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Characterization of the molecular motions of constitutively active G protein-coupled receptors for parathyroid hormone
BIOPHYSICAL CHEMISTRY
Peptide hormone binding to G-protein-coupled receptors: Structural characterization via NMR techniques
MEDICINAL RESEARCH REVIEWS
Functional expression of M-1, M-3 and M-5 muscarinic acetylcholine receptors in yeast
JOURNAL OF NEUROCHEMISTRY
Photoaffinity labeling of mutant neurokinin-1 receptors reveals additionalstructural features of the substance P/NK-1 receptor complex
BIOCHEMISTRY
Studies on the structure of the G-protein-coupled receptor rhodopsin including the putative G-protein binding site in unactivated and activated forms
BIOCHEMISTRY
Thermal destabilization of rhodopsin and opsin by proteolytic cleavage in bovine rod outer segment disk membranes
BIOCHEMISTRY
Life history and developmental processes in the basidiomycete Coprinus cinereus
MICROBIOLOGY AND MOLECULAR BIOLOGY REVIEWS
Three dimensional structure of the seventh transmembrane helical domain ofthe G-protein receptor, rhodopsin
MOLECULAR VISION
The C terminus of the Saccharomyces cerevisiae alpha-factor receptor contributes to the formation of preactivation complexes with its cognate G protein
MOLECULAR AND CELLULAR BIOLOGY
Domain approach to three-dimensional structure of rhodopsin using high-resolution nuclear magnetic resonance
VERTEBRATE PHOTOTRANSDUCTION AND THE VISUAL CYCLE, PART A
Lack of interaction in recombinant human FSH receptor and both TSAb and TSBAb
LIFE SCIENCES
Characterization of parathyroid hormone/receptor interactions: Structure of the first extracellular loop
BIOCHEMISTRY
Parathyroid hormone and parathyroid hormone-related protein: Model systemsfor the development of an osteoporosis therapy
CURRENT PHARMACEUTICAL DESIGN
Signaling pathways involved in thyroid hyperfunction and growth in Graves'disease
BIOCHIMIE
Regulation of opioid receptor activities
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Conserved extracellular cysteine pair in the M-3 muscarinic acetylcholine receptor is essential for proper receptor cell surface localization but notfor G protein coupling
JOURNAL OF NEUROCHEMISTRY
Expression and function of the gonadotropin-releasing hormone receptor aredependent on a conserved apolar amino acid in the third intracellular loop
JOURNAL OF BIOLOGICAL CHEMISTRY
Identification and molecular characterization of m3 muscarinic receptor dimers
JOURNAL OF BIOLOGICAL CHEMISTRY
Use of a disulfide cross-linking strategy to study muscarinic receptor structure and mechanisms of activation
JOURNAL OF BIOLOGICAL CHEMISTRY
U50,488H-induced internalization of the human kappa opioid receptor involves a beta-arrestin- and dynamin-dependent mechanism - kappa receptor internalization is not required for mitogen-activated protein kinase activation
JOURNAL OF BIOLOGICAL CHEMISTRY
Nonselective coupling of the human mu-opioid receptor to multiple inhibitory G-protein isoforms
EUROPEAN JOURNAL OF BIOCHEMISTRY
Structural characterization of peptide hormone/receptor interactions by NMR spectroscopy
BIOPOLYMERS
MECHANISMS GOVERNING THE ACTIVATION AND TRAFFICKING OF YEAST G-PROTEIN-COUPLED RECEPTORS
Molecular biology of the cell
TOXIC THYROID ADENOMA - ABSENCE OF DNA MUTATIONS OF THE TSH RECEPTOR AND GS-ALPHA
European journal of endocrinology
USE OF A G-PROTEIN-COUPLED RECEPTOR TO COMMUNICATE - A SUCCESS DURINGEVOLUTION
Comptes rendus de l'Academie des sciences. Serie 3, Sciences de la vie
Structural correlates for down-regulation of m1 and m2 muscarinic receptorsubtypes
BRAIN RESEARCH BULLETIN
STRUCTURE OF THE G-PROTEIN-COUPLED RECEPTOR, RHODOPSIN - A DOMAIN APPROACH
Biochemical Society transactions
DOMINANT-NEGATIVE MUTATIONS IN THE G-PROTEIN-COUPLED ALPHA-FACTOR RECEPTOR MAP TO THE EXTRACELLULAR ENDS OF THE TRANSMEMBRANE SEGMENTS
Molecular and cellular biology
CONTRASTING INTERNALIZATION KINETICS OF HUMAN AND CHICKEN GONADOTROPIN-RELEASING-HORMONE RECEPTORS MEDIATED BY C-TERMINAL TAIL
Journal of Endocrinology
THE 2ND INTRACELLULAR LOOP OF THE M5 MUSCARINIC RECEPTOR IS THE SWITCH WHICH ENABLES G-PROTEIN COUPLING
The Journal of biological chemistry
DELETIONS IN THE 3RD INTRACELLULAR LOOP OF THE THYROTROPIN RECEPTOR -A NEW MECHANISM FOR CONSTITUTIVE ACTIVATION
The Journal of biological chemistry
BINDING DOMAIN OF HUMAN PARATHYROID-HORMONE RECEPTOR - FROM CONFORMATION TO FUNCTION
Biochemistry (Easton)
STRUCTURE FUNCTION RELATIONSHIPS OF A G-PROTEIN COUPLING POCKET FORMED BY THE 3RD INTRACELLULAR LOOP OF THE M5 MUSCARINIC RECEPTOR/
Biochemistry
SIGNALING IN THE YEASTS - AN INFORMATIONAL CASCADE WITH LINKS TO THE FILAMENTOUS FUNGI
Microbiology and molecular biology reviews
PHEROMONE SIGNALING AND POLARIZED MORPHOGENESIS IN YEAST
Current opinion in genetics & development
HOW RECEPTORS TALK TO TRIMERIC G-PROTEINS
Current opinion in cell biology
GLYCOSYLATION VARIANTS OF HUMAN TSH SELECTIVELY ACTIVATE SIGNAL-TRANSDUCTION PATHWAYS
Molecular and cellular endocrinology
STRUCTURE FUNCTION RELATIONSHIPS OF CALCITONIN ANALOGS AS AGONISTS, ANTAGONISTS, OR INVERSE AGONISTS IN A CONSTITUTIVELY ACTIVATED RECEPTORCELL SYSTEM/
Molecular pharmacology
RESIDUES SPECIFICALLY INVOLVED IN DOWN-REGULATION BUT NOT INTERNALIZATION OF THE M1 MUSCARINIC ACETYLCHOLINE-RECEPTOR
Journal of neurochemistry
PHE(576) PLAYS AN IMPORTANT ROLE IN THE SECONDARY STRUCTURE AND INTRACELLULAR SIGNALING OF THE HUMAN LUTEINIZING-HORMONE CHORIONIC-GONADOTROPIN RECEPTOR
The Journal of clinical endocrinology and metabolism
CYCLOOXYGENASE-DEPENDENT THYROID-CELL PROLIFERATION INDUCED BY IMMUNOGLOBULINS FROM PATIENTS WITH GRAVES-DISEASE
The Journal of clinical endocrinology and metabolism
RANDOM MUTAGENESIS OF THE CAMP CHEMOATTRACTANT RECEPTOR, CAR1, OF DICTYOSTELIUM - EVIDENCE FOR MULTIPLE STATES OF ACTIVATION
The Journal of biological chemistry
INTERRUPTION OF G-PROTEIN-COUPLING IN CXCR2 DOES NOT ALTER LIGAND-BINDING, BUT ELIMINATES LIGAND-ACTIVATION OF GTP-GAMMA-S-35 BINDING, CALCIUM MOBILIZATION, AND CHEMOTAXIS
Biochemistry
TSH RECEPTOR AND LH RECEPTOR, 1996
Endocrine journal
AUTOIMMUNITY AND THYROID GROWTH - WHERE DO WE STAND
European journal of endocrinology
MONITORING THE TRANSFECTION EFFICIENCY OF THE HUMAN FOLLICLE-STIMULATING-HORMONE RECEPTOR CDNA IN COS-7 CELLS - EVALUATION OF THE GROWTH-HORMONE TRANSIENT GENE-EXPRESSION ASSAY SYSTEM
Journal of endocrinological investigation
MOLECULAR ARCHITECTURE OF G-PROTEIN-COUPLED RECEPTORS
Drug development research
AGONIST-SPECIFIC CONFORMATIONAL-CHANGES IN THE YEAST ALPHA-FACTOR PHEROMONE RECEPTOR
Molecular and cellular biology
ALANINE SCANNING MUTAGENESIS OF CONSERVED ARGININE LYSINE-ARGININE/LYSINE-X-X-ARGININE/LYSINE G-PROTEIN-ACTIVATING MOTIFS ON M1 MUSCARINIC ACETYLCHOLINE-RECEPTORS/
Molecular pharmacology
SEQUESTRATION OF THE SHORT AND LONG ISOFORMS OF DOPAMINE D-2 RECEPTORS EXPRESSED IN CHINESE-HAMSTER OVARY CELLS
Molecular pharmacology
INTERACTION OF THE COOH-TERMINAL DOMAIN OF THE NEUROTENSIN RECEPTOR WITH A G-PROTEIN DOES NOT CONTROL THE PHOSPHOLIPASE-C ACTIVATION BUT ISINVOLVED IN THE AGONIST-INDUCED INTERNALIZATION
Molecular pharmacology
SINGLE AMINO-ACID SUBSTITUTIONS IN THE PM2 MUSCARINIC RECEPTOR ALTER RECEPTOR G PROTEIN COUPLING WITHOUT CHANGING PHYSIOLOGICAL-RESPONSES/
Molecular pharmacology
EPITOPES FOR THYROID-STIMULATING ANTIBODIES IN GRAVES SERA - A POSSIBLE LINK OF HETEROGENEITY TO DIFFERENCES IN RESPONSE TO ANTITHYROID DRUG-TREATMENT
The Journal of clinical endocrinology and metabolism
IDENTIFICATION OF A REGION REQUIRED FOR SUBTYPE-SPECIFIC AGONIST-INDUCED SEQUESTRATION OF THE M2 MUSCARINIC ACETYLCHOLINE-RECEPTOR
The Journal of biological chemistry
HUMAN MUSCARINIC CHOLINERGIC RECEPTOR HM1 INTERNALIZES VIA CLATHRIN-COATED VESICLES
The Journal of biological chemistry
CONSTITUTIVE ACTIVATION OF CHIMERIC M2 M5 MUSCARINIC RECEPTORS AND DELINEATION OF G-PROTEIN COUPLING SELECTIVITY DOMAINS/
Biochemical pharmacology
CONSTITUTIVE ACTIVATION OF THE THYROTROPIN RECEPTOR BY MUTATING CYS-636 IN THE 6TH TRANSMEMBRANE SEGMENT
Biochemical and biophysical research communications
CYSTEINE-699, A POSSIBLE PALMITOYLATION SITE OF THE THYROTROPIN RECEPTOR, IS NOT CRUCIAL FOR CAMP OR PHOSPHOINOSITIDE SIGNALING BUT IS NECESSARY FOR FULL SURFACE EXPRESSION
Biochemical and biophysical research communications
CHARACTERIZATION OF HETEROGENEOUS MUTATIONS CAUSING CONSTITUTIVE ACTIVATION OF THE LUTEINIZING-HORMONE RECEPTOR IN FAMILIAL MALE PRECOCIOUSPUBERTY
Human molecular genetics
G PROTEIN-COUPLED RECEPTOR STRUCTURE AND FUNCTION - THE IMPACT OF DISEASE-CAUSING MUTATIONS
Bailliere's clinical endocrinology and metabolism
RECEPTORS AND G-PROTEINS AS PRIMARY COMPONENTS OF TRANSMEMBRANE SIGNAL-TRANSDUCTION .1. G-PROTEIN-COUPLED RECEPTORS - STRUCTURE AND FUNCTION
Journal of molecular medicine
CHOLECYSTOKININ AND GASTRIN ARE NOT EQUALLY SENSITIVE TO GTP-GAMMA-S AT CCKB RECEPTORS - IMPORTANCE OF THE SULFATED TYROSINE
European journal of pharmacology. Molecular pharmacology section
TSH RECEPTOR AND LH RECEPTOR, 1995
Endocrine journal
MOLECULAR-BASIS OF THE FUNCTIONAL COUPLIN G OF RECEPTORS TO GTP-BINDING PROTEINS
Biologiceskie membrany
MUTATION OF CARBOXYL-TERMINAL THREONINE RESIDUES IN HUMAN M3 MUSCARINIC ACETYLCHOLINE-RECEPTOR MODULATES THE EXTENT OF SEQUESTRATION AND DESENSITIZATION
Molecular pharmacology
SUBGROUPS OF GRAVES PATIENTS IDENTIFIED ON THE BASIS OF THE BIOCHEMICAL ACTIVITIES OF THEIR IMMUNOGLOBULINS
The Journal of clinical endocrinology and metabolism
A NOVEL MUTATION OF THE LUTEINIZING-HORMONE RECEPTOR GENE CAUSING MALE GONADOTROPIN-INDEPENDENT PRECOCIOUS PUBERTY
The Journal of clinical endocrinology and metabolism
A NEW CONSTITUTIVELY ACTIVATING POINT MUTATION IN THE LUTEINIZING-HORMONE CHORIOGONADOTROPIN RECEPTOR GENE IN CASES OF MALE-LIMITED PRECOCIOUS PUBERTY
The Journal of clinical endocrinology and metabolism
GENETIC ALTERATIONS IN THYROID HYPERFUNCTIONING ADENOMAS
The Journal of clinical endocrinology and metabolism
STRUCTURE-FUNCTION OF MUSCARINIC RECEPTOR COUPLING TO G-PROTEINS - RANDOM SATURATION MUTAGENESIS IDENTIFIES A CRITICAL DETERMINANT OF RECEPTOR AFFINITY FOR G-PROTEINS
The Journal of biological chemistry
ACTIVATING AND INACTIVATING MUTATIONS IN N-TERMINAL AND C-TERMINAL I3LOOP JUNCTIONS OF MUSCARINIC ACETYLCHOLINE HM1 RECEPTORS
The Journal of biological chemistry
CONSTITUTIVE ACTIVATION OF THE THYROTROPIN RECEPTOR BY DELETION OF A PORTION OF THE EXTRACELLULAR DOMAIN
Biochemical and biophysical research communications
THYROTROPIN STIMULATION OF THE LUTROPIN CHORIOGONADOTROPIN RECEPTOR -DIFFERENT SITES MEDIATE AGONIST ACTIVITY AND HIGH-AFFINITY BINDING/
Thyroid
INSERTION MUTAGENESIS AS A TOOL TO PREDICT THE SECONDARY STRUCTURE OFA MUSCARINIC RECEPTOR DOMAIN DETERMINING SPECIFICITY OF G-PROTEIN COUPLING
Proceedings of the National Academy of Sciences of the United Statesof America
DELETION MUTATION IN THE PUTATIVE 3RD INTRACELLULAR LOOP OF THE RAT NEUROTENSIN RECEPTOR ABOLISHES POLYPHOSPHOINOSITIDE HYDROLYSIS BUT NOT CYCLIC-AMP FORMATION IN CHO-K1 CELLS
Molecular pharmacology
INTERNALIZATION OF THE GASTRIN-RELEASING PEPTIDE RECEPTOR IS MEDIATEDBY BOTH PHOSPHOLIPASE C-DEPENDENT AND C-INDEPENDENT PROCESSES
Molecular pharmacology
DISRUPTION OF THE FIRST EXTRACELLULAR LOOP OF THYROTROPIN RECEPTOR PREVENTS LIGAND-BINDING
Life sciences
A SPORADIC CASE OF MALE-LIMITED PRECOCIOUS PUBERTY HAS THE SAME CONSTITUTIVELY ACTIVATING POINT MUTATION IN LUTEINIZING-HORMONE CHORIOGONADOTROPIN RECEPTOR GENE AS FAMILIAL CASES
The Journal of clinical endocrinology and metabolism
OVERLAPPING MULTISITE DOMAINS OF THE MUSCARINIC CHOLINERGIC HM1 RECEPTOR INVOLVED IN SIGNAL-TRANSDUCTION AND SEQUESTRATION
The Journal of biological chemistry
SEQUESTRATION OF MUSCARINIC ACETYLCHOLINE-RECEPTOR M2 SUBTYPES - FACILITATION BY G-PROTEIN-COUPLED RECEPTOR KINASE (GRK2) AND ATTENUATION BY A DOMINANT-NEGATIVE MUTANT OF GRK2
The Journal of biological chemistry
IDENTIFICATION OF AN INTRACELLULAR TYROSINE RESIDUE CRITICAL FOR MUSCARINIC RECEPTOR-MEDIATED STIMULATION OF PHOSPHATIDYLINOSITOL HYDROLYSIS
The Journal of biological chemistry
CONSTITUTIVE ACTIVATION OF CYCLIC-AMP BUT NOT PHOSPHATIDYLINOSITOL SIGNALING CAUSED BY 4 MUTATIONS IN THE 6TH TRANSMEMBRANE HELIX OF THE HUMAN THYROTROPIN RECEPTOR
FEBS letters
THE 3RD EXOPLASMIC LOOP OF THE THYROTROPIN RECEPTOR IS PARTIALLY INVOLVED IN SIGNAL-TRANSDUCTION
FEBS letters
DELETION ANALYSIS OF THE M4 MUSCARINIC ACETYLCHOLINE-RECEPTOR - MOLECULAR DETERMINANTS FOR ACTIVATION OF BUT NOT COUPLING TO THE G(I) GUANINE-NUCLEOTIDE-BINDING REGULATORY PROTEIN REGULATE RECEPTOR INTERNALIZATION
European journal of biochemistry
AGONIST-INDUCED MUSCARINIC CHOLINERGIC RECEPTOR INTERNALIZATION, RECYCLING AND DEGRADATION IN CULTURED NEURONAL CELLS - CELLULAR MECHANISMSAND ROLE IN DESENSITIZATION
Biochemical pharmacology
THE INTRACELLULAR REGION ADJACENT TO PLASMA-MEMBRANE (RESIDUES 684-692) OF THE THYROTROPIN RECEPTOR IS IMPORTANT FOR PHOSPHOINOSITIDE SIGNALING BUT NOT FOR AGONIST-INDUCED ADENYLATE-CYCLASE ACTIVATION
Biochemical and biophysical research communications
MUTATIONAL ANALYSIS OF MUSCARINIC ACETYLCHOLINE-RECEPTORS - STRUCTURAL BASIS OF LIGAND-RECEPTOR G-PROTEIN INTERACTIONS
Life sciences
HYDROPHOBIC AMINO-ACID IN THE I2-LOOP PLAYS A KEY ROLE IN RECEPTOR-G-PROTEIN COUPLING
The Journal of biological chemistry
MOLECULAR-BASIS OF MUSCARINIC ACETYLCHOLINE-RECEPTOR FUNCTION
Trends in pharmacological sciences