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Neurogenic inflammation in the context of migraine
MICROSCOPY RESEARCH AND TECHNIQUE
An orally active, water-soluble neurokinin-1 receptor antagonist suitable for both intravenous and oral clinical administration
JOURNAL OF MEDICINAL CHEMISTRY
The anti-migraine 5-HT1B/1D agonist rizatriptan inhibits neurogenic dural vasodilation in anaesthetized guinea-pigs
BRITISH JOURNAL OF PHARMACOLOGY
Role of opioid receptors in neurogenic dural vasodilation and sensitization of trigeminal neurones in anaesthetized rats
BRITISH JOURNAL OF PHARMACOLOGY
The history and pharmacology of ergotamine and dihydroergotamine
DRUG TREATMENT OF MIGRAINE AND OTHER HEADACHES
The pharmacology and mechanisms of action of rizatriptan
DRUG TREATMENT OF MIGRAINE AND OTHER HEADACHES
Pharmacology and potential mechanisms of action of rizatriptan
CEPHALALGIA
Localization of N-methyl-D-aspartate NR2B subunits on primary sensory neurons that give rise to small-caliber sciatic nerve fibers in rats
NEUROSCIENCE
The novel NK1 receptor antagonist MK-0869 (L-754,030) and its water soluble phosphoryl prodrug, L758,298, inhibit acute and delayed cisplatin-inducedemesis in ferrets
NEUROPHARMACOLOGY
Mechanisms of action of serotonin 5-HT1B/1D agonists: Insights into migraine pathophysiology using rizatriptan
NEUROLOGY
Pathophysiology of migraine - New insights
CANADIAN JOURNAL OF NEUROLOGICAL SCIENCES
Dural vasodilation causes a sensitization of rat caudal trigeminal neurones in vivo that is blocked by a 5-HT1B/1D agonist
BRITISH JOURNAL OF PHARMACOLOGY
Pathophysiology and pharmacology of migraine. Is there a place for antiemetics in future treatment strategies?
CEPHALALGIA
Differential effects of the 5HT(1B/1D) receptor agonist naratriptan on trigeminal versus spinal nociceptive responses
CEPHALALGIA
DISTINCT MECHANISM FOR ANTIDEPRESSANT ACTIVITY BY BLOCKADE OF CENTRALSUBSTANCE-P RECEPTORS
Science
SENSITIZATION OF CAUDAL TRIGEMINAL NEURONS BY DURAL ARTERY DILATATION
Neurology
The effects of 5-HT1A, 5-HT1B and 5-HT1D receptor agonists on trigeminal nociceptive neurotransmission in anaesthetized rats
EUROPEAN JOURNAL OF PHARMACOLOGY
RETINAL PLASMA EXTRAVASATION IN ANIMALS BUT NOT IN HUMANS - IMPLICATIONS FOR THE PATHOPHYSIOLOGY OF MIGRAINE
Brain (Print)
INTRAVITAL MICROSCOPE STUDIES ON THE EFFECTS OF NEUROKININ AGONISTS AND CALCITONIN-GENE-RELATED PEPTIDE ON DURAL VESSEL DIAMETER IN THE ANESTHETIZED RAT
Cephalalgia
SUMATRIPTAN INHIBITS NEUROGENIC VASODILATION OF DURAL BLOOD-VESSELS IN THE ANESTHETIZED RAT - INTRAVITAL MICROSCOPE STUDIES
Cephalalgia
DIFFERENTIAL-EFFECTS OF 5-HT1B 1D RECEPTOR AGONISTS ON NEUROGENIC DURAL PLASMA EXTRAVASATION AND VASODILATION IN ANESTHETIZED RATS/
Neuropharmacology
RIZATRIPTAN SHOWS CRANIOVASCULAR SELECTIVITY FOR HUMAN ISOLATED MIDDLE MENINGEAL OVER CORONARY-ARTERIES - A COMPARISON WITH SUMATRIPTAN
Neurology
RIZATRIPTAN INHIBITS NEUROGENIC DURAL VASODILATION - AN INTRAVITAL MICROSCOPE STUDY IN RATS
Neurology
TRIGEMINAL NEURONS THAT RECEIVE NONNOCICEPTIVE VIBRISSAL INPUT IN THEANESTHETIZED RAT - EFFECTS OF CONVERGENT NOCICEPTIVE INPUT FROM THE DURA-MATER AND OF A 5-HT1B 1D AGONIST/
Journal of physiology
RIZATRIPTAN HAS CENTRAL ANTINOCICEPTIVE EFFECTS AGAINST DURALLY EVOKED-RESPONSES
European journal of pharmacology
THE NOVEL ANTIMIGRAINE AGENT RIZATRIPTAN INHIBITS NEUROGENIC DURAL VASODILATION AND EXTRAVASATION
European journal of pharmacology
IN-VITRO AND IN-VIVO PREDICTORS OF THE ANTIEMETIC ACTIVITY OF TACHYKININ NK1 RECEPTOR ANTAGONISTS
European journal of pharmacology
NEUROKININ-RECEPTOR ANTAGONISTS - PHARMACOLOGICAL TOOLS AND THERAPEUTIC DRUGS
Canadian journal of physiology and pharmacology
RIZATRIPTAN INHIBITS TRIGEMINAL NOCICEPTIVE RESPONSES IN AN ELECTROPHYSIOLOGICAL ASSAY IN THE ANESTHETIZED RAT
British Journal of Pharmacology
PREDICTION OF THE ANTIEMETIC ACTIVITY OF NK1 RECEPTOR ANTAGONISTS IN FERRETS BY THEIR ABILITY TO INHIBIT GR73632-INDUCED FOOT TAPPING IN GERBILS
British Journal of Pharmacology
THE CHEMICAL EVOLUTION OF 2-[5-(1,2,4-TRIAZOL-4-YL)-1H-INDOL-3-YL]ETHYLAMINE (L-741,604) AND ANALOGS - POTENT AND SELECTIVE AGONISTS FOR 5-HT1D RECEPTORS
Bioorganic & medicinal chemistry letters
TACHYKININ NK1 RECEPTOR ANTAGONISTS ACT CENTRALLY TO INHIBIT EMESIS INDUCED BY THE CHEMOTHERAPEUTIC AGENT CISPLATIN IN FERRETS
Neuropharmacology
N-HETEROARYL-2-PHENYL-3-(BENZYLOXY)PIPERIDINES - A NOVEL CLASS OF POTENT ORALLY-ACTIVE HUMAN NK1 ANTAGONISTS
Journal of medicinal chemistry
L-733,060, A NOVEL TACHYKININ NK1 RECEPTOR ANTAGONIST - EFFECTS IN [CA2+](I) MOBILIZATION, CARDIOVASCULAR AND DURAL EXTRAVASATION ASSAYS
European journal of pharmacology
EFFECTS OF A PARTIAL AGONIST AND A FULL ANTAGONIST ACTING AT THE GLYCINE SITE OF THE NMDA RECEPTOR ON INFLAMMATION-INDUCED MECHANICAL HYPERALGESIA IN RATS
British Journal of Pharmacology
EFFECT OF THE NK1 RECEPTOR ANTAGONISTS, L-733,060 AND CP-99,994, AND MORPHINE IN THE RABBIT SPINAL REFLEX PREPARATION
British Journal of Pharmacology
STUDIES ON THE SYMPATHOLYTIC EFFECTS OF SOME 5-HT1D RECEPTOR AGONISTSIN PITHED RATS AND GUINEA-PIGS
British Journal of Pharmacology
DIRECT MEASUREMENT OF DURAL BLOOD-VESSEL DIAMETER IN THE RAT USING INTRAVITAL MICROSCOPY
British Journal of Pharmacology
ACIDIC FIBROBLAST GROWTH-FACTOR STIMULATES MOTOR AND SENSORY AXON REGENERATION AFTER SCIATIC-NERVE CRUSH IN THE RAT
Neuroscience
THE NEUROPROTECTIVE EFFECT OF THE GLYCINE SITE ANTAGONIST 3R-(-CIS-4-METHYL-HA966 (L-687,414) IN A RAT MODEL OF FOCAL ISCHEMIA())
Journal of cerebral blood flow and metabolism
CALCITONIN-GENE-RELATED PEPTIDE AS AN ENDOGENOUS VASODILATOR - IMMUNOBLOCKADE STUDIES IN-VIVO WITH AN ANTI-CALCITONIN GENE-RELATED PEPTIDE MONOCLONAL-ANTIBODY AND ITS FAB-'-FRAGMENT
Clinical science
COMPARISON OF THE EFFECTS OF SUMATRIPTAN AND THE NK1 ANTAGONIST CP-99,994 ON PLASMA EXTRAVASATION IN DURA-MATER AND C-FOS MESSENGER-RNA EXPRESSION IN TRIGEMINAL NUCLEUS CAUDALIS OF RATS
Neuropharmacology
ENANTIOSPECIFIC INHIBITION OF EMESIS INDUCED BY NICOTINE IN THE HOUSEMUSK SHREW (SUNCUS-MURINUS) BY THE NEUROKININ(1) (NK1) RECEPTOR ANTAGONIST CP-99,994
Neuropharmacology
SYNTHESIS AND SEROTONERGIC ACTIVITY OF HYL-2-[5-(1,2,4-TRIAZOL-1-YLMETHYL)-1H-INDOL-3-YL] ETHYLAMINE AND ANALOGS - POTENT AGONISTS FOR 5-HT1D RECEPTORS
Journal of medicinal chemistry
ENANTIOSELECTIVE INHIBITION OF APOMORPHINE-INDUCED EMESIS IN THE FERRET BY THE NEUROKININ(1) RECEPTOR ANTAGONIST CP-99,994
Neuropharmacology
BIOLOGICAL PROPERTIES OF THE BENZODIAZEPINE AMIDINE DERIVATIVE L-740,093, A CHOLECYSTOKININ-B GASTRIN RECEPTOR ANTAGONIST WITH HIGH-AFFINITY IN-VITRO AND HIGH POTENCY IN-VIVO
Molecular pharmacology
ACIDIC FIBROBLAST GROWTH-FACTOR (AFGF) STIMULATES RAT SCIATIC-NERVE REGENERATION AFTER A CRUSH INJURY
Journal of physiology
SYNTHESIS AND BIOLOGICAL-ACTIVITY OF ETHYL-1,2,5-THIADIAZOLIDIN-2-YL)-METHYL]-1H-INDOLE AND ANALOGS - AGONISTS FOR THE 5-HT1D RECEPTOR
Journal of medicinal chemistry
CALCITONIN-GENE-RELATED PEPTIDE (CGRP) AS AN ENDOGENOUS VASODILATOR -IN-VIVO IMMUNOBLOCKADES STUDIES WITH AN ANTI-CGRP MONOCLONAL-ANTIBODYAND ITS FAB' FRAGMENT
British Journal of Pharmacology
NEUROPROTECTIVE NMDA ANTAGONISTS - THE CONTROVERSY OVER THEIR POTENTIAL FOR ADVERSE-EFFECTS ON CORTICAL NEURONAL MORPHOLOGY
Acta neurochirurgica
COMPETITIVE AS WELL AS UNCOMPETITIVE N-METHYL-D-ASPARTATE RECEPTOR ANTAGONISTS AFFECT CORTICAL NEURONAL MORPHOLOGY AND CEREBRAL GLUCOSE-METABOLISM
Neurochemical research
SYNTHESIS AND SEROTONERGIC ACTIVITY OF 5-(OXADIAZOLYL)TRYPTAMINES - POTENT AGONISTS FOR 5-HT(1D) RECEPTORS
Journal of medicinal chemistry
THE TACHYKININ NK(1) RECEPTOR ANTAGONIST CP-99,994 ATTENUATES CISPLATIN-INDUCED EMESIS IN THE FERRET
European journal of pharmacology
L-694,247 - A POTENT 5-HT(1D) RECEPTOR AGONIST
British Journal of Pharmacology
LACK OF EFFECT OF L-687,414 ((-CIS-4-METHYL-HA-966), AN NMDA RECEPTORANTAGONIST ACTING AT THE GLYCINE SITE, ON CEREBRAL GLUCOSE-METABOLISMAND CORTICAL NEURONAL MORPHOLOGY())
British Journal of Pharmacology
EFFECT OF RP 67580, A NONPEPTIDE NEUROKININ(1) RECEPTOR ANTAGONIST, ON FACILITATION OF A NOCICEPTIVE SPINAL FLEXION REFLEX IN THE RAT
British Journal of Pharmacology