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Comparison of [F-18]altanserin and [F-18]deuteroaltanserin for PET imagingof serotonin(2A) receptors in baboon brain: pharmacological studies
NUCLEAR MEDICINE AND BIOLOGY
Melatonin protects against the effects of chronic stress on sexual behaviour in male rats
NEUROREPORT
Reproducibility of in vivo brain measures of 5-HT2A receptors with PET and[F-18]deuteroaltanserin
PSYCHIATRY RESEARCH-NEUROIMAGING
Apomorphine-induced aggressive behaviour in para-chlorophenylalanine-treated male rats: Implications to brain [H-3]Ketanserin binding and monoamine content
PHARMACOLOGY & TOXICOLOGY
Role of 5-HT2A and 5-HT2B/2C receptors in the behavioral interactions between serotonin and catecholamine reuptake inhibitors
NEUROPSYCHOPHARMACOLOGY
Analyses of [F-18]altanserin bolus injection PET data. II: Consideration of radiolabeled metabolites in humans
SYNAPSE
Different receptor subtypes are involved tn the serotonin-induced modulation of epileptiform activity in rat frontal cortex in vitro
JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY
A major role for thalamocortical afferents in serotonergic hallucinogen receptor function in the rat neocortex
NEUROSCIENCE
Serotonin-2A-receptor and -transporter polymorphisms: lack of association in patients with major depression
NEUROSCIENCE LETTERS
Involvement of adenosine in the effect of antidepressants on glutamate andaspartate release in the rat prefrontal cortex
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY
Cardiovascular effects of SL65.0472, a 5-HT receptor antagonist
EUROPEAN JOURNAL OF PHARMACOLOGY
Evidence for 5-HT1B/1D and 5-HT2A receptors mediating constriction of the canine internal carotid circulation
BRITISH JOURNAL OF PHARMACOLOGY
In-vivo assessment of 5-HT2A and 5-HT2C antagonistic properties of newer antipsychotics
BEHAVIOURAL PHARMACOLOGY
Behavioral evidence for interactions between a hallucinogenic drug and group II metabotropic glutamate receptors
NEUROPSYCHOPHARMACOLOGY
Agonist high and low affinity state ratios predict drug intrinsic activityand a revised ternary complex mechanism at serotonin 5-HT2A and 5-HT2C receptors
SYNAPSE
The role of serotonin in hot flushes
MATURITAS
Kinetic analysis of the 5-HT2A ligand [C-11]MDL 100,907
JOURNAL OF CEREBRAL BLOOD FLOW AND METABOLISM
Measurement of striatal and extrastriatal dopamine D-1 receptor binding potential with [C-11]NNC 112 in humans: Validation and reproducibility
JOURNAL OF CEREBRAL BLOOD FLOW AND METABOLISM
Serotonergic modulation of ethanol-induced electrophysiological depressionin young and aged rats
ALCOHOLISM-CLINICAL AND EXPERIMENTAL RESEARCH
Melatonin enhances sexual behavior in the male rat
PHYSIOLOGY & BEHAVIOR
Activation of 5-HT2A receptors impairs response control of rats in a five-choice serial reaction time task
NEUROPHARMACOLOGY
Serotonergic mechanisms involved in the attentional and vigilance task performance of rats and the palliative action of aniracetam
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY
ALEPH-2, a suspected anxiolytic and putative hallucinogenic phenylisopropylamine derivative, is a 5-HT2a and 5-HT2c receptor agonist
LIFE SCIENCES
S18327 (1-{2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)piperid-1-yl]ethyl}3-phenyl imidazolin-2-one), a novel, potential antipsychotic displaying marked antagonist properties at alpha(1) and alpha(2)-adrenergic receptors: I. Receptorial, neurochemical, and electrophysiological profile
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Role of striatal serotonin(2A) and serotonin(2C) receptor subtypes in the control of in vivo dopamine outflow in the rat striatum
JOURNAL OF NEUROCHEMISTRY
Ketanserin reverses dizocilpine-suppression of morphine dependence but nottolerance in mice
BRAIN RESEARCH
Induction of a high-affinity ketanserin binding site at the 5-hydroxytryptamine(1B) receptor by modification of its carboxy-terminal intracellular portion
BIOCHEMICAL PHARMACOLOGY
The T102C polymorphism of the 5-HT2A-receptor gene in fibromyalgia
NEUROBIOLOGY OF DISEASE
LSD and DOB: interaction with 5-HT2A receptors to inhibit NMDA receptor-mediated transmission in the rat prefrontal cortex
EUROPEAN JOURNAL OF NEUROSCIENCE
Serotonin-glutamate interactions: A new target for antipsychotic drugs
NEUROPSYCHOPHARMACOLOGY
Serotonin and hallucinogens
NEUROPSYCHOPHARMACOLOGY
PET studies of binding competition between endogenous dopamine and the D-1radiotracer [C-11]NNC 756
SYNAPSE
Apomorphine-induced upregulation of serotonin 5-HT2A receptors in male rats is independent from development of aggressive behaviour
JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY
[H-3]-ketanserin binding and elevated plus-maze behavior after chronic antidepressant treatment in DSP-4 and P-CPA pretreated rats: Evidence for partial involvement of 5-HT2A receptors
METHODS AND FINDINGS IN EXPERIMENTAL AND CLINICAL PHARMACOLOGY
Dopamine and serotonin interactions in the modulation of the expression ofthe immediate-early transcription factor, nerve growth factor-inducible B,in the striatum
NEUROSCIENCE
Binding affinity of sarpogrelate to 5-HT2A receptor ligand recognition sites in rat renal cortical and mesangial cells in culture
GENERAL PHARMACOLOGY
Pharmacological characteristics and regulation of 5-HT receptor-stimulatedphosphoinositide hydrolysis in the rat spinal cord
GENERAL PHARMACOLOGY
The influence of gender and page on neonatal rat hypothalamic 5-HT1A and 5-HT2A receptors
CELLULAR AND MOLECULAR NEUROBIOLOGY
c-Fos proteins, induced by the serotonin receptor agonist DOI, are not expressed in 5-HT2A positive cortical neurons
MOLECULAR BRAIN RESEARCH
Involvement of the serotonergic neuronal system in phencyclidine-induced place aversion in rats
BEHAVIOURAL BRAIN RESEARCH
Serotonin(2A) receptor modulation of D-1 dopamine receptor-mediated grooming behavior
PHARMACOLOGY BIOCHEMISTRY AND BEHAVIOR
The effects of the peptide-coupling agent, EEDQ, on 5-HT2A receptor binding and function in rat frontal cortex
NEUROPHARMACOLOGY
Role of serotonin(2A) and serotonin(2B/2C) receptor subtypes in the control of accumbal and striatal dopamine release elicited in vivo by dorsal raphe nucleus electrical stimulation
JOURNAL OF NEUROCHEMISTRY
Conformationally restricted butyrophenones with mixed dopaminergic (D-2) and serotoninergic (5-MT2A) affinities. Synthesis of 5-aminoethyl- and 6-aminomethyl-4-oxotetrahydroindoles as potential atypical antipsychotics
CHEMICAL & PHARMACEUTICAL BULLETIN
Behavioural pharmacology of the new generation of antipsychotic agents
BRITISH JOURNAL OF PSYCHIATRY
Evidence for a role for central 5-HT2B as well as 5-HT2A receptors in cardiovascular regulation in anaesthetized rats
BRITISH JOURNAL OF PHARMACOLOGY
5-hydroxytryptamine receptors mediating contraction in human small muscular pulmonary arteries: importance of the 5-HT1B receptor
BRITISH JOURNAL OF PHARMACOLOGY
Functional characterization and m-RNA expression of 5-HT receptors mediating contraction in human umbilical artery
BRITISH JOURNAL OF PHARMACOLOGY
Electrophysiological examination of the effects of sustained flibanserin administration on serotonin receptors in rat brain
BRITISH JOURNAL OF PHARMACOLOGY
Prolactin response to d-fenfluramine in major depression before and after treatment with serotonin reuptake inhibitors
BIOLOGICAL PSYCHIATRY
Regional changes in 5-HT1A but not in 5-HT2A receptors in mouse brain after Semliki Forest virus infection: radioligand binding and autoradiographic studies
JOURNAL OF NEUROVIROLOGY
ON THE RELATIONSHIP OF 5-HYDROXYTRYPTAMINE NEURONS TO 5-HYDROXYTRYPTAMINE 2A RECEPTOR-IMMUNOREACTIVE NEURONAL PROCESSES IN THE BRAIN-STEM OF RATS - A DOUBLE IMMUNOLABELING ANALYSIS
NeuroReport
M100907 AND CLOZAPINE, BUT NOT HALOPERIDOL OR RACLOPRIDE, PREVENT PHENCYCLIDINE-INDUCED BLOCKADE OF NMDA RESPONSES IN PYRAMIDAL NEURONS OF THE RAT MEDIAL PREFRONTAL CORTICAL SLICE
Neuropsychopharmacology
I-123-5-I-R91150, a new single-photon emission tomography ligand for 5-HT2A receptors: influence of age and gender in healthy subjects
EUROPEAN JOURNAL OF NUCLEAR MEDICINE
DIFFERENTIAL-EFFECTS OF NEONATAL HANDLING ON ANXIETY, CORTICOSTERONE RESPONSE TO STRESS, AND HIPPOCAMPAL GLUCOCORTICOID AND SEROTONIN (5-HT)(2A) RECEPTORS IN LEWIS RATS
Psychoneuroendocrinology
LOCALIZATION AND PHARMACOLOGICAL CHARACTERIZATION OF [H-3]PEROSPIRONE-BINDING SITES IN RAT-BRAIN
General pharmacology
AMPEROZIDE INFLUENCES FEEDING INDEPENDENTLY OF 5-HT2A RECEPTOR ANTAGONISM
Neuropsychobiology
POSITRON EMISSION TOMOGRAPHIC ANALYSIS OF DOSE-DEPENDENT MDL-100,907 BINDING TO 5-HYDROXYTRYPTAMINE-2A RECEPTORS IN THE HUMAN BRAIN
Journal of clinical psychopharmacology
STIMULATION OF 5-HT2A RECEPTORS ON ASTROCYTES IN PRIMARY CULTURE OPENS VOLTAGE-INDEPENDENT CA2+ CHANNELS
Neurochemistry international
ACTION OF THE 5-HT2A ANTAGONIST AMPEROZIDE ON ALCOHOL-INDUCED POIKILOTHERMIA IN RATS
Pharmacology, biochemistry and behavior
EFFECTS OF HOUSING CONDITIONS AND 5-HT2A ACTIVATION ON MALE-RAT SEXUAL-BEHAVIOR
Physiology & behavior
I-123 MSP AND F[C-11]MSP - NEW SELECTIVE 5-HT2A RECEPTOR RADIOPHARMACEUTICALS FOR IN-VIVO STUDIES OF NEURONAL 5-HT2 SEROTONIN RECEPTORS - SYNTHESIS, IN-VITRO BINDING STUDY WITH UNLABELED ANALOGS AND PRELIMINARY IN-VIVO EVALUATION IN MICE
Life sciences (1973)
REGULATION OF SEROTONIN(2A) RECEPTOR EXPRESSION BY AN ANTISENSE OLIGODEOXYNUCLEOTIDE
Journal of neurochemistry
CHRONIC IMIPRAMINE ADMINISTRATION AMPLIFIES THE SEROTONIN(2A) RECEPTOR-INDUCED INTRACELLULAR CA2-CELLS THROUGH A CALMODULIN-DEPENDENT PATHWAY( MOBILIZATION IN C6 GLIOMA)
Journal of neurochemistry
ANALYSIS OF THE 5-HT1A RECEPTOR INVOLVEMENT IN PASSIVE-AVOIDANCE IN THE RAT
British Journal of Pharmacology
THE ROLE OF 5-HT RECEPTOR SUBTYPES IN THE ANXIOLYTIC EFFECTS OF SELECTIVE SEROTONIN REUPTAKE INHIBITORS IN THE RAT ULTRASONIC VOCALIZATION TEST
Psychopharmacology
AUTORADIOGRAPHIC MAPPING OF BRAIN 5-HT2A BINDING-SITES IN P AND IN AAALCOHOL-PREFERRING RATS
Brain research bulletin
RECEPTOR-BINDING PROFILE AND ANXIOLYTIC-TYPE ACTIVITY OF DERAMCICLANE(EGIS-3886) IN ANIMAL-MODELS
Drug development research
PLATELET SEROTONERGIC INDEXES IN MAJOR DEPRESSION - UP-REGULATION OF 5-HT2A RECEPTORS UNCHANGED BY ANTIDEPRESSANT TREATMENT
Psychiatry research
EFFECTS OF CHRONIC ETHANOL-CONSUMPTION AND AGING ON 5-HT2A RECEPTORS AND 5-HT REUPTAKE SITES
Alcoholism, clinical and experimental research
SELECTIVE VISUALIZATION OF RAT-BRAIN 5-HT2A RECEPTORS BY AUTORADIOGRAPHY WITH [H-3] MDL-100,907
Naunyn-Schmiedeberg's archives of pharmacology
DEFICITS IN D-FENFLURAMINE-SENSITIVE POOL OF BRAIN 5-HT FOLLOWING WITHDRAWAL FROM CHRONIC COCAINE EXPOSURE
Life sciences
IN-VIVO REGULATION OF SEROTONIN 5-HT2A RECEPTORS IN RAT-BRAIN BY SUBCHRONIC ADMINISTRATION OF SIGMA-RECEPTOR LIGAND NE-100
Life sciences
PROTEIN-KINASE-C ACTIVATION BY SEROTONIN POTENTIATES AGONIST-INDUCED STIMULATION OF CAMP PRODUCTION IN CULTURED RAT RETINAL-PIGMENT EPITHELIAL-CELLS
Experimental Eye Research
REPEATED DOI AND SR 46349B TREATMENTS DO NOT AFFECT ELEVATED PLUS-MAZE ANXIETY DESPITE OPPOSITE EFFECTS ON CORTICAL 5-HT2A RECEPTORS
European journal of pharmacology
CHARACTERIZATION OF THE CONTRACTION TO 5-HT IN THE CANINE COLON LONGITUDINAL MUSCLE
British Journal of Pharmacology
VISUALIZATION OF LOSS OF 5-HT2A RECEPTORS WITH AGE IN HEALTHY-VOLUNTEERS USING [F-18] ALTANSERIN AND POSITRON EMISSION TOMOGRAPHIC IMAGING
PSYCHIATRY RESEARCH-NEUROIMAGING
DIFFERENTIAL EFFICACY OF SEROTONERGIC DRUGS FG5974, FG5893, AND AMPEROZIDE IN REDUCING ALCOHOL-DRINKING IN P-RATS
Alcohol
OPIATE AND 5-HT2A RECEPTORS IN ALCOHOL-DRINKING - PREFERENCE IN HAD RATS IS INHIBITED BY COMBINATION TREATMENT WITH NALTREXONE AND AMPEROZIDE
Alcohol
NATURALLY-OCCURRING CLAVINES - ANTAGONISM PARTIAL AGONISM AT 5-HT2A RECEPTORS AND ANTAGONISM AT ALPHA(1)-ADRENOCEPTORS IN BLOOD-VESSELS
Planta medica
PROTECTIVE ACTIONS OF THE 5-HT2A 2C, RECEPTOR AGONIST, DOI, ON 5-HT1ARECEPTOR-MEDIATED INHIBITION OF LORDOSIS BEHAVIOR/
Neuropharmacology
SEQUENTIAL ONSET OF 3 5-HT RECEPTORS DURING THE 5-HYDROXYTRYPTAMINERGIC DIFFERENTIATION OF THE MURINE 1C11 CELL-LINE
British Journal of Pharmacology
DESIPRAMINE ADMINISTRATION IN THE OLFACTORY BULBECTOMIZED RAT - CHANGES IN BRAIN BETA-ADRENOCEPTOR AND 5-HT2A BINDING-SITES AND THEIR RELATIONSHIP TO BEHAVIOR
British Journal of Pharmacology
PARTICIPATION OF 5-HT1-LIKE AND 5-HT2A RECEPTORS IN THE CONTRACTION OF HUMAN TEMPORAL ARTERY BY 5-HYDROXYTRYPTAMINE AND RELATED DRUGS
British Journal of Pharmacology
DOI DISRUPTION OF PREPULSE INHIBITION OF STARTLE IN THE RAT IS MEDIATED BY 5-HT2A AND NOT BY 5-HT2C RECEPTORS
Behavioural pharmacology
USE OF THE PITHED RAT MODEL TO DETERMINE THE RELATIVE POTENCIES OF 5-HT2A 2C RECEPTOR ANTAGONISTS FOLLOWING ACUTE INTRAVENOUS AND ORAL-ADMINISTRATION/
Methods and findings in experimental and clinical pharmacology
6-DI(HETEROARYL)-2-(N-METHYLPIPERAZINO)PYRIMIDINES AS NEW, POTENT 5-HT2A RECEPTOR LIGANDS - A VERIFICATION OF THE TOPOGRAPHIC MODEL
Archiv der pharmazie
SEROTONERGIC REGULATION OF ASSOCIATIVE LEARNING
Behavioural brain research
EVIDENCE THAT 5-HT2A RECEPTORS ARE NOT INVOLVED IN 5-HT-MEDIATED THERMOREGULATION IN MICE
Pharmacology, biochemistry and behavior
BIMT-17, A 5-HT1A RECEPTOR AGONIST 5-HT2A RECEPTOR ANTAGONIST, DIRECTLY ACTIVATES POSTSYNAPTIC 5-HT INHIBITORY RESPONSES IN THE RAT CEREBRAL-CORTEX
Naunyn-Schmiedeberg's archives of pharmacology
5-HT1-LIKE AND 5-HT2A RECEPTORS MEDIATE 5-HYDROXYTRYPTAMINE-INDUCED CONTRACTION OF RABBIT ISOLATED MESENTERIC-ARTERY
Naunyn-Schmiedeberg's archives of pharmacology
THE PHARMACOLOGY AND DISTRIBUTION OF HUMAN 5-HYDROXYTRYPTAMINE(2B) (5-HT2B) RECEPTOR GENE-PRODUCTS - COMPARISON WITH 5-HT2A AND 5-HT2C RECEPTORS
British Journal of Pharmacology
5-HYDROXYTRYPTAMINE RECEPTORS THAT FACILITATE EXCITATORY NEUROMUSCULAR-TRANSMISSION IN THE GUINEA-PIG ISOLATED DETRUSOR MUSCLE
British Journal of Pharmacology
CEREBRAL TRYPTOPHAN-HYDROXYLASE ACTIVITY, AND 5-HT1A RECEPTOR, 5-HT2A, RECEPTOR, AND 5-HT TRANSPORTER BINDING IN GROUPED AND ISOLATED ROMANRHA AND RLA RATS - RELATIONSHIPS WITH BEHAVIORS IN 2 MODELS OF ANXIETY
Psychopharmacology
LONG-LASTING EFFECTS OF AN ACUTE STRESS ON THE NEUROCHEMISTRY AND FUNCTION OF 5-HYDROXYTRYPTAMINERGIC NEURONS IN THE MOUSE-BRAIN
Psychopharmacology
EFFECT OF THE R(-) AND S(-CELLS EXPRESSING 5-HT2A OR 5-HT2C RECEPTORS() ISOMERS OF MDA AND MDMA ON PHOSPHOTIDYL INOSITOL TURNOVER IN CULTURED)
Neuroscience letters
IN-VIVO PROPERTIES OF SB 200646A, A 5-HT2C 2B RECEPTOR ANTAGONIST/
British Journal of Pharmacology