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In vitro and in vivo m2 muscarinic subtype selectivity of some dibenzodiazepinones and pyridobenzodiazepinones
BRAIN RESEARCH
Pharmacokinetic computer simulations of the relationship between in vivo and in vitro neuroreceptor subtype selectivity of radioligands
NUCLEAR MEDICINE AND BIOLOGY
IN-VIVO COMPETITION STUDIES OF Z-(-,-)-[I-125]IQNP AGAINST 3-QUINUCLIDINYL 2-(5-BROMOTHIENYL)-2-THIENYLGLYCOLATE (BRQNT) DEMONSTRATING IN-VIVO M2 MUSCARINIC SUBTYPE SELECTIVITY FOR BRQNT
Journal of molecular neuroscience
SYNTHESIS OF SOME SUBSTITUTED DIBENZODIAZEPINONES AND PYRIDOBENZODIAZEPINONES
Journal of heterocyclic chemistry
CORRECTION OF THE STEREOCHEMICAL ASSIGNMENT OF THE BENZILIC ACID CENTER IN (R)-(-)-3-QUINUCLIDINYL (S)-(-4-IODOBENZILATE [(R,S)-4-IQNB]())
Applied radiation and isotopes
IN-VIVO AUTORADIOGRAPHY OF RADIOIODINATED (R)-3-QUINUCLIDINYL (S)-4-IODOBENZILATE [(R,S)-IQNB] AND (R)-3-QUINUCLIDINYL (R)-4-IODOBENZILATE [(R,R)-IQNB] - COMPARISON OF THE RADIOLABELED PRODUCTS OF A NOVEL TRIBUTYLSTANNYL PRECURSOR WITH THOSE OF THE ESTABLISHED TRIAZENE AND EXCHANGE METHODS
Applied radiation and isotopes
PREPARATION AND CHARACTERIZATION OF (R,S)-[BR-76]BRQNB - AN ANALOG OFQNB FOR PET
Journal of labelled compounds & radiopharmaceuticals
AUTORADIOGRAPHIC EVIDENCE THAT 3-QUINUCLIDINYL-4-FLUOROBENZILATE (FQNB) DISPLAYS IN-VIVO SELECTIVITY FOR THE M2 SUBTYPE
NeuroImage
AUTORADIOGRAPHIC EVIDENCE THAT (R)-3-QUINUCLIDINYL (S)-4-FLUOROMETHYLBENZILATE ((R,S)-FMEQNB) DISPLAYS IN-VIVO SELECTIVITY FOR THE MUSCARINIC M2 SUBTYPE
Nuclear medicine and biology
SPECIFIC BINDING-COMPONENT OF THE INACTIVE STEREOISOMER (S,S)-[I-125]IQNB TO RAT-BRAIN MUSCARINIC RECEPTORS IN-VIVO
Nuclear medicine and biology
AUTORADIOGRAPHIC EVIDENCE THAT QUINUCLIDINYL 4-(BROMOPHENYL)-2-THIENYLGLYCOLATE (QBPTG) DISPLAYS IN-VIVO SELECTIVITY FOR THE MUSCARINIC M2 SUBTYPE
NeuroImage
AUTORADIOGRAPHIC EVIDENCE THAT QNB DISPLAYS IN-VIVO SELECTIVITY FOR THE M2 SUBTYPE
NeuroImage
COMPARISON OF THE IN-VIVO RAT-BRAIN REGIONAL PHARMACOKINETICS OF [H-3] QNB, (R,S)-[I-125]-4IQNB, AND (R,R)-[I-125]-4IQNB BINDING TO THE MUSCARINIC ACETYLCHOLINE-RECEPTOR IN RELATIONSHIP TO THE REGIONAL SUBTYPECOMPOSITION
Receptor
THEORETICAL RELATIONSHIPS OF RECEPTOR AND DELIVERY SENSITIVITIES AND MEASURABLE PARAMETERS IN IN-VIVO NEURORECEPTOR-RADIOLIGAND INTERACTIONS
IEEE transactions on medical imaging
NOVEL POTENT AND M(2)-SELECTIVE ANTIMUSCARINIC COMPOUNDS WHICH PENETRATE THE BLOOD-BRAIN-BARRIER
European journal of medicinal chemistry
CHARACTERIZATION OF IN-VIVO BRAIN MUSCARINIC ACETYLCHOLINE-RECEPTOR SUBTYPE SELECTIVITY BY COMPETITION STUDIES AGAINST (R,S)-[I-125]IQNB (VOL 687, PG 71, 1995)
Brain research
CHARACTERIZATION OF IN-VIVO BRAIN MUSCARINIC ACETYLCHOLINE-RECEPTOR SUBTYPE SELECTIVITY BY COMPETITION STUDIES AGAINST (R,S)-[I-125]IQNB
Brain research
GRAPHICAL ANALYSIS OF FLUOROALKYL QNB DEMONSTRATING IN-VIVO M2 MACHR SELECTIVITY
The Journal of nuclear medicine
[H-3] QNB DISPLAYS IN-VIVO SELECTIVITY FOR THE M2 SUBTYPE
Life sciences
SYNTHESIS OF SOME DIBENZODIAZEPIONE DERIVATIVES AS POTENT AND M2-SELECTIVE ANTIMUSCARINIC COMPOUNDS
Journal of heterocyclic chemistry
ESTIMATION OF RELATIVE REGIONAL NEURORECEPTOR CONCENTRATION BY PET ORSPECT - THEORETICAL COMPARISONS OF USING A SINGLE LATE IMAGE OR A LATE PLUS EARLY IMAGE
IEEE transactions on medical imaging
EVALUATION OF RECONSTRUCTION ALGORITHMS IN SPECT NEUROIMAGING .1. COMPARISON OF STATISTICAL NOISE IN SPECT NEUROIMAGES WITH NAIVE AND REALISTIC PREDICTIONS
Physics in medicine and biology
EVALUATION OF RECONSTRUCTION ALGORITHMS IN SPECT NEUROIMAGING .2. COMPUTATION OF DETERMINISTIC AND STATISTICAL ERROR-COMPONENTS
Physics in medicine and biology
A NOVEL MUSCARINIC RECEPTOR-LIGAND WHICH PENETRATES THE BLOOD-BRAIN-BARRIER AND DISPLAYS IN-VIVO SELECTIVITY FOR THE M2 SUBTYPE
Life sciences