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Comparative antiplatelet efficacy of a novel, nonpeptide GPIIb/IIIa antagonist (XV454) and abciximab (c7E3) in flow models of thrombosis
ARTERIOSCLEROSIS THROMBOSIS AND VASCULAR BIOLOGY
Synthesis and pharmacology of modified amidine isoxazoline glycoprotein IIb/IIIa receptor antagonists
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Integrin-binding peptides containing RGD produce coronary arteriolar dilation via cyclooxygenase activation
AMERICAN JOURNAL OF PHYSIOLOGY-HEART AND CIRCULATORY PHYSIOLOGY
Effects in humans of intravenously administered endotoxin on soluble cell-adhesion molecule and inflammatory markers: A model of human diseases
CLINICAL AND EXPERIMENTAL PHARMACOLOGY AND PHYSIOLOGY
beta-endorphin-containing memory-cells and mu-opioid receptors undergo transport to peripheral inflamed tissue
JOURNAL OF NEUROIMMUNOLOGY
Comparison of the effect of different platelet GPIIb/IIa antagonists on the dynamics of platelet/fibrin-mediated clot strength induced using thromboelastography
THROMBOSIS RESEARCH
Selective alpha(v)beta(3)-receptor blockade reduces macrophage infiltration and restenosis after balloon angioplasty in the atherosclerotic rabbit
CIRCULATION
Platelet GPIIb/IIIa binding characteristics of small molecule RGD mimetic:distinct binding profile for Roxifiban
BRITISH JOURNAL OF PHARMACOLOGY
Opioid peptide-expressing leukocytes - Identification, recruitment, and simultaneously increasing inhibition of inflammatory pain
ANESTHESIOLOGY
Small molecule alpha(v) integrin antagonists: novel anticancer agents
EXPERT OPINION ON INVESTIGATIONAL DRUGS
Potential role of platelet glycoprotein IIb/IIIa antagonists in cerebrovascular disorders
CNS DRUGS
Comparative in vitro efficacy of different platelet glycoprotein IIb/IIIa antagonists on platelet-mediated clot strength induced by tissue factor with use of thromboelastography - Differentiation among glycoprotein IIb/IIIa antagonists
ARTERIOSCLEROSIS THROMBOSIS AND VASCULAR BIOLOGY
Template-constrained cyclic peptide analogues of somatostatin: Subtype-selective binding to somatostatin receptors and antiangiogenic activity
BIOORGANIC & MEDICINAL CHEMISTRY
Ring constrained analogues of beta-alanine-containing GPIIb/IIIa receptor antagonists
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Human platelet alpha IIb beta 3 integrin binding affinity end specificity of SJ874: antiplatelet efficacy versus aspirin
CORONARY ARTERY DISEASE
Antiangiogenesis efficacy of nitric oxide donors
JOURNAL OF CELLULAR BIOCHEMISTRY
Hypoxia induces differential expression of the integrin receptors alpha(v beta 3) and alpha(v beta 5) cultured human endothelial cells
JOURNAL OF CELLULAR BIOCHEMISTRY
Immunocytochemical studies of the gonadotropic cells in the pituitary gland of male mullet, Mugil cephalus, during the annual reproductive cycle in both natural habitat and captivity
JOURNAL OF APPLIED ICHTHYOLOGY-ZEITSCHRIFT FUR ANGEWANDTE ICHTHYOLOGIE
Co-expression of beta-endorphin with adhesion molecules in a model of inflammatory pain
JOURNAL OF NEUROIMMUNOLOGY
Comparative efficacy of different low-molecular-weight heparins (LMWHs) and drug interactions with LMWH: Implications for management of vascular disorders
SEMINARS IN THROMBOSIS AND HEMOSTASIS
A nonpeptide integrin antagonist can inhibit epithelial cell ingestion of Streptococcus pyogenes by blocking formation of integrin alpha 5 beta 1-fibronectin-M1 protein complexes
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
Isoxazolines as potent antagonists of the integrin alpha(v)beta(3)
JOURNAL OF MEDICINAL CHEMISTRY
Disubstituted indazoles as potent antagonists of the integrin alpha(v)beta(3)
JOURNAL OF MEDICINAL CHEMISTRY
Implication of somatolactin in the regulation of sexual maturation and spawning of Mugil cephalus
JOURNAL OF EXPERIMENTAL ZOOLOGY
Differential antiplatelet efficacy for various GPIIb/IIIa antagonists: Role of plasma calcium levels
CARDIOVASCULAR RESEARCH
Immobilized platelets support human colon carcinoma cell tethering, rolling, and firm adhesion under dynamic flow conditions
BLOOD
Domain 5 of high molecular weight kininogen (kininostatin) down-regulates endothelial cell proliferation and migration and inhibits angiogenesis
BLOOD
Regulation of angiogenesis in vivo by ligation of integrin alpha 5 beta 1 with the central cell-binding domain of fibronectin
AMERICAN JOURNAL OF PATHOLOGY
Antiplatelet therapies: from aspirin to GPIIb/IIIa-receptor antagonists and beyond
DRUG DISCOVERY TODAY
Anti-integrins as a potential therapeutic target in angiogenesis
EXPERT OPINION ON THERAPEUTIC PATENTS
Intravenous and oral antithrombotic efficacy of the novel platelet GPIIb/IIIa antagonist roxifiban (DMP754) and its free acid form, XV459
ARTERIOSCLEROSIS THROMBOSIS AND VASCULAR BIOLOGY
Isoxazoline GPIIb/IIIa antagonists bearing a phosphoramidate
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Platelet glycoprotein IIb/IIIa receptor antagonists derived from isoxazolidines
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Role of hypoxia and extracellular matrix-integrin binding in the modulation of angiogenic growth factors secretion by retinal pigmented epithelial cells
JOURNAL OF CELLULAR BIOCHEMISTRY
Novel small molecule alpha v integrin antagonists: Comparative anti-cancerefficacy with known angiogenesis inhibitors
ANTICANCER RESEARCH
alpha(v)beta(3) integrin binding affinity and specificity of SM256 in various species
JOURNAL OF CARDIOVASCULAR PHARMACOLOGY
Disposition and exposure of the fibrinogen receptor antagonist XV459 on alpha(IIB)beta(3), binding sites in the guinea pig
BIOPHARMACEUTICS & DRUG DISPOSITION
Orally active isoxazoline glycoprotein IIb/IIIa antagonists with extended duration of action
JOURNAL OF MEDICINAL CHEMISTRY
Immunocytochemical and histological studies on the hypophyseal-gonadal system in the freshwater Nile tilapia, Oreochromis niloticus (L.), during sexual maturation and spawning in different habitats
JOURNAL OF EXPERIMENTAL ZOOLOGY
Immunocytochemical study on the localization and distribution of the somatolactin cells in the pituitary gland and the brain of Oreochromis niloticus(Teleostei, Cichlidae)
GENERAL AND COMPARATIVE ENDOCRINOLOGY
Pain control in inflammation governed by selectins
NATURE MEDICINE
NOVEL TC-99M-LABELED PLATELET GPIIB IIIA RECEPTOR ANTAGONISTS AS POTENTIAL IMAGING AGENTS FOR VENOUS AND ARTERIAL THROMBOSIS/
Coronary artery disease
RESTORATION OF CORONARY FLOW BY POTENT PLATELET GPIIB IIIA ANTAGONISTWITHOUT EXOGENOUS THROMBOLYTICS/
The FASEB journal
INHIBITION OF PLATELET-MEDIATED CLOT RETRACTION BY INTEGRIN ANTAGONISTS
The FASEB journal
COMPARATIVE EFFICACY OF DIFFERENT PLATELET GPIIB IIIA RECEPTOR ANTAGONISTS ON PLATELET-MEDIATED CLOT STRENGTH USING TISSUE FACTOR-THROMBOELASTOGRAPHY/
The FASEB journal
INTEGRINS IN HUMAN RETINAL PIGMENTED EPITHELIAL (RPE) CELLS - ROLE OFEXTRACELLULAR-MATRIX PROTEINS (ECMS) AND HYPOXIA ON THE SECRETION OF GROWTH-FACTORS
The FASEB journal
ROLE OF ESTROGEN-RECEPTOR ON AV-BETA-3-MEDIATED CELL-ADHESION, MIGRATION AND SECRETION OF BFGF AND VEGF IN HUMAN ENDOTHELIAL AND ENDOMETRIAL CELLS
The FASEB journal
ROLE OF ALPHA-V-BETA-3 INTEGRIN IN ENDOTHELIAL AND SMOOTH-MUSCLE CELL-MIGRATION - POTENTIAL ROLE IN CORONARY-ARTERY DISEASES
The FASEB journal
XV454, A NOVEL NONPEPTIDE SMALL-MOLECULE PLATELET GIIB IIIA ANTAGONIST WITH COMPARABLE PLATELET ALPHA(IIB)BETA(3)-BINDING KINETICS TO C7E3/
Journal of cardiovascular pharmacology
ORAL ANTIPLATELET EFFICACY AND SPECIFICITY OF A NOVEL NONPEPTIDE PLATELET GPIIB IIIA RECEPTOR ANTAGONIST, DMP-802/
Journal of cardiovascular pharmacology
INTRAVENOUS AND ORAL ANTIPLATELET ANTITHROMBOTIC EFFICACY AND SPECIFICITY OF XR300, A NOVEL NONPEPTIDE PLATELET GPIIB/IIIA ANTAGONIST/
Journal of cardiovascular pharmacology
INTRANASAL ANTIPLATELET ANTITHROMBOTIC EFFICACY OF A NOVEL PLATELET GPIIB/IIIA RECEPTOR ANTAGONIST DMP755/
Thrombosis research
GLYCOPROTEIN IIB IIIA RECEPTOR ANTAGONISTS INHIBIT THE DEVELOPMENT OFPLATELET PROCOAGULANT ACTIVITY/
Thrombosis research
INHIBITION OF PLATELET-MEDIATED CLOT RETRACTION BY INTEGRIN ANTAGONISTS
Thrombosis research
ORAL ANTIPLATELET EFFICACY OF THE PLATELET GPIIB IIIA ANTAGONIST, DMP754 IN NONHUMAN-PRIMATES/
Thrombosis research
DISSOCIATION BETWEEN THE ANTI-AGGREGATORY AND ANTI-SECRETORY EFFECTS OF PLATELET INTEGRIN ALPHA-IIB-BETA-3 (GPIIB IIIA) ANTAGONISTS, C7E3 AND DMP728 (VOL 88, PG 137, 1997)/
Thrombosis research
ELEVATION OF CIRCULATING SMOOTH-MUSCLE CELL CHEMOATTRACTANTS MITOGENSAND ENDOTHELIAL-CELL DYSFUNCTION IN CONGESTIVE-HEART-FAILURE PATIENTS- POTENTIAL ROLE OF ALPHA-V-BETA-3 INTEGRIN/
Naunyn-Schmiedeberg's archives of pharmacology
ANTITHROMBOTIC EFFICACY OF PLATELET GPIIB IIIA RECEPTOR ANTAGONISTS AS COMPARED TO OTHER ANTIPLATELET AND ANTICOAGULANT STRATEGIES/
Naunyn-Schmiedeberg's archives of pharmacology
ACTIVATION-DEPENDENT ALPHA-V-BETA-3 ON PLATELETS AND LYMPHOCYTES BINDS VITRONECTIN AND OSTEOPONTIN
Naunyn-Schmiedeberg's archives of pharmacology
ANTIPLATELET EFFICACY OF XV459, A NOVEL NONPEPTIDE PLATELET GPIIB IIAANTAGONIST - COMPARATIVE PLATELET BINDING PROFILES WITH C7E3/
The Journal of pharmacology and experimental therapeutics
PHARMACODYNAMICS AND PHARMACOKINETICS OF DMP-728, A PLATELET GPIIB IIIA ANTAGONIST, IN HEALTHY-SUBJECTS/
Clinical pharmacology and therapeutics
ACTIVATION-DEPENDENT ALPHA-V-BETA-3 ON PLATELETS AND LYMPHOCYTES BINDS VITRONECTIN AND OSTEOPONTIN - POTENTIAL SURROGATE FOR MONITORING ANTI-ALPHA-V-BETA-3 INTEGRIN EFFICACY
Circulation
DISCOVERY OF A KEY ROLE FOR THE ALPHA-NU-BETA-3 INTEGRIN IN ACUTE ANDDELAYED VASCULAR OCCLUSION AND REOCCLUSION WITHOUT EFFECTS ON HEMOSTASIS
Circulation
THE ROLE OF INTEGRINS ALPHA(V)BETA(3) AND ALPHA(ILB)BETA(3) IN AN EXPERIMENTAL ARTERIAL INJURY MODEL
Circulation
ANTAGONISTS OF VASCULAR CELL INTEGRIN ALPHA-5-BETA-1 INHIBIT ANGIOGENESIS
Circulation
RECENT ADVANCES IN CELL-ADHESION MOLECULES AND EXTRACELLULAR-MATRIX PROTEINS - POTENTIAL CLINICAL IMPLICATIONS
Drug discovery today
SOLID-PHASE SYNTHESIS OF A SELECTIVE ALPHA(V)BETA(3) INTEGRIN ANTAGONIST LIBRARY
Bioorganic & medicinal chemistry letters
COMBINED ALPHA-V-BETA-3 AND PLATELET IIB IIIA INTEGRIN BLOCKADE POTENTLY LIMITS NEOINTIMAL HYPERPLASIA AND LUMEN STENOSIS IN THE PORCINE CORONARY INJURY MODEL/
Journal of the American College of Cardiology
ANTIPLATELET EFFICACY OF ORALLY-ADMINISTERED DMP802, A GPIIB IIIA RECEPTOR ANTAGONIST, IN THE CONSCIOUS DOG/
Journal of the American College of Cardiology
TEMPORAL AND SPATIAL VARIATION IN ALPHA-V-BETA-3 INTEGRIN EXPRESSION FOLLOWING DEEP ARTERIAL INJURY IN THE PORCINE CORONARY RESTENOSIS MODEL
Journal of the American College of Cardiology
INTRANASAL ANTIPLATELET ANTITHROMBOTIC EFFICACY OF THE PLATELET GPIIB/IIIA ANTAGONIST, DMP754/
Journal of the American College of Cardiology
INTRAVENOUS AND ORAL ANTITHROMBOTIC EFFICACY OF A NOVEL NONPEPTIDE ANTIPLATELET GPIIB IIIA ANTAGONIST, DMP-754 AS COMPARED TO OTHER ANTIPLATELET AND ANTICOAGULANT STRATEGIES/
Thrombosis and haemostasis
PLATELET GPIIBIIIA RECEPTOR ANTAGONISTS INHIBIT PLATELET PROCOAGULANTACTIVITY
Thrombosis and haemostasis
DISCOVERY OF NOVEL ORALLY-ACTIVE NONPEPTIDE ANTIPLATELET GPIIB IIIA ANTAGONIST, DMP754 - COMPARATIVE PLATELET BINDING-AFFINITY PROFILES WITH DMP728 AND C7E3/
Thrombosis and haemostasis
DISSOCIATION BETWEEN THE ANTI-AGGREGATORY AND ANTI-SECRETORY EFFECTS OF PLATELET INTEGRIN ALPHA(IIB)BETA(3) (GPIIB IIIA) ANTAGONISTS, C7E3 AND DMP728/
Thrombosis research
BIOLOGICAL MATRIX-DEPENDENT PHARMACOKINETIC AND PHARMACODYNAMIC PARAMETERS OF A NOVEL PLATELET GLYCOPROTEIN IIB IIIA RECEPTOR ANTAGONIST, XU063, IN BEAGLE DOGS/
Thrombosis research
PREVENTION OF CAROTID-ARTERY THROMBOSIS BY ORAL PLATELET GPIIB IIIA ANTAGONIST IN DOGS/
Stroke
INTRANASAL ABSORPTION OF THE PLATELET GLYCOPROTEIN IIB IIIA RECEPTOR ANTAGONIST, DMP-755, AND THE EFFECT OF ANESTHESIA ON NASAL BIOAVAILABILITY/
Journal of pharmaceutical sciences
THE DISCOVERY OF POTENT ISOXAZOLINE GLYCOPROTEIN-IIB IIIA RECEPTOR ANTAGONISTS. (VOL 40, PG 53, 1997)/
Journal of medicinal chemistry
DISCOVERY OF AN ORALLY-ACTIVE SERIES OF ISOXAZOLINE GLYCOPROTEIN IIB IIIA ANTAGONISTS/
Journal of medicinal chemistry
DISCOVERY OF POTENT ISOXAZOLINE GLYCOPROTEIN IIB IIIA RECEPTOR ANTAGONISTS/
Journal of medicinal chemistry
AGONIST-ACTIVATED ALPHA-NU-BETA-3 ON PLATELETS AND LYMPHOCYTES BINDS TO THE MATRIX PROTEIN OSTEOPONTIN
The Journal of biological chemistry
CORTICOTROPIN-RELEASING FACTOR IN ANTINOCICEPTION AND INFLAMMATION
European journal of pharmacology
PLATELET GPIIBIIIA RECEPTOR ANTAGONISTS INHIBIT PLATELET PROCOAGULANTACTIVITY
Circulation
ACTIVATION-DEPENDENT ALPHA-V BETA-3 ON PLATELETS AND LYMPHOCYTES BINDS VITRONECTIN AND OSTEOPONTIN
Circulation
XV454, A NOVEL NONPEPTIDE ANTIPLATELET AGENT WITH COMPARABLE PLATELETALPHA-IIB-BETA-3 BINDING-KINETICS TO C7E3 AND LONG-LASTING ANTIPLATELET EFFICACY AFTER SINGLE INTRAVENOUS OR ORAL-ADMINISTRATION IN NONHUMAN-PRIMATES
Circulation
SELECTIVE ALPHA-V-BETA-3 INTEGRIN BLOCKADE POTENTLY LIMITS NEOINTIMALHYPERPLASIA AND LUMEN STENOSIS FOLLOWING DEEP CORONARY ARTERIAL STENTINJURY - EVIDENCE FOR THE FUNCTIONAL IMPORTANCE OF INTEGRIN ALPHA-V-BETA-3 AND OSTEOPONTIN EXPRESSION DURING NEOINTIMA FORMATION
Cardiovascular Research
ANGIOGENESIS PROMOTERS AND INHIBITORS - POTENTIAL THERAPEUTIC IMPLICATIONS
Molecular medicine today
NOVEL NONPEPTIDE ANTIPLATELET GLYCOPROTEIN IIB IIIA RECEPTOR ANTAGONIST, DMP754 - RECEPTOR-BINDING AFFINITY AND SPECIFICITY/
Coronary artery disease
ANIMAL-MODEL OF ARTERIAL AND VENOUS THROMBOSIS IN DOGS - ASSESSMENT OF THE EFFICACY OF VARIOUS ANTITHROMBOTIC STRATEGIES
The FASEB journal
ANTITHROMBOTIC EFFICACY OF NITRIC-OXIDE DONOR IN ARTERIAL AND VENOUS THROMBOSIS MODEL IN PIGS
The FASEB journal
PLATELET - ENDOTHELIAL-CELL INTERACTIONS IN MEDIATING THE RELEASE OF PLASMINOGEN-ACTIVATOR INHIBITOR-1
Biochemical archives
ENHANCEMENT OF THE INTESTINAL-ABSORPTION OF PEPTIDES AND NONPEPTIDES
Journal of controlled release
ANTAGONISTS OF INTEGRIN ALPHA(V)BETA(3) INHIBIT RETINAL NEOVASCULARIZATION IN A MURINE MODEL
Laboratory investigation
SYNTHESIS AND SOLUTION CONFORMATION OF CYCLO[RGDRGD] - A CYCLIC PEPTIDE WITH SELECTIVITY FOR THE ALPHA-V-BETA-3 RECEPTOR
Journal of medicinal chemistry
LOCAL UP-REGULATION OF CORTICOTROPIN-RELEASING HORMONE AND INTERLEUKIN-1 RECEPTORS IN RATS WITH PAINFUL HINDLIMB INFLAMMATION
European journal of pharmacology
SELECTIVE ALPHA-V BETA-3 INTEGRIN BLOCKADE LIMITS NEOINTIMAL HYPERPLASIA AND LUMEN STENOSIS IN THE STENTED PORCINE CORONARY-ARTERY INJURY MODEL
Circulation
ORAL ANTIPLATELET EFFECTS OF DMP-754 IN DOGS AND NONHUMAN-PRIMATES
Circulation
INTRAVENOUS AND ORAL ANTIPLATELET ANTITHROMBOTIC EFFICACY AND SPECIFICITY OF XR300, A NOVEL NON PEPTIDE PLATELET GPIIB/IIIA ANTAGONIST/
Circulation
DISCOVERY OF A NOVEL NON PEPTIDE ANTIPLATELET GPIIB IIIA RECEPTOR ANTAGONIST, DMP-754 - RECEPTOR-BINDING AFFINITY AND SPECIFICITY/
Circulation