Per ulteriori informazioni selezionare i riferimenti di interesse.
Treating type 2 diabetes - today's targets, tomorrow's goals
DIABETES OBESITY & METABOLISM
Thiazolidinediones and liver toxicity
DIABETES & METABOLISM
Health care costs associated with escalation of drug treatment in type 2 diabetes mellitus
AMERICAN JOURNAL OF HEALTH-SYSTEM PHARMACY
Nateglinide
AMERICAN JOURNAL OF HEALTH-SYSTEM PHARMACY
Factors associated with discontinuing insulin therapy after diabetic ketoacidosis in adult diabetic patients
DIABETIC MEDICINE
Antihyperglycemic activity of new 1,2,4-oxadiazolidine-3,5-diones
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Type-2-diabetes in children and adolescents
MONATSSCHRIFT KINDERHEILKUNDE
Repaglinide - A review of its therapeutic use in type 2 diabetes mellitus
DRUGS
Improved diabetic syndrome in C57BL/KsJ-db/db mice by oral administration of the Na+-glucose cotransporter inhibitor T-1095
BRITISH JOURNAL OF PHARMACOLOGY
Synthesis and hypoglycemic activity of some new flavone derivatives - 4th Communication: 6-Flavonyl-2,4-thiazolidinediones
ARZNEIMITTEL-FORSCHUNG-DRUG RESEARCH
Pioglitazone hydrochloride in combination with sulfonylurea therapy improves glycemic control in patients with type 2 diabetes mellitus: A randomized, placebo-controlled study
AMERICAN JOURNAL OF MEDICINE
Patent focus on antidiabetic agents: September 1999-February 2000
EXPERT OPINION ON THERAPEUTIC PATENTS
Synthetic ligands for PPAR gamma - review of patent literature 1994-1999
EXPERT OPINION ON THERAPEUTIC PATENTS
The basal SAR of a novel insulin receptor activator
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Combining pioglitazone with a sulphonylurea or metformin in the managementof type 2 diabetes
EXPERIMENTAL AND CLINICAL ENDOCRINOLOGY & DIABETES
A PPAR gamma mutant serves as a dominant negative inhibitor of PPAR signaling and is localized in the nucleus
MOLECULAR AND CELLULAR ENDOCRINOLOGY
New azolidinediones as inhibitors of protein tyrosine phosphatase 1B with antihyperglycemic properties
JOURNAL OF MEDICINAL CHEMISTRY
A rational approach to drug therapy of type 2 diabetes mellitus
DRUGS
Synthesis and hypoglycemic activity of some new flavone derivatives - 3rd communication: 3 '-flavonyl-2,4-thiazolidinediones
ARZNEIMITTEL-FORSCHUNG-DRUG RESEARCH
Synthesis and hypoglycemic activity of some new flavone derivatives - 2nd communication: 4 '-flavonyl-2,4-thiazolidinediones
ARZNEIMITTEL-FORSCHUNG-DRUG RESEARCH
Physiology, pathology and pharmacology of insulin secretion
ACTA CLINICA BELGICA
Recent developments in oral hypoglycemic agents
DRUG DISCOVERY TODAY
A review of metabolic and cardiovascular effects of oral antidiabetic agents: beyond glucose-level lowering
JOURNAL OF CARDIOVASCULAR RISK
Three-dimensional quantitative structure activity relationships (3-D-QSAR)of antihyperglycemic agents
BIOORGANIC & MEDICINAL CHEMISTRY
Non-thiazolidinedione antihyperglycaemic agents. Part 3: The effects of stereochemistry on the potency of alpha-methoxy-beta-phenylpropanoic acids
BIOORGANIC & MEDICINAL CHEMISTRY
Stereoselective follow-up reactions of (S)-2-sulfanyl nitriles
TETRAHEDRON-ASYMMETRY
Non-thiazolidinedione antihyperglycaemic agents. Part 4: Synthesis of ( plus /-)-, (R)-(+)- and (S)-(-)-enantiomers of 2-oxy-3-arylpropanoic acids
TETRAHEDRON-ASYMMETRY
Non-thiazolidinedione antihyperglycaemic agents. Part 5: Asymmetric aldol synthesis of (S)-(-)-2-oxy-3-arylpropanoic acids
TETRAHEDRON-ASYMMETRY
Mechanism of action of a new class of insulin secretagogues
EXPERIMENTAL AND CLINICAL ENDOCRINOLOGY & DIABETES
Troglitazone inhibits expression of the phosphoenolpyruvate carboxykinase gene by an insulin-independent mechanism
BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR CELL RESEARCH
Pharmacological management of diabetes: Recent progress and future perspective in daily drug treatment
PHARMACOLOGY & THERAPEUTICS
A risk-benefit assessment of metformin in type 2 diabetes mellitus
DRUG SAFETY
Solid-liquid phase transfer catalyzed novel glycosylation reaction of phenols
SYNTHETIC COMMUNICATIONS
Novel euglycemic and hypolipidemic agents. 4. Pyridyl- and quinolinyl-containing thiazolidinediones
JOURNAL OF MEDICINAL CHEMISTRY
Effects of vanadium complexes with organic ligands on glucose metabolism: a comparison study in diabetic rats
BRITISH JOURNAL OF PHARMACOLOGY
Oral bioavailability and pharmacokinetics of the new insulin sensitizer DRF-2189 in Wistar rats
ARZNEIMITTEL-FORSCHUNG-DRUG RESEARCH
Reduction of vascular tone by introduction of troglitazone to the canine coronary artery
ARZNEIMITTEL-FORSCHUNG-DRUG RESEARCH
Pharmacologic therapy for type 2 diabetes mellitus
ANNALS OF INTERNAL MEDICINE
TROGLITAZONE - AN ANTIDIABETIC AGENT (REPRINTED)
American journal of health-system pharmacy
NOVEL EUGLYCEMIC AND HYPOLIPIDEMIC AGENTS - PART-2 - ANTIOXIDANT MOIETY AS STRUCTURAL MOTIF
Bioorganic & medicinal chemistry letters
PHARMACOLOGICAL TREATMENT OF DIABETIC-PATIENTS WITH CARDIOVASCULAR COMPLICATIONS
Journal of internal medicine
Combined glibenclamide plus metformin improves insulin sensitivity in non-obese Type 2 diabetic patients
DIABETES NUTRITION & METABOLISM
IDENTIFICATION OF HIGH-AFFINITY BINDING-SITES FOR THE INSULIN SENSITIZER ROSIGLITAZONE (BRL-49653) IN RODENT AND HUMAN ADIPOCYTES USING A RADIOIODINATED LIGAND FOR PEROXISOMAL PROLIFERATOR-ACTIVATED RECEPTOR-GAMMA
The Journal of pharmacology and experimental therapeutics
NOVEL -PROPYNYL)-5-(ARYLSULFONYL)THIAZOLIDINE-2,4-DIONES AS ANTIHYPERGLYCEMIC AGENTS
Journal of medicinal chemistry
ISOXAZOLIDINE-3,5-DIONE AND NONCYCLIC 1,3-DICARBONYL COMPOUNDS AS HYPOGLYCEMIC AGENTS
Journal of medicinal chemistry
NOVEL EUGLYCEMIC AND HYPOLIPIDEMIC AGENTS - 1
Journal of medicinal chemistry
N-(2-benzoylphenyl)-L-tyrosine PPAR gamma agonists. 1. Discovery of a novel series of potent antihyperglycemic and antihyperlipidemic agents
JOURNAL OF MEDICINAL CHEMISTRY
N-(2-benzoylphenyl)-L-tyrosine PPAR gamma agonists. 2. Structure-activity relationship and optimization of the phenyl alkyl ether moiety
JOURNAL OF MEDICINAL CHEMISTRY
ACTIONS OF NOVEL ANTIDIABETIC THIAZOLIDINEDIONE, T-174, IN ANIMAL-MODELS OF NON-INSULIN-DEPENDENT DIABETES-MELLITUS (NIDDM) AND IN CULTUREDMUSCLE-CELLS
British Journal of Pharmacology
PHARMACOLOGICAL AND PHARMACOKINETIC STUDIES OF THE NEWLY SYNTHESIZED THIAZOLIDINEDIONE DERIVATIVE ROPANECARBONYLAMINO)BENZYL)-THIAZOLIDINE-2,4-DIONE
Arzneimittel-Forschung
APPROACH TO THE PATIENT WITH DIABETES UNDERGOING A VASCULAR OR INTERVENTIONAL PROCEDURE
Journal of vascular and interventional radiology
NOVEL INDOLE CONTAINING THIAZOLIDINEDIONE DERIVATIVES AS POTENT EUGLYCEMIC AND HYPOLIPEMIC AGENTS
Bioorganic & medicinal chemistry letters
REGULATION OF THE UNCOUPLING PROTEIN GENE-EXPRESSION
European journal of endocrinology
SYNTHETIC APPROACHES TO BENZOFURAN CONTAINING INSULIN SENSITIVITY ENHANCER COMPOUNDS FOR TREATMENT OF TYPE-II DIABETES
Heterocycles
STUDIES ON COMPOUNDS WITH ANTIOXIDANT ACTIVITY - DEVELOPMENT OF HYPOGLYCEMIC AGENTS, TROGLITAZONE (CS-045)
Yakugaku zasshi
PIOGLITAZONE REDUCES SMOOTH-MUSCLE CELL-DENSITY OF RAT CAROTID ARTERIAL INTIMA INDUCED BY BALLOON CATHETERIZATION
Hormone and Metabolic Research
NOVEL BENZOXAZOLE 2,4-THIAZOLIDINEDIONES AS POTENT HYPOGLYCEMIC AGENTS - SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS
Chemical and Pharmaceutical Bulletin
HYPOGLYCEMIC EFFECTS OF THE NOVEL ANTIDIABETIC AGENT REPAGLINIDE IN RATS AND DOGS
British Journal of Pharmacology
STUDIES ON THE METABOLISM OF THE NEW ANTIDIABETIC AGENT PIOGLITAZONE - IDENTIFICATION OF METABOLITES IN RATS AND DOGS
Arzneimittel-Forschung
PHARMACOLOGICAL REGULATION OF BLOOD-GLUCOSE LEVELS IN NON-INSULIN-DEPENDENT DIABETES-MELLITUS
Archives of internal medicine
HIGH-PERFORMANCE LIQUID-CHROMATOGRAPHIC DETERMINATION OF PIOGLITAZONEAND ITS METABOLITES IN HUMAN SERUM AND URINE
Journal of chromatography B. Biomedical applications
NEW THERAPEUTIC AGENTS FOR THE TREATMENT OF INSULIN-RESISTANCE AND NIDDM
Drug discovery today
PEROXISOME PROLIFERATOR-ACTIVATED RECEPTORS - A NUCLEAR RECEPTOR SIGNALING PATHWAY IN LIPID PHYSIOLOGY
Annual review of cell and developmental biology
ACARBOSE - AN ALPHA-GLUCOSIDASE INHIBITOR
American journal of health-system pharmacy
NON THIAZOLIDINEDIONE ANTIHYPERGLYCEMIC AGENTS .1. ALPHA-HETEROATOM SUBSTITUTED BETA-PHENYLPROPANOIC ACIDS
Bioorganic & medicinal chemistry letters
DIFFERENTIAL INHIBITORY EFFECTS OF ANTIDIABETIC DRUGS ON ARTERIAL SMOOTH-MUSCLE CELL-PROLIFERATION
American journal of hypertension
ORAL ANTIDIABETIC DRUGS - AN OVERVIEW
Diabetic medicine
DEPRESSED INSULIN-SECRETION IN RESPONSE TO DIFFERENT STIMULI IS A FEATURE OF SECONDARY FAILURE IN NORMAL-WEIGHT NON-INSULIN-DEPENDENT DIABETICS ON SULFONYLUREAS
Diabetes, nutrition & metabolism
CONCISE APPROACH TO 1-THIAHYDANTOCIDIN
Synthetic communications
HYPOGLYCEMIC ACTIVITY OF A SERIES OF ALPHA-ALKYLTHIO AND ALPHA-ALKOXYCARBOXYLIC-ACIDS RELATED TO CIGLITAZONE
Journal of medicinal chemistry
MICROBIOLOGICAL N-DEOXYGENATION AND C-OXYGENATION OF PIOGLITAZONE-N-OXIDE IN A SINGLE FERMENTATION
Journal of antibiotics
CHOLESTATIC HEPATITIS INDUCED BY GLYBENCL AMIDE IN A PATIENT WITH HEPATITIS-C VIRUS
Revista espanola de enfermedades digestivas
15-DEOXY-DELTA(12,14)-PROSTAGLANDIN J(2) IS A LIGAND FOR THE ADIPOCYTE DETERMINATION FACTOR PPAR-GAMMA
Cell
STUDIES ON NEW ACIDIC AZOLES AS GLUCOSE-LOWERING AGENTS IN OBESE, DIABETIC DB DB MICE/
Journal of medicinal chemistry
DOSE PROPORTIONALITY STUDIES OF NOVEL THIAZOLIDINEDIONE DERIVATIVES AS POTENT ANTIDIABETIC AGENTS IN MICE
Arzneimittel-Forschung
EUGLYCEMIC AND BIOLOGICAL-ACTIVITIES OF NOVEL THIAZOLIDINE-2,4-DIONE DERIVATIVES
Arzneimittel-Forschung
PHARMACOKINETICS OF SOME NEW ORAL BLOOD GLUCOSE-LOWERING AGENTS IN DOGS
Arzneimittel-Forschung
THE SYNTHESIS OF BRL-49653 - A NOVEL AND POTENT ANTIHYPERGLYCEMIC AGENT
Bioorganic & medicinal chemistry letters
OCYCLYLAMINO)ALKOXY]BENZYL]-2,4-THIAZOLIDINEDIONES AS POTENT ANTIHYPERGLYCEMIC AGENTS
Journal of medicinal chemistry
SYNTHESIS AND ALDOSE REDUCTASE INHIBITORY ACTIVITY OF O[4H-1-BENZOPYRAN-4,4'-IMIDAZOLIDINE]-2',5'-DIONES
Arzneimittel-Forschung
PHARMACOLOGICAL TREATMENT OF THE OBESE-DIABETIC PATIENT
Diabete et metabolisme
ANTIHYPERGLYCEMIC ACTIVITY OF NOVEL NAPHTHALENYL 3H-1,2,3,5-OXATHIADIAZOLE 2-OXIDES
Journal of medicinal chemistry
HYDROXYUREA DERIVATIVES AS HYPOGLYCEMIC AGENTS
Journal of medicinal chemistry