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Optimisation of the allylsilane approach to C-10 deoxo carba analogues of dihydroartemisinin: synthesis and in vitro antimalarial activity of new, metabolically stable C-10 analogues
JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 1
Is breath-hold time an objective index of exertional dyspnoea in humans?
EUROPEAN JOURNAL OF APPLIED PHYSIOLOGY
P-glycoprotein and transporter MRP1 reduce HIV protease inhibitor uptake in CD4 cells: potential for accelerated viral drug resistance?
AIDS
Is reversal of chloroquine resistance ready for the clinic?
LANCET
Regioselective Mukaiyama hydroperoxysilylation of 2-alkyl- or 2-aryl-prop-2-en-1-ols: application to a new synthesis of 1,2,4-trioxanes
TETRAHEDRON LETTERS
Diamidine compounds: Selective uptake and targeting in Plasmodium falciparum
MOLECULAR PHARMACOLOGY
Effects of prior exercise on oxygen uptake and phosphocreatine kinetics during high-intensity knee-extension exercise in humans
JOURNAL OF PHYSIOLOGY-LONDON
Influence of exercise intensify on the on- and off-transient kinetics of pulmonary oxygen uptake in humans
JOURNAL OF PHYSIOLOGY-LONDON
Synthesis, antimalarial activity, biomimetic iron(II) chemistry, and in vivo metabolism of novel, potent C-10-phenoxy derivatives of dihydroartemisinin
JOURNAL OF MEDICINAL CHEMISTRY
The role of glutathione in the neurotoxicity of artemisinin derivatives invitro
BIOCHEMICAL PHARMACOLOGY
Novel quinoline antimalarials
ANTIMALARIAL CHEMOTHERAPY
Definitive proof for a role of pfmdr 1 in quinoline resistance in Plasmodium falciparum
DRUG RESISTANCE UPDATES
Chance and determinism in the development of isolated communities
GLOBAL ECOLOGY AND BIOGEOGRAPHY
Insulation integrity of GIS/GITL systems and management of particle contamination
IEEE ELECTRICAL INSULATION MAGAZINE
Relative contribution of cytochromes P-450 and flavin-containing monoxygenases to the metabolism of albendazole by human liver microsomes
BRITISH JOURNAL OF CLINICAL PHARMACOLOGY
Estimating the parameters of aerobic function during exercise using an exponentially increasing work rate protocol
MEDICAL & BIOLOGICAL ENGINEERING & COMPUTING
Biliary metabolites of beta-artemether in rats: Biotransformations of an antimalarial endoperoxide
DRUG METABOLISM AND DISPOSITION
Potent enhancement of the sensitivity of Plasmodium falciparum to chloroquine by the bisbenzylisoquinoline akaloid cepharanthin
ANTIMICROBIAL AGENTS AND CHEMOTHERAPY
Control of the exercise hyperpnoea in humans: a modeling perspective
RESPIRATION PHYSIOLOGY
Intersample fluctuations in phosphocreatine concentration determined by P-31-magnetic resonance spectroscopy and parameter estimation of metabolic responses to exercise in humans
JOURNAL OF PHYSIOLOGY-LONDON
Biomimetic Fe(II)-mediated degradation of arteflene (Ro-42-1611). The first EPR spin-trapping evidence for the previously postulated secondary carbon-centered cyclohexyl radical.
JOURNAL OF ORGANIC CHEMISTRY
Molecular cloning of a gene encoding a 20S proteasome beta subunit from Plasmodium falciparum
INTERNATIONAL JOURNAL FOR PARASITOLOGY
Simultaneous determination of muscle P-31 and O-2 uptake kinetics during whole body NMR spectroscopy
JOURNAL OF APPLIED PHYSIOLOGY
Simultaneous determination of artemether and its major metabolite dihydroartemisinin in plasma by gas chromatography-mass spectrometry-selected ion monitoring
JOURNAL OF CHROMATOGRAPHY B
Altered binding of chloroquine to ferriprotoporphyrin IX is the basis for chloroquine resistance
DRUG RESISTANCE UPDATES
Diagnostic utility of metabolic exercise testing in a patient with cardiovascular disease
HEART
Post partum creatine phosphokinase and its muscle-brain isoenzyme elevation and transient Q-wave in a patient with idiopathic hypertrophic subaortic stenosis
INTERNATIONAL JOURNAL OF OBSTETRIC ANESTHESIA
Effect of altered body CO2 stores on pulmonary gas exchange dynamics during incremental exercise in humans
EXPERIMENTAL PHYSIOLOGY
An integrated model of chloroquine action
PARASITOLOGY TODAY
Na+/H+ antiporter, chloroquine uptake and drug resistance: Inconsistenciesin a newly proposed model
PARASITOLOGY TODAY
Application of the TMSOTf-AgClO4 activator system to the synthesis of novel, potent, C-10 phenoxy derivatives of dihydroartemisinin
TETRAHEDRON LETTERS
Inferences from pulmonary O-2 uptake with respect to intramuscular [phosphocreatine] kinetics during moderate exercise in humans
JOURNAL OF PHYSIOLOGY-LONDON
Novel, potent, semisynthetic antimalarial carba analogues of the first-generation 1,2,4-trioxane artemether
JOURNAL OF MEDICINAL CHEMISTRY
New 4-aminoquinoline mannich base antimalarials. 1. Effect of an alkyl substituent in the 5 '-position of the 4 '-hydroxyanilino side chain
JOURNAL OF MEDICINAL CHEMISTRY
Cellular uptake of chloroquine is dependent on binding to ferriprotoporphyrin IX and is independent of NHE activity in Plasmodium falciparum
JOURNAL OF CELL BIOLOGY
Phenotypic and genotypic characteristics of recently adapted isolates of Plasmodium falciparum from Thailand
AMERICAN JOURNAL OF TROPICAL MEDICINE AND HYGIENE
Energy expenditure and substrate utilization in adults with cystic fibrosis and diabetes mellitus
AMERICAN JOURNAL OF CLINICAL NUTRITION
THE EFFECT OF 2,2'-SUBSTITUTION ON THE METABOLISM AND TOXICITY OF DAPSONE IN-VITRO AND IN-VIVO
Environmental toxicology and pharmacology
ELECTRODE ROUGHNESS EFFECTS ON THE BREAKDOWN OF AIR-INSULATED APPARATUS
IEEE transactions on dielectrics and electrical insulation
EFFECTS OF PRIOR ARM EXERCISE ON PULMONARY GAS-EXCHANGE KINETICS DURING HIGH-INTENSITY LEG EXERCISE IN HUMANS
Experimental physiology
INFERENCES FROM PULMONARY O-2 UPTAKE KINETICS WITH RESPECT TO TISSUE ENERGETICS DURING EXERCISE
The FASEB journal
DETERMINANTS AND CONTROL OF BREATHING DURING MUSCULAR EXERCISE
British journal of sports medicine
PALEO-BIOENERGETICS - THE METABOLIC-RATE OF MARCHING ROMAN LEGIONARIES
British journal of sports medicine
Equilibrium theory and alternative stable equilibria
JOURNAL OF BIOGEOGRAPHY
Cover estimates of epiphytic coralline algae (Corallinales, Rhodophyta): Braun-Blanquet vs computer image analysis
CRYPTOGAMIE ALGOLOGIE
CLONING, PHARMACOLOGICAL CHARACTERIZATION AND DISTRIBUTION OF A NOVELGALANIN RECEPTOR (VOL 51, PG 49, 1997)
Molecular brain research
A COMPARISON OF THE PHENOMENOLOGY AND GENETICS OF MULTIDRUG-RESISTANCE IN CANCER-CELLS AND QUINOLINE RESISTANCE IN PLASMODIUM-FALCIPARUM
Pharmacology & therapeutics
4-AMINOQUINOLINES - PAST, PRESENT, AND FUTURE - A CHEMICAL PERSPECTIVE
Pharmacology & therapeutics
THE ROLE OF IRON IN NEUROTOXICITY - A STUDY OF NOVEL ANTIMALARIAL-DRUGS
Neurotoxicology
MORPHOLOGICAL AND IMMUNOCYTOCHEMICAL EFFECTS OF DIHYDROARTEMISININ ONDIFFERENTIATING NB2A NEUROBLASTOMA-CELLS
Neurotoxicology
BINDING OF DIHYDROARTEMISININ TO DIFFERENTIATING NEUROBLASTOMA-CELLS AND RAT CORTICAL HOMOGENATE
Neurotoxicology
EFFECT OF DISPOSITION OF MANNICH ANTIMALARIAL AGENTS ON THEIR PHARMACOLOGY AND TOXICOLOGY
Antimicrobial agents and chemotherapy
RELATIONSHIP BETWEEN ANTIMALARIAL DRUG ACTIVITY, ACCUMULATION, AND INHIBITION OF HEME POLYMERIZATION IN PLASMODIUM-FALCIPARUM IN-VITRO
Antimicrobial agents and chemotherapy
CENTRAL ROLE OF HEMOGLOBIN DEGRADATION IN MECHANISMS OF ACTION OF 4-AMINOQUINOLINES, QUINOLINE METHANOLS, AND PHENANTHRENE METHANOLS
Antimicrobial agents and chemotherapy
A CARBONYL OXIDE ROUTE TO ANTIMALARIAL YINGZHAOSU-A ANALOGS - SYNTHESIS AND ANTIMALARIAL ACTIVITY
Tetrahedron letters
NEURAL-NET WIZARD
Science
MUTUALISTIC BENEFITS GENERATE AN UNEQUAL DISTRIBUTION OF RISKY ACTIVITIES AMONG UNRELATED GROUP MEMBERS
Naturwissenschaften
ACCESS TO HEMATIN - THE BASIS OF CHLOROQUINE RESISTANCE
Molecular pharmacology
EFFECTS OF EXERCISE INTENSITY ON THE PARAMETERS OF V-O2 KINETICS IN HUMANS
Journal of physiology
SIMULTANEOUS DETERMINATION OF INTRAMUSCULAR HIGH-ENERGY PHOSPHATE ANDPULMONARY OXYGEN-UPTAKE KINETICS FOR QUADRICEPS EXERCISE DURING WHOLE-BODY P-31-NMR SPECTROSCOPY (VOL 506P, PG 97P, 1998)
Journal of physiology
SIMULTANEOUS DETERMINATION OF INTRAMUSCULAR HIGH-ENERGY PHOSPHATE ANDPULMONARY OXYGEN-UPTAKE KINETICS FOR QUADRICEPS EXERCISE DURING WHOLE-BODY P-31-NMR SPECTROSCOPY
Journal of physiology
THE ROLE OF GLUTATHIONE IN THE IN-VITRO NEUROTOXICITY OF NOVEL ANTIMALARIAL-DRUGS
Journal of neurochemistry
MORTALITY DURING DISPERSAL AND THE COST OF HOST-SPECIFICITY IN PARASITES - HOW MANY APHIDS FIND HOSTS
Journal of Animal Ecology
SOIL MICROFLORA AS HOSTS OF REDLEGGED EARTH MITE (HALOTYDEUS DESTRUCTOR)
Entomologia experimentalis et applicata
THE EFFECT OF IRON CHELATORS ON THE NEUROTOXICITY OF ARTEMISININ DERIVATIVES IN-VITRO
British Journal of Pharmacology
THE BILIARY METABOLITES OF BETA-ARTEMETHER, AN ENDOPEROXIDE ANTIMALARIAL
British Journal of Pharmacology
THE FREE RADICAL-MEDIATED NEUROTOXICITY OF ARTEMISININ DERIVATIVES IN-VITRO
British Journal of Pharmacology
THYMIDYLATE SYNTHASE (TS) AND P53 PROTEIN EXPRESSION IN PATIENTS WITHRECTAL-CANCER TREATED WITH PREOPERATIVE 5-FLUOROURACIL (5-FU) BASED CHEMORADIOTHERAPY (CRT)
British Journal of Cancer
CONTEXT-DEPENDENT BEHAVIOR AND THE BENEFITS OF COMMUNAL NESTING
The American naturalist
HEPATIC CYTOCHROME-P450 CYP2C ACTIVITY IN PSORIASIS - STUDIES USING PROGUANIL AS A PROBE COMPOUND
Acta dermato-venereologica
THE INTERACTION OF VOLCANISM AND SEDIMENTATION IN THE PROXIMAL AREAS OF A MIDTERTIARY VOLCANIC DOME FIELD, CENTRAL ARIZONA, USA
Journal of sedimentary research
SIMULTANEOUS DETERMINATION OF INTRAMUSCULAR HIGH-ENERGY PHOSPHATE ANDPULMONARY O-2 UPTAKE KINETICS FOR QUADRICEPS EXERCISE DURING WHOLE-BODY NMR-SPECTROSCOPY
The FASEB journal
CLONING, PHARMACOLOGICAL CHARACTERIZATION AND DISTRIBUTION OF A NOVELGALANIN RECEPTOR
Molecular brain research
THE BIOMIMETIC IRON-MEDIATED DEGRADATION OF ARTEFLENE (RO-42-1611), AN ENDOPEROXIDE ANTIMALARIAL - IMPLICATIONS FOR THE MECHANISM OF ANTIMALARIAL ACTIVITY
Tetrahedron letters
QUINOLINE RESISTANCE MECHANISMS IN PLASMODIUM-FALCIPARUM - THE DEBATEGOES ON
Parasitology
AVOIDING PSEUDO LACTATE THRESHOLDS FROM PULMONARY GAS-EXCHANGE INDEXES DURING INCREMENTAL EXERCISE
Journal of physiology
ASSESSING THE REDOX STATE OF CYTOCHROME AA(3) IN SKELETAL-MUSCLE DURING EXHAUSTING MUSCULAR EXERCISE IN HUMANS BY MEANS OF NEAR-INFRARED SPECTROSCOPY
Journal of physiology
SYNTHESIS, ANTIMALARIAL ACTIVITY, AND MOLECULAR MODELING OF TEBUQUINEANALOGS
Journal of medicinal chemistry
ENHANCED IN-VITRO NEUROTOXICITY OF ARTEMISININ DERIVATIVES IN THE PRESENCE OF HEMIN
Biochemical pharmacology
EFFECTS OF PRIOR EXERCISE ON PULMONARY GAS-EXCHANGE KINETICS DURING HIGH-INTENSITY EXERCISE IN HUMANS
Journal of applied physiology
THE EFFECT OF FLUORINE SUBSTITUTION ON THE ANTIMALARIAL ACTIVITY OF TEBUQUINE
Bioorganic & medicinal chemistry letters
IN-VITRO SELECTION OF HALOFANTRINE RESISTANCE IN PLASMODIUM-FALCIPARUM IS NOT ASSOCIATED WITH INCREASED EXPRESSION OF PGH1
Molecular and biochemical parasitology
AMODIAQUINE ACCUMULATION IN PLASMODIUM-FALCIPARUM AS A POSSIBLE EXPLANATION FOR ITS SUPERIOR ANTIMALARIAL ACTIVITY OVER CHLOROQUINE
Molecular and biochemical parasitology
MANIPULATION OF THE N-ALKYL SUBSTITUENT IN AMODIAQUINE TO OVERCOME THE VERAPAMIL-SENSITIVE CHLOROQUINE RESISTANCE COMPONENT
Antimicrobial agents and chemotherapy
4-AMINOQUINOLINE RESISTANCE OF PLASMODIUM-FALCIPARUM - INSIGHTS FROM THE STUDY OF AMODIAQUINE UPTAKE
Molecular pharmacology
PHYSICOCHEMICAL PROPERTIES CORRELATED WITH DRUG-RESISTANCE AND THE REVERSAL OF DRUG-RESISTANCE IN PLASMODIUM-FALCIPARUM
Molecular pharmacology
EFFECT OF BODY CO2 STORES ON PULMONARY GAS-EXCHANGE DYNAMICS DURING INCREMENTAL EXERCISE
Journal of physiology
THE SLOW PHASE OF O-2 UPTAKE KINETICS DURING MUSCULAR EXERCISE IN SPRINT-TRAINED AND ENDURANCE-TRAINED HUMANS
Journal of physiology
THE INFLUENCE OF HYPOXIA ON OXYGEN-UPTAKE KINETICS FOR HIGH-INTENSITYEXERCISE IN HUMANS
Journal of physiology
PULMONARY O-2 UPTAKE KINETICS AND FEMORAL-ARTERY BLOOD-FLOW FOLLOWINGHIGH-INTENSITY EXERCISE IN HUMANS
Journal of physiology
THE INFLUENCE OF ACUTE METABOLIC ACIDEMIA ON VENTILATORY KINETICS DURING MODERATE EXERCISE IN HUMANS
Journal of physiology
ESTIMATING THE METABOLIC-RATE OF MARCHING ROMAN LEGIONARIES
Journal of physiology
MECHANISM-BASED DESIGN OF PARASITE-TARGETED ARTEMISININ DERIVATIVES -SYNTHESIS AND ANTIMALARIAL ACTIVITY OF BENZYLAMINO AND ALKYLAMINO ETHER ANALOGS OF ARTEMISININ
Journal of medicinal chemistry
THE INFLUENCE OF HEPATIC-METABOLISM ON THE NEUROTOXICITY OF ARTEMISININ DERIVATIVES ON CULTURED NB2A NEUROBLASTOMA-CELLS
British Journal of Pharmacology
DIFFICULTIES IN RECRUITING ACADEMIC STAFF
British Dental Journal
THE ROLE OF DRUG ACCUMULATION IN 4-AMINOQUINOLINE ANTIMALARIAL POTENCY - THE INFLUENCE OF STRUCTURAL SUBSTITUTION AND PHYSICOCHEMICAL PROPERTIES
Biochemical pharmacology
THE EFFECT OF FLUORINE SUBSTITUTION ON THE HAEMOTOXICITY OF PRIMAQUINE
Bioorganic & medicinal chemistry letters
THE ROLE OF S-MEPHENYTOIN HYDROXYLASE (CYP2C19) IN THE METABOLISM OF THE ANTIMALARIAL BIGUANIDES
British journal of clinical pharmacology
OBLIGATORY ANAEROBIOSIS RESULTING FROM OXYGEN UPTAKE-TO-BLOOD FLOW RATIO DISPERSION IN SKELETAL-MUSCLE - A MODEL
European journal of applied physiology and occupational physiology
BREATH-HOLD DURATION AND RESPIRATORY SENSATION DURING MUSCULAR EXERCISE IN HUMANS
Biological psychology