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Use of fluorescence spectroscopy to study conformational changes in the beta(2)-adrenoceptor
G PROTEIN PATHWAYS, PT A, RECEPTORS
Delineating structure-function relationships in the dopamine transporter from natural and engineered Zn2+ binding sites
LIFE SCIENCES
Water transport by the human Na+-coupled glutamate cotransporter expressedin Xenopus oocytes
JOURNAL OF PHYSIOLOGY-LONDON
Functional differences between full and partial agonists: Evidence for ligand-specific receptor conformations
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Biophysical characterization of the cocaine binding pocket in the serotonin transporter using a fluorescent cocaine analogue as a molecular reporter
JOURNAL OF BIOLOGICAL CHEMISTRY
Engineered Zn2+ switches in the gamma-aminobutyric acid (GABA) transporter-1 - Differential effects on GABA uptake and currents
JOURNAL OF BIOLOGICAL CHEMISTRY
Activation of the beta(2)-adrenergic receptor involves disruption of an ionic lock between the cytoplasmic ends of transmembrane segments 3 and 6
JOURNAL OF BIOLOGICAL CHEMISTRY
Agonist-induced conformational changes at the cytoplasmic side of transmembrane segment 6 in the beta(2) adrenergic receptor mapped by site-selectivefluorescent labeling
JOURNAL OF BIOLOGICAL CHEMISTRY
Uncovering molecular mechanisms involved in activation of G protein-coupled receptors
ENDOCRINE REVIEWS
The effect of pH on beta(2) adrenoceptor function - Evidence for protonation-dependent activation
JOURNAL OF BIOLOGICAL CHEMISTRY
Structural probing of a microdomain in the dopamine transporter by engineering of artificial Zn2+ binding sites
BIOCHEMISTRY
Assessing adrenergic receptor conformation using chemically reactive fluorescent probes
ADRENERGIC RECEPTOR PROTOCOLS
Characterization of ligand-induced conformational states in the beta(2) adrenergic receptor
JOURNAL OF RECEPTOR AND SIGNAL TRANSDUCTION RESEARCH
Effects of guanine, inosine, and xanthine nucleotides on beta(2)-adrenergic receptor/G(s) interactions: Evidence for multiple receptor conformations
MOLECULAR PHARMACOLOGY
Mutation of a highly conserved aspartic acid in the beta(2) adrenergic receptor: Constitutive activation, structural instability, and conformational rearrangement of transmembrane segment 6
MOLECULAR PHARMACOLOGY
Defining proximity relationships in the tertiary structure of the dopaminetransporter - Identification of a conserved glutamic acid as a third coordinate in the endogenous Zn2+-binding site
JOURNAL OF BIOLOGICAL CHEMISTRY
Examining the efficiency of receptor/G-protein coupling with a cleavable beta(2)-adrenoceptor-G(s alpha) fusion protein
EUROPEAN JOURNAL OF BIOCHEMISTRY
DELINEATION OF AN ENDOGENOUS ZINC-BINDING SITE IN THE HUMAN DOPAMINE TRANSPORTER
EMBO journal (Print)
CONSTITUTIVE ACTIVATION AND STRUCTURAL INSTABILITY OF THE BETA-2 ADRENOCEPTOR BY MUTATION OF A HIGHLY CONSERVED ASPARTIC-ACID
Naunyn-Schmiedeberg's archives of pharmacology
SITE-SELECTIVE FLUORESCENT LABELING OF THE BETA-2 ADRENOCEPTOR - MAPPING AGONIST-INDUCED CONFORMATIONAL-CHANGES AT THE CYTOPLASMIC SIDE OF TRANSMEMBRANE SEGMENT VI
Naunyn-Schmiedeberg's archives of pharmacology
DELINEATING STRUCTURAL-CHANGES INVOLVED IN ACTIVATION OF G-PROTEIN COUPLED RECEPTORS BY FLUORESCENCE SPECTROSCOPY
Naunyn-Schmiedeberg's archives of pharmacology
DIFFERENTIAL-EFFECTS OF PARTIAL AGONISTS ON G-PROTEIN COUPLING OF THEBETA(2)-ADRENOCEPTOR AND A CONSTITUTIVELY ACTIVE MUTANT OF THE BETA(2)-ADRENOCEPTOR
Naunyn-Schmiedeberg's archives of pharmacology
DELINEATING STRUCTURAL-CHANGES INVOLVED IN ACTIVATION OF G-PROTEIN COUPLED RECEPTORS BY FLUORESCENCE SPECTROSCOPY
Naunyn-Schmiedeberg's archives of pharmacology
IDENTIFICATION OF AN ENDOGENOUS ZN(2-SITE IN THE DOPAMINE TRANSPORTERUNCOVERS DOMAINS CRITICAL FOR SUBSTRATE TRANSLOCATION() BINDING)
Naunyn-Schmiedeberg's archives of pharmacology
EXAMINATION OF LIGAND-INDUCED CONFORMATIONAL-CHANGES IN THE BETA(2) ADRENERGIC-RECEPTOR
Life sciences
DIFFERENT EFFECTS OF G(S)ALPHA SPLICE VARIANTS ON BETA(2)-ADRENORECEPTOR-MEDIATED SIGNALING - THE BETA(2)-ADRENORECEPTOR COUPLED TO THE LONG SPLICE VARIANT OF G(S)ALPHA HAS PROPERTIES OF A CONSTITUTIVELY ACTIVE RECEPTOR
The Journal of biological chemistry
G-PROTEIN-COUPLED RECEPTORS - II - MECHANISM OF AGONIST ACTIVATION
The Journal of biological chemistry
DIFFERENT EFFECTS OF G(S)ALPHA SPLICE VARIANTS ON BETA(2)-ADRENORECEPTOR-MEDIATED SIGNALING - THE BETA(2)-ADRENORECEPTOR COUPLED TO THE LONG SPLICE VARIANT OF G(S)ALPHA HAS PROPERTIES OF A CONSTITUTIVELY ACTIVE RECEPTOR. (VOL 273, PG 5109, 1998)
The Journal of biological chemistry
AGONISTS INDUCE CONFORMATIONAL-CHANGES IN TRANSMEMBRANE DOMAIN-III AND DOMAIN-VI OF THE BETA(2) ADRENOCEPTOR
EMBO journal
EFFECTIVE RECEPTOR G-PROTEIN COUPLING IN A BETA-2-ADRENOCEPTOR/GS-ALPHA FUSION PROTEIN/
Naunyn-Schmiedeberg's archives of pharmacology
STRUCTURAL INSTABILITY OF A CONSTITUTIVELY ACTIVE G-PROTEIN-COUPLED RECEPTOR - AGONIST-INDEPENDENT ACTIVATION DUE TO CONFORMATIONAL FLEXIBILITY
The Journal of biological chemistry
THE ACTIVATION STATE OF G(S-ALPHA) DETERMINES THE AGONIST AND INVERSEAGONIST PROPERTIES OF BETA(2)-ADRENOCEPTOR LIGANDS
Naunyn-Schmiedeberg's archives of pharmacology
LIGAND STABILIZATION OF THE BETA(2) ADRENERGIC-RECEPTOR - EFFECT OF DTT ON RECEPTOR CONFORMATION MONITORED BY CIRCULAR-DICHROISM AND FLUORESCENCE SPECTROSCOPY
Biochemistry
TACHYKININ NONPEPTIDE ANTAGONISTS - BINDING DOMAIN AND MOLECULAR-MODEOF ACTION
Biochemical Society transactions
FLUORESCENT LABELING OF PURIFIED BETA(2) ADRENERGIC-RECEPTOR - EVIDENCE FOR LIGAND-SPECIFIC CONFORMATIONAL-CHANGES
The Journal of biological chemistry
MOLECULAR MECHANISM OF ACTIVATION AND INHIBITION OF 7TM PEPTIDE RECEPTORS
European journal of pharmaceutical sciences
EVIDENCE FOR A COMMON MOLECULAR-MODE OF ACTION FOR CHEMICALLY DISTINCT NONPEPTIDE ANTAGONISTS AT THE NEUROKININ-1 (SUBSTANCE-P) RECEPTOR
Molecular pharmacology
THE SPECIES SELECTIVITY OF CHEMICALLY DISTINCT TACHYKININ NONPEPTIDE ANTAGONISTS IS DEPENDENT ON COMMON DIVERGENT RESIDUES OF THE RAT AND HUMAN NEUROKININ-1 RECEPTORS
Molecular pharmacology
SPECIFIC RESIDUES AT THE TOP OF TRANSMEMBRANE SEGMENT-V AND SEGMENT-VI OF THE NEUROKININ-1 RECEPTOR INVOLVED IN BINDING OF THE NONPEPTIDE ANTAGONIST CP 96,345. (VOL 269, PG 23959, 1994)
The Journal of biological chemistry
MUTATIONS ALONG TRANSMEMBRANE SEGMENT-II OF THE NK-1 RECEPTOR AFFECT SUBSTANCE-P COMPETITION WITH NONPEPTIDE ANTAGONISTS BUT NOT SUBSTANCE-P BINDING
The Journal of biological chemistry
SPECIFIC RESIDUES AT THE TOP OF TRANSMEMBRANE SEGMENT-V AND SEGMENT-VI OF THE NEUROKININ-1 RECEPTOR INVOLVED IN BINDING OF THE NONPEPTIDE ANTAGONIST CP-96,345
The Journal of biological chemistry
BINDING EPITOPES FOR PEPTIDE AND NONPEPTIDE LIGANDS ON THE NK1 (SUBSTANCE-P) RECEPTOR
Regulatory peptides
A SOLUBLE DIVALENT CLASS-I MAJOR HISTOCOMPATIBILITY COMPLEX MOLECULE INHIBITS ALLOREACTIVE T-CELLS AT NANOMOLAR CONCENTRATIONS
Proceedings of the National Academy of Sciences of the United Statesof America
2 NONPEPTIDE TACHYKININ ANTAGONISTS ACT THROUGH EPITOPES ON CORRESPONDING SEGMENTS OF THE NK1 AND NK2 RECEPTORS
Proceedings of the National Academy of Sciences of the United Statesof America
RECOMBINANTLY EXPRESSED Y1 RECEPTORS FOR NPY - DISTINCT SEQUENCE ELEMENTS CONTROL G-PROTEIN ACTIVATION
Journal of neurochemistry
IDENTIFICATION OF BINDING EPITOPES FOR NONPEPTIDE ANTAGONISTS ON THE TACHYKININ RECEPTORS THROUGH CONSTRUCTION OF CHIMERIC NK-1 NK-2 AND NK-1/NK-3 RECEPTORS/
Journal of neurochemistry
CONSERVED HIS(VI-17) OF THE NK-1 RECEPTOR IS INVOLVED IN BINDING OF NONPEPTIDE ANTAGONISTS BUT NOT SUBSTANCE-P
FEBS letters