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Update on the role of acyl-CoA : cholesterol acyltransferase inhibitors inatherosclerosis
EXPERT OPINION ON THERAPEUTIC PATENTS
A role for smooth endoplasmic reticulum membrane cholesterol ester in determining the intracellular location and regulation of sterol-regulatory-element-binding protein-2
BIOCHEMICAL JOURNAL
Overexpression of CYP27 in hepatic and extrahepatic cells: role in the regulation of cholesterol homeostasis
AMERICAN JOURNAL OF PHYSIOLOGY-GASTROINTESTINAL AND LIVER PHYSIOLOGY
Monoclonal antibody detection of plasma membrane cholesterol microdomains responsive to cholesterol trafficking
JOURNAL OF LIPID RESEARCH
NTE-122, an acyl-CoA : cholesterol acyltransferase inhibitor, prevents theprogression of atherogenesis in cholesterol-fed rabbits
JAPANESE JOURNAL OF PHARMACOLOGY
Postprandial hyperlipidemia in Zucker diabetic fatty fa/fa rats, an animalmodel of type II diabetes, and its amelioration by acyl-CoA : cholesterol acyltransferase inhibition
JAPANESE JOURNAL OF PHARMACOLOGY
Pharmacological properties of R-755, a novel acyl-CoA : cholesterol acyltransferase inhibitor, in cholesterol-fed rats, hamsters and rabbits
JAPANESE JOURNAL OF PHARMACOLOGY
A target for cholesterol absorption inhibitors in the enterocyte brush border membrane
BIOCHIMICA ET BIOPHYSICA ACTA-MOLECULAR AND CELL BIOLOGY OF LIPIDS
Modulation of endoplasmic reticulum-bound cholesterol regulatory enzymes by iron/ascorbate-mediated lipid peroxidation
FREE RADICAL BIOLOGY AND MEDICINE
ApoB100 secretion from HepG2 cells is decreased by the ACAT inhibitor CI-1011 - An effect associated with enhanced intracellular degradation of ApoB
ARTERIOSCLEROSIS THROMBOSIS AND VASCULAR BIOLOGY
Regulation of guinea pig hepatic acyl-CoA : cholesterol acyltransferase activity by dietary fat saturation and cholesterol
JOURNAL OF NUTRITIONAL BIOCHEMISTRY
Activities of acyl-CoA : cholesterol acyltransferase and cholesteryl esterhydrolase in the yolk sac membrane of the alligator (Alligator mississippiensis) embryo
COMPARATIVE BIOCHEMISTRY AND PHYSIOLOGY B-BIOCHEMISTRY & MOLECULAR BIOLOGY
Bile duct cells: a novel in vitro model for the study of lipid metabolism and bile acid production
AMERICAN JOURNAL OF PHYSIOLOGY-GASTROINTESTINAL AND LIVER PHYSIOLOGY
Paradoxical effect on atherosclerosis of hormone-sensitive lipase overexpression in macrophages
JOURNAL OF LIPID RESEARCH
Effects of NTE-122, an acyl-CoA : cholesterol acyltransferase inhibitor, on cholesterol esterification and lipid secretion from CaCo-2 cells, and cholesterol absorption in rats
JAPANESE JOURNAL OF PHARMACOLOGY
Effects of NTE-122, a novel acyl-CoA : cholesterol acyltransferase inhibitor, on cholesterol esterification and secretions of apolipoprotein B-containing lipoprotein and bile acids in HepG2
JAPANESE JOURNAL OF PHARMACOLOGY
Effects of NTE-122, a novel acyl-CoA : cholesterol acyltransferase inhibitor, on cholesterol esterification and high-density lipoprotein-induced cholesterol efflux in macrophages
JAPANESE JOURNAL OF PHARMACOLOGY
THE ACAT INHIBITOR HL-004 INHIBITS CHOLESTEROL ABSORPTION AND LOWERS SERUM-CHOLESTEROL IN RATS
General pharmacology
GEMFIBROZIL REDUCES NON-HIGH-DENSITY LIPOPROTEIN CHOLESTEROL IN EXOGENOUSLY HYPERCHOLESTEROLEMIC (EXHC) RATS FED A HIGH-CHOLESTEROL DIET
Comparative biochemistry and physiology. B. Comparative biochemistry
SYNTHETIC STUDY OF ALPHA-PYRONE MEROTERPE NOIDS, PYRIPYROPENES
Yuki Gosei Kagaku Kyokaishi
DIETARY FATTY-ACIDS AND THE REGULATION OF PLASMA LOW-DENSITY-LIPOPROTEIN CHOLESTEROL CONCENTRATIONS
The Journal of nutrition
EFFECTS OF F-1394, AN ACYL-COA-CHOLESTEROL ACYLTRANSFERASE (ACAT) INHIBITOR, ON ACAT ACTIVITY IN HEPG2 CELLS AND ON HEPATIC SECRETION OF LIPIDS IN TRITON WR-1339-INDUCED HYPERLIPIDEMIC RATS - POSSIBLE ROLE OF HEPATIC ACAT IN VERY-LOW-DENSITY LIPOPROTEIN SECRETION
Japanese Journal of Pharmacology
Cholesterol-lowering effects of NTE-122, a novel acyl-CoA : cholesterol acyltransferase (ACAT) inhibitor, on cholesterol diet-fed rats and rabbits
JAPANESE JOURNAL OF PHARMACOLOGY
MOLECULAR-CLONING, FUNCTIONAL EXPRESSION AND TISSUE DISTRIBUTION OF RAT ACYL-COENZYME A-CHOLESTEROL ACYLTRANSFERASE
Biochimica et biophysica acta, L. Lipids and lipid metabolism
INHIBITORY EFFECT OF A NEW UREIDOPHENOL DERIVATIVE T-2591 ON LDL OXIDATION AND ACAT ACTIVITY
Biological & pharmaceutical bulletin
INHIBITORY EFFECT OF MONATEPIL MALEATE ON ACYL-COA-CHOLESTEROL ACYLTRANSFERASE ACTIVITY IN THE LIVER OF CHOLESTEROL-FED JAPANESE MONKEYS
American journal of hypertension
EXOGENOUSLY HYPERCHOLESTEROLEMIC RATS, COMPARED WITH THEIR PROGENITORSPRAGUE-DAWLEY RATS, HAVE ALTERED MESSENGER-RNAS FOR CHOLESTEROL 7-ALPHA-HYDROXYLASE AND LOW-DENSITY-LIPOPROTEIN RECEPTOR AND ACTIVITIES OFCHOLESTEROL 7-ALPHA-HYDROXYLASE AND ACYL-COA - CHOLESTEROL ACYLTRANSFERASE IN THE LIVER IN RESPONSE TO DIETARY-CHOLESTEROL
Comparative biochemistry and physiology. B. Comparative biochemistry
EFFECTS OF FR145237, AN ACYL-COA-CHOLESTEROL ACYLTRANSFERASE INHIBITOR, ON DIET-INDUCED HYPERCHOLESTEROLEMIA IN DIABETIC RATS
Life sciences
POTENT HYPOCHOLESTEROLEMIC ACTIVITY OF NOVEL UREIDO PHENOXYISOBUTYRATES CORRELATES WITH THEIR INTRINSIC FIBRATE POTENCY AND NOT WITH THEIR ACAT INHIBITORY ACTIVITY
Journal of lipid research
PHARMACOLOGICAL PROPERTIES OF YM17E, AN ACYL-COA-CHOLESTEROL ACYLTRANSFERASE INHIBITOR, AND DIARRHEAL EFFECT IN BEAGLE DOGS
Japanese Journal of Pharmacology
ACTIVATION OF ACYL-COA - CHOLESTEROL ACYLTRANSFERASE IN RAT-LIVER MICROSOMES BY 25-HYDROXYCHOLESTEROL
Biochemical pharmacology
ACYL-COA-BINDING PROTEIN (ACBP) REGULATES ACYL-COA-CHOLESTEROL ACYLTRANSFERASE (ACAT) IN HUMAN MONONUCLEAR PHAGOCYTES
Biochimica et biophysica acta, L. Lipids and lipid metabolism
THE HYPOLIPIDEMIC ACTION OF THE ACAT INHIBITOR HL-004 IN HAMSTERS FEDNORMAL CHOW
General pharmacology
EFFECT OF ETHANOL ON THE SYNTHESIS AND SECRETION OF APOA-I-CONTAININGAND APO-B-CONTAINING LIPOPROTEINS IN HEPG2 CELLS
Journal of lipid research
ANTIATHEROSCLEROTIC EFFECT OF E5324, AN INHIBITOR OF ACYL-COA-CHOLESTEROL ACYLTRANSFERASE, IN WATANABE HERITABLE HYPERLIPIDEMIC RABBITS
Atherosclerosis
PLASMA-CHOLESTEROL REDUCING EFFECT OF FR129169, A NOVEL ACYL-COA-CHOLESTEROL ACYLTRANSFERASE INHIBITOR, IN THE RAT
Japanese Journal of Pharmacology
2 NEW MONOTERPENE GLYCOSIDES FROM KU-DING-CHA - INHIBITORS OF ACYL-COA - CHOLESTEROL ACYLTRANSFERASE (ACAT)
Chemical and Pharmaceutical Bulletin
HYPOLIPEMIC PROPERTIES OF A POTENT AND BIOAVAILABLE ALKLYSULFINYL-DIPHENYLIMIDAZOLE ACAT INHIBITOR (RP-73163) IN ANIMALS FED DIETS LOW IN CHOLESTEROL
Biochemical pharmacology
CHOLESTEROL ESTERIFICATION IS NOT ESSENTIAL FOR SECRETION OF LIPOPROTEIN COMPONENTS BY HEPG2 CELLS
Biochimica et biophysica acta, L. Lipids and lipid metabolism
GENETIC-DIFFERENCES OF LIPID-METABOLISM IN MACROPHAGES FROM C57BL 6J AND C3H/HEN MICE/
Arteriosclerosis, thrombosis, and vascular biology
CHOLESTEROL-LOWERING EFFECT OF AN ACYL-COENZYME-A - CHOLESTEROL ACYLTRANSFERASE INHIBITOR, FR145237, IN HYPERCHOLESTEROLEMIC RABBITS FED A HIGH-CHOLESTEROL DIET AND A CHOLESTEROL-FREE CASEIN DIET
Drug development research
BIOCHEMICAL-ALTERATIONS IN GUINEA-PIG ADRENAL-CORTEX FOLLOWING ADMINISTRATION OF PD-132301-2, AN INHIBITOR OF ACYL-COA-CHOLESTEROL ACYLTRANSFERASE
Life sciences
TMP-153, A NOVEL ACAT INHIBITOR, INHIBITS CHOLESTEROL ABSORPTION AND LOWERS PLASMA-CHOLESTEROL IN RATS AND HAMSTERS
Atherosclerosis
HYPOCHOLESTEROLEMIC ACTION AND PREVENTION OF CHOLESTEROL ABSORPTION VIA THE GUT BY F-1394, A POTENT ACYL-COA-CHOLESTEROL ACYLTRANSFERASE (ACAT) INHIBITOR, IN CHOLESTEROL DIET-FED RATS
Japanese Journal of Pharmacology
EFFECT OF E5324, A NOVEL INHIBITOR OF ACYL-COA-CHOLESTEROL ACYLTRANSFERASE, ON CHOLESTERYL ESTER SYNTHESIS AND ACCUMULATION IN MACROPHAGES
Japanese Journal of Pharmacology
STUDIES ON ACYL-COA-CHOLESTEROL ACYLTRANSFERASE (ACAT) INHIBITORY EFFECTS AND ENZYME SELECTIVITY OF F-1394, A PANTOTHEIC ACID-DERIVATIVE
Japanese Journal of Pharmacology
EFFECT OF FR145237, A NOVEL ACAT INHIBITOR, ON ATHEROGENESIS IN CHOLESTEROL-FED AND WHHL RABBITS - EVIDENCE FOR A DIRECT EFFECT ON THE ARTERIAL-WALL
Biochimica et biophysica acta, L. Lipids and lipid metabolism
EFFECT OF MEMBRANE ENVIRONMENT ON INHIBITION OF ACYL-COA-CHOLESTEROL ACYLTRANSFERASE BY A RANGE OF SYNTHETIC INHIBITORS
Biochimica et biophysica acta, L. Lipids and lipid metabolism
INHIBITION OF ACYL-COA-CHOLESTEROL ACYLTRANSFERASE IN CHINESE-HAMSTEROVARY (CHO) CELLS BY SHORT-CHAIN CERAMIDE AND DIHYDROCERAMIDE
Biochimica et biophysica acta, L. Lipids and lipid metabolism
GUAR-GUM EFFECTS ON PLASMA LOW-DENSITY-LIPOPROTEIN AND HEPATIC CHOLESTEROL-METABOLISM IN GUINEA-PIGS FED LOW-CHOLESTEROL AND HIGH-CHOLESTEROL DIETS - A DOSE-RESPONSE STUDY
The American journal of clinical nutrition
IMIDAZOLYLBENZOPYRANE DERIVATIVES - A NEW CLASS OF ACYL-COA - CHOLESTEROL ACYLTRANFERASE (ACAT) INHIBITORS
Journal of enzyme inhibition
PRICKLY PEAR (OPUNTIA SP) PECTIN ALTERS HEPATIC CHOLESTEROL-METABOLISM WITHOUT AFFECTING CHOLESTEROL ABSORPTION IN GUINEA-PIGS FED A HYPERCHOLESTEROLEMIC DIET
The Journal of nutrition
DIETARY-FAT SATURATION AND CHAIN-LENGTH MODULATE GUINEA-PIG HEPATIC CHOLESTEROL-METABOLISM
The Journal of nutrition
LACK OF REQUIREMENT FOR STEROL CARRIER PROTEIN-2 IN THE INTRACELLULARTRAFFICKING OF LYSOSOMAL CHOLESTEROL
Journal of lipid research
EFFECTS OF SUPPLEMENTING WITH VITAMIN-E ON THE UPTAKE OF LOW-DENSITY-LIPOPROTEIN AND THE STIMULATION OF CHOLESTERYL ESTER FORMATION IN MACROPHAGES
Atherosclerosis
EFFECT OF THE ACYL-COA-CHOLESTEROL ACYLTRANSFERASE INHIBITOR, E5324, ON EXPERIMENTAL ATHEROSCLEROSIS IN RABBITS
Atherosclerosis
COMPARISON OF THE EFFECT OF HYPERINSULINEMIA ON ACYL-COA-CHOLESTEROL ACYLTRANSFERASE ACTIVITY IN THE LIVER AND INTESTINE OF THE RAT
Atherosclerosis
HYPOCHOLESTEROLEMIC PROPERTIES OF PLANT INDOLES - INHIBITION OF ACYL-COA-CHOLESTEROL ACYLTRANSFERASE ACTIVITY AND REDUCTION OF SERUM LDL VLDL CHOLESTEROL LEVELS BY GLUCOBRASSICIN DERIVATIVES/
Biochemical pharmacology
CITRUS PECTIN AND CHOLESTEROL INTERACT TO REGULATE HEPATIC CHOLESTEROL HOMEOSTASIS AND LIPOPROTEIN METABOLISM - A DOSE-RESPONSE STUDY IN GUINEA-PIGS
The American journal of clinical nutrition
REGULATION OF LOW-DENSITY-LIPOPROTEIN RECEPTOR AND 3-HYDROXY-3-METHYL-GLUTARYL-COA REDUCTASE ACTIVITIES ARE DIFFERENTIALLY AFFECTED IN NIEMANN-PICK TYPE-C AND TYPE-D FIBROBLASTS
Biochemistry and cell biology
THE LIPID-LOWERING EFFECTS OF RHUBARB STALK FIBER - A NEW SOURCE OF DIETARY FIBER
Nutrition research
IMPORTANCE OF EXOGENOUS CHOLESTEROL IN DIABETIC RATS - EFFECTS OF TREATMENT WITH INSULIN OR WITH AN ACYL-COA-CHOLESTEROL ACYLTRANSFERASE INHIBITOR
Annals of nutrition & metabolism
SPHINGOSINE INHIBITS SPHINGOMYELINASE-INDUCED CHOLESTERYL ESTER FORMATION IN CULTURED FIBROBLASTS
Biochimica et biophysica acta
STIMULATION OF ACYL-COA-CHOLESTEROL ACYLTRANSFERASE ACTIVITY BY BREFELDIN-A IN MACROPHAGE J774 CELLS
Biochimica et biophysica acta