST-ONCOLOGY-GROUP STUDY
Cancer
DECREASED POTENCY OF MDR-MODULATORS UNDER SERUM CONDITIONS DETERMINEDBY A FUNCTIONAL ASSAY
British Journal of Haematology
CONTINUOUS-INFUSION VERAPAMIL WITH ETOPOSIDE IN RELAPSED OR RESISTANTPEDIATRIC CANCERS
British Journal of Cancer
CHARACTERIZATION OF MULTIDRUG-RESISTANCE P-GLYCOPROTEIN TRANSPORT FUNCTION WITH AN ORGANOTECHNETIUM CATION
Biochemistry
THE EFFECT OF CROWN-ETHERS, TETRAALKYLAMMONIUM SALTS, AND POLYOXYETHYLENE AMPHIPHILES ON PIRARUBICIN INCORPORATION IN K562 RESISTANT CELLS
Biochemical pharmacology
IN-VITRO EFFECTS OF PENTOXIFYLLINE AND DOXORUBICIN ON CELL-SURVIVAL AND DNA-DAMAGE IN SENSITIVE AND MDR-P388 LEUKEMIA-CELLS
Cancer biotherapy
MULTIDRUG-RESISTANCE CIRCUMVENTION AND INHIBITION OF [H-3] AZIDOPINE PHOTOLABELING OF P-GLYCOPROTEIN BY NEW DIHYDROPYRIDINE DERIVATIVES DISPLAYING A LOW-AFFINITY FOR CALCIUM CHANNELS
International journal of oncology
SDZ 280-125 - A CYCLOPEPTOLIDE ENDOWED WITH AN IN-VITRO CYCLOSPORINE A-LIKE PROFILE OF ACTIVITY FOR THE REVERSION OF THE P-GLYCOPROTEIN-MEDIATED MULTIDRUG-RESISTANCE OF TUMOR-CELLS
Anti-cancer drugs
REVERSAL EFFECTS OF SEVERAL CA2-ENTRY BLOCKERS, NEUROLEPTICS AND LOCAL-ANESTHETICS ON P-GLYCOPROTEIN-MEDIATED VINCRISTINE RESISTANCE OF L1210()VCR MOUSE LEUKEMIC-CELL LINE/
Drugs under experimental and clinical research
SELECTIVE POTENTIATION OF PLATINUM DRUG CYTOTOXICITY IN CISPLATIN-SENSITIVE AND CISPLATIN-RESISTANT HUMAN OVARIAN-CARCINOMA CELL-LINES BY AMPHOTERICIN-B
Cancer chemotherapy and pharmacology
REVERSAL OF THE HUMAN AND MURINE MULTIDRUG-RESISTANCE PHENOTYPE WITH MEGESTROL-ACETATE
Cancer chemotherapy and pharmacology
DIFFERENTIAL EFFECTIVENESS OF A RANGE OF NOVEL DRUG-RESISTANCE MODULATORS, RELATIVE TO VERAPAMIL, IN INFLUENCING VINBLASTINE OR TENIPOSIDE CYTOTOXICITY IN HUMAN LYMPHOBLASTOID CCRF-CEM SUBLINES EXPRESSING CLASSIC OR ATYPICAL MULTIDRUG-RESISTANCE
Cancer chemotherapy and pharmacology
IN-VIVO REVERSAL OF MULTIDRUG-RESISTANCE BY 2 NEW DIHYDROPYRIDINE DERIVATIVES, S16317 AND S16324
Acta oncologica
TETRAVALENT PLATINUM COMPLEXES WITH AMMINE AMINE CARRIER LIGAND CONFIGURATION - CIRCUMVENTION OF PLATINUM RESISTANCE IN-VIVO
Anti-cancer drug design
SYNTHESIS AND BIOLOGICAL-ACTIVITY OF 3'-DEAMINO-3'-HALOANTHRACYCLINES
Anti-cancer drug design
EFFECT OF S9788, CYCLOSPORINE-A AND VERAPAMIL ON INTRACELLULAR-DISTRIBUTION OF THP-DOXORUBICIN IN MULTIDRUG-RESISTANT K562 TUMOR-CELLS, AS STUDIED BY LASER CONFOCAL MICROSPECTROFLUOROMETRY
Anticancer research
FLOW CYTOMETRIC DETERMINATION OF THE MULTIDRUG-RESISTANT PHENOTYPE INACUTE-LEUKEMIA
Cytometry
MODULATION OF DOXORUBICIN-TOXICITY BY TAMOXIFEN IN MULTIDRUG-RESISTANT TUMOR-CELLS IN-VITRO AND IN-VIVO
Journal of cancer research and clinical oncology
CLINICAL RELEVANCE OF P-GLYCOPROTEIN EXPRESSION IN HEMATOLOGICAL MALIGNANCIES
Leukemia research
REVERSAL OF CHEMORESISTANCE IN MALIGNANT GLIOMAS BY CALCIUM-ANTAGONISTS - CORRELATION WITH THE EXPRESSION OF MULTIDRUG-RESISTANT P-GLYCOPROTEIN
Journal of neurosurgery
DERIVATIVES OF A NOVEL CYCLOPEPTOLIDE .2. SYNTHESIS, ACTIVITY AGAINSTMULTIDRUG-RESISTANCE IN CHO AND KB CELLS IN-VITRO, AND STRUCTURE-ACTIVITY-RELATIONSHIPS
Journal of medicinal chemistry
MODULATION OF CYTOSTATIC DRUGS BY NIFEDIPINE IN 2 HETEROTRANSPLANTED HUMAN TESTICULAR-CANCER CELL-LINES DIFFERING IN THEIR SENSITIVITY TO STANDARD AGENTS
International journal of cancer
P-GLYCOPROTEIN-MEDIATED EFFLUX OF HYDROXYRUBICIN, A NEUTRAL ANTHRACYCLINE DERIVATIVE, IN RESISTANT K562 CELLS
FEBS letters
REVERSAL OF MULTIDRUG-RESISTANCE BY RU-486
Cancer research
QUANTITATIVE CYTOLOGICAL STUDY OF THE ACT IVITY OF A NEW RESISTANCE MODULATOR, S-9788, ON HUMAN LEUKEMIC-CELLS USING MULTIPARAMETRIC IMAGE-ANALYSIS
Bulletin du cancer
PHARMACOLOGICAL PROPERTIES OF S9788, A NE W MULTIDRUG-RESISTANCE MODULATOR
Bulletin du cancer
TIME-SCHEDULE DEPENDENT REVERSION OF MULTIDRUG-RESISTANCE BY S9788 INHUMAN TUMOR-CELL LINES
Bulletin du cancer
EFFECTS OF A NEW ANTIESTROGEN, IDOXIFENE, ON CISPLATIN-SENSITIVE AND DOXORUBICIN-SENSITIVE AND DOXORUBICIN-RESISTANT HUMAN OVARIAN-CARCINOMA CELL-LINES
British Journal of Cancer
COMPARATIVE-EVALUATION OF S9788, VERAPAMIL, AND CYCLOSPORINE-A IN K562 HUMAN LEUKEMIA-CELL LINES AND IN P-GLYCOPROTEIN-EXPRESSING SAMPLES PATIENTS WITH HEMATOLOGIC MALIGNANCIES
Blood
STRUCTURALLY DISTINCT MDR MODULATORS SHOW SPECIFIC PATTERNS OF REVERSAL AGAINST P-GLYCOPROTEINS BEARING UNIQUE MUTATIONS AT SERINE(939 941)/
Biochemistry
CYTOTOXIC EFFECT OF THE PROTEIN-DOXORUBICIN CONJUGATES ON THE MULTIDRUG-RESISTANT HUMAN MYELOGENOUS LEUKEMIA-CELL LINE, K562, IN-VITRO
Tumor biology
IDARUBICIN IS ACTIVE ON MDR CELLS - EVALUATION OF DNA-SYNTHESIS INHIBITION ON P388 CELL-LINES
Annals of hematology
MULTIDRUG-RESISTANCE (MDR) GENES IN HEMATOLOGICAL MALIGNANCIES
Cytotechnology