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Species differences in [C-11]clorgyline binding in brain
NUCLEAR MEDICINE AND BIOLOGY
[(11)]Cocaine: PET studies of cocaine pharmacokinetics, dopamine transporter availability and dopamine transporter occupancy
NUCLEAR MEDICINE AND BIOLOGY
Effects of endogenous neurotransmitters on the in vivo binding of dopamineand 5-HT radiotracers in mice
NEUROPSYCHOPHARMACOLOGY
A consideration of the dopamine D2 receptor monomer-dimer equilibrium and the anomalous binding properties of the dopamine D2 receptor ligand, N-methyl spiperone
JOURNAL OF NEURAL TRANSMISSION
Loss of dopamine transporters in methamphetamine abusers recovers with protracted abstinence
JOURNAL OF NEUROSCIENCE
Therapeutic doses of oral methylphenidate significantly increase extracellular dopamine in the human brain
JOURNAL OF NEUROSCIENCE
Non-MAO A binding of clorgyline in white matter in human brain
JOURNAL OF NEUROCHEMISTRY
Imaging brain cholinergic activity with positron emission tomography: Its role in the evaluation of cholinergic treatments in Alzheimer's dementia
BIOLOGICAL PSYCHIATRY
Association of dopamine transporter reduction with psychomotor impairment in methamphetamine abusers
AMERICAN JOURNAL OF PSYCHIATRY
Higher cortical and lower subcortical metabolism in detoxified methamphetamine abusers
AMERICAN JOURNAL OF PSYCHIATRY
Locomotor activity and occupancy of brain cannabinoid CB1 receptors by theantagonist/inverse agonist AM281
SYNAPSE
Sensitivity of binding of high-affinity dopamine receptor radioligands to increased synaptic dopamine
SYNAPSE
Resting brain metabolic activity in a 4 tesla magnetic field
MAGNETIC RESONANCE IN MEDICINE
Effect of amphetamine-induced dopamine release on radiotracer binding to D-1 and D-2 receptors in rat brain striatal slices
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY
Effects of route of administration on cocaine induced dopamine transporterblockade in the human brain
LIFE SCIENCES
Cocaine abusers show a blunted response to alcohol intoxication in limbic brain regions
LIFE SCIENCES
Comparison between intraperitoneal and oral methylphenidate administration: A microdialysis and locomotor activity study
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Cannabinoid receptor-mediated inhibition of acetylcholine release from hippocampal and cortical synaptosomes
BRITISH JOURNAL OF PHARMACOLOGY
The ratio of striatal D1 to muscarinic receptors changes in aging rats housed in an enriched environment
BRAIN RESEARCH
Measuring dopamine D-2 receptors - Dr. Volkow and colleagues reply
AMERICAN JOURNAL OF PSYCHIATRY
Association between age-related decline in brain dopamine activity and impairment in frontal and cingulate metabolism
AMERICAN JOURNAL OF PSYCHIATRY
Untitled
NUCLEAR MEDICINE AND BIOLOGY
Comparable changes in synaptic dopamine induced by methylphenidate and by cocaine in the baboon brain
SYNAPSE
Methylphenidate and cocaine have a similar in vivo potency to block dopamine transporters in the human brain
LIFE SCIENCES
Reinforcing effects of psychostimulants in humans are associated with increases in brain dopamine and occupancy of D-2 receptors
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Large receptor reserve for cannabinoid actions in the central nervous system
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Blockade of striatal dopamine transporters by intravenous methylphenidate is not sufficient to induce self-reports of "high"
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Potentiation of the action of anandamide on hippocampal slices by the fatty acid amide hydrolase inhibitor, palmitylsulphonyl fluoride (AM 374)
EUROPEAN JOURNAL OF PHARMACOLOGY
Prediction of reinforcing responses to psychostimulants in humans by braindopamine D-2 receptor levels
AMERICAN JOURNAL OF PSYCHIATRY
Association of methylphenidate-induced craving with changes in right striato-orbitofrontal metabolism in cocaine abusers: Implications in addiction
AMERICAN JOURNAL OF PSYCHIATRY
Dopamine transporter occupancy after intravenous doses of cocaine and methylphenidate in mice and humans
PSYCHOPHARMACOLOGY
Studies of the brain cannabinoid system using positron and single-photon emission tomography
MARIHUANA AND MEDICINE
IN-VITRO AND EX-VIVO AUTORADIOGRAPHIC STUDIES OF NICOTINIC ACETYLCHOLINE-RECEPTORS USING [F-18] FLUORONORCHLOROEPIBATIDINE IN RODENT AND HUMAN BRAIN
Nuclear medicine and biology
MEASURING DOPAMINE TRANSPORTER OCCUPANCY BY COCAINE IN-VIVO - RADIOTRACER CONSIDERATIONS
Synapse
EVALUATION OF THE IMPORTANCE OF REBINDING TO RECEPTORS IN SLOWING THEAPPROACH TO EQUILIBRIUM OF HIGH-AFFINITY PET AND SPECT RADIOTRACERS
Synapse
ADDICTION AND IMAGING OF THE LIVING HUMAN BRAIN
Drug and alcohol dependence
PET studies of peripheral catechol-O-methyltransferase in non-human primates using [F-18]Ro41-0960
JOURNAL OF NEURAL TRANSMISSION
ON IMAGING NEUROTRANSMITTER RECEPTOR OCCUPANCIES - THE BRAIN CANNABINOID CB1 RECEPTOR SYSTEM
The Journal of nuclear medicine
DOSE-RESPONSE TO METHYLPHENIDATE-INDUCED CHANGES IN [C-11] RACLOPRIDEBINDING
The Journal of nuclear medicine
AN ACUTE DOSE OF NICOTINE DOES NOT INHIBIT BABOON BRAIN MAO-B IN-VIVO
The Journal of nuclear medicine
DOPAMINE TRANSPORTER OCCUPANCY BY INTRAVENOUS METHYLPHENIDATE - RELATIONSHIP TO ITS REINFORCING EFFECTS
The Journal of nuclear medicine
ORAL METHYLPHENIDATE INDUCES SIGNIFICANT LEVELS OF DOPAMINE TRANSPORTER OCCUPANCY
The Journal of nuclear medicine
QUANTIFICATION OF RODENT TISSUE BINDING-SITES FOR ADENOVIRUSES USING RADIOIODINATED FIBER PROTEIN
The Journal of nuclear medicine
AN ACUTE DOSE OF NICOTINE DOES NOT INHIBIT MAO-B IN BABOON BRAIN IN-VIVO
Life sciences
IMAGING THE BRAIN MARIJUANA RECEPTOR - DEVELOPMENT OF A RADIOLIGAND THAT BINDS TO CANNABINOID CB1 RECEPTORS IN-VIVO
Journal of neurochemistry
ENHANCED SENSITIVITY TO BENZODIAZEPINES IN ACTIVE COCAINE-ABUSING SUBJECTS - A PET STUDY
The American journal of psychiatry
DOPAMINE TRANSPORTER OCCUPANCIES IN THE HUMAN BRAIN INDUCED BY THERAPEUTIC DOSES OF ORAL METHYLPHENIDATE
The American journal of psychiatry
FLUORO-NORCHLOROEPIBATIDINE - PRECLINICAL ASSESSMENT OF ACUTE TOXICITY
Nuclear medicine and biology
CONCENTRATION AND OCCUPANCY OF DOPAMINE TRANSPORTERS IN COCAINE ABUSERS WITH [C-11] COCAINE AND PET
Synapse
EFFECT OF THE CANNABINOID RECEPTOR SPECT AGENT, AM-281, ON HIPPOCAMPAL ACETYLCHOLINE-RELEASE FROM RAT-BRAIN SLICES
Neuroscience letters
COMPARISON OF [C-11] COCAINE AND [C-11] D-THREO-METHYLPHENIDATE FOR ASSESSING DOPAMINE TRANSPORTER (DAT) OCCUPANCY BY COCAINE
The Journal of nuclear medicine
DECREASED STRIATAL AND ENHANCED THALAMIC DOPAMINERGIC RESPONSIVITY INDETOXIFIED COCAINE ABUSERS
The Journal of nuclear medicine
DOPAMINE TRANSPORTER OCCUPANCY BY RTI-55, INHIBITION OF DOPAMINE TRANSPORT AND STIMULATION OF LOCOMOTOR-ACTIVITY
The Journal of nuclear medicine
NOVEL RADIOHALOGENATED LIGANDS FOR IMAGING CANNABINOID RECEPTORS (CBRS)
The Journal of nuclear medicine
PET STUDIES OF [18F]NORCHLOROFLUOROEPIBATIDINE IN MAPPING NICOTINIC ACETYLCHOLINE-RECEPTORS (NACHR)
The Journal of nuclear medicine
SPECT IMAGING OF BRAIN CANNABINOID RECEPTORS
The Journal of nuclear medicine
PRECLINICAL TESTING OF F-18 AND I-123 RADIOLIGANDS INVOLVING AUTORADIOGRAPHY AND A PHOSPHOR-IMAGING DEVICE
The Journal of nuclear medicine
ESTIMATING THE CONCENTRATION AND DEGREE OF OCCUPANCY OF DOPAMINE TRANSPORTERS (DAT) IN COCAINE ABUSERS
The Journal of nuclear medicine
COMPARISON OF THE IN-VIVO AND IN-VITRO TIME-COURSE OF BINDING OF A HIGH-AFFINITY RADIOLIGAND
The Journal of nuclear medicine
RELATIONSHIP BETWEEN SUBJECTIVE EFFECTS OF COCAINE AND DOPAMINE TRANSPORTER OCCUPANCY
Nature
DECREASED STRIATAL DOPAMINERGIC RESPONSIVENESS IN DETOXIFIED COCAINE-DEPENDENT SUBJECTS
Nature
BINDING OF THE NONCLASSICAL CANNABINOID CP-55,940, AND THE DIARYLPYRAZOLE AM251 TO RODENT BRAIN CANNABINOID RECEPTORS
Life sciences
EXAMINATION OF THE EFFECT OF THE CANNABINOID RECEPTOR AGONIST, CP-55,940, ON ELECTRICALLY-EVOKED TRANSMITTER RELEASE FROM RAT-BRAIN SLICES
European journal of pharmacology
MODEL FOR ESTIMATING DOPAMINE TRANSPORTER OCCUPANCY AND SUBSEQUENT INCREASES IN SYNAPTIC DOPAMINE USING POSITRON EMISSION TOMOGRAPHY AND CARBON-11-LABELED COCAINE
Biochemical pharmacology
CHIRAL DRUGS - COMPARISON OF THE PHARMACOKINETICS OF [C-11] D-THREO AND I-THREO-METHYLPHENIDATE IN THE HUMAN AND BABOON BRAIN
Psychopharmacology
[F-18] HALOPERIDOL BINDING IN BABOON BRAIN IN-VIVO
Nuclear medicine and biology
MEASURING AGE-RELATED-CHANGES IN DOPAMINE D-2 RECEPTORS WITH C-11 RACLOPRIDE AND F-18 N-METHYLSPIROPERIDOL
PSYCHIATRY RESEARCH-NEUROIMAGING
COCAINE UPTAKE IS DECREASED IN THE BRAIN OF DETOXIFIED COCAINE ABUSERS
Neuropsychopharmacology
COCAINE DOSES EQUIVALENT TO THOSE ABUSED BY HUMANS OCCUPY MOST OF THEDOPAMINE TRANSPORTERS
Synapse
MAPPING NICOTINIC ACETYLCHOLINE-RECEPTORS WITH PET
Synapse
ENDOGENOUSLY RELEASED DOPAMINE INHIBITS THE BINDING OF DOPAMINERGIC PET AND SPECT LIGANDS IN SUPERFUSED RAT STRIATAL SLICES
Synapse
I-123 LABELED DERIVATIVES OF METHYLPHENIDATE - POTENTIAL SPECT RADIOPHARMACEUTICALS FOR BRAIN DOPAMINE TRANSPORTERS
Journal of labelled compounds & radiopharmaceuticals
PREPARATION OF I-123 LABELED AM251 - A POTENTIAL SPECT RADIOLIGAND FOR THE BRAIN CANNABINOID CB1 RECEPTOR
Journal of labelled compounds & radiopharmaceuticals
PET EVALUATION OF THE DOPAMINE SYSTEM OF THE HUMAN BRAIN
The Journal of nuclear medicine
RELATIONSHIP BETWEEN DOPAMINE TRANSPORTER OCCUPANCY AND METHYLPHENIDATE INDUCED HIGH IN HUMANS
The Journal of nuclear medicine
I-123 LABELED AM-261 - A RADIOLIGAND WHICH BINDS IN-VIVO TO MOUSE-BRAIN CANNABINOID RECEPTORS
The Journal of nuclear medicine
SENSITIVITIES OF DOPAMINE D1 AND D2 RECEPTOR RADIOLIGANDS TO CHANGES IN SYNAPTIC DOPAMINE
The Journal of nuclear medicine
DOPAMINE TRANSPORTERS DECREASE WITH AGE
The Journal of nuclear medicine
RELATIONSHIP BETWEEN PSYCHOSTIMULANT-INDUCED HIGH AND DOPAMINE TRANSPORTER OCCUPANCY
Proceedings of the National Academy of Sciences of the United Statesof America
PLACE PREFERENCE AND MICRODIALYSIS STUDIES WITH 2 DERIVATIVES OF METHYLPHENIDATE
Life sciences
AFFINITIES OF METHYLPHENIDATE DERIVATIVES FOR DOPAMINE, NOREPINEPHRINE AND SEROTONIN TRANSPORTERS
Life sciences
I-123 LABELED AM251 - A RADIOIODINATED LIGAND WHICH BINDS IN-VIVO TO MOUSE-BRAIN CANNABINOID CB1 RECEPTORS
European journal of pharmacology
DISPLACEMENT OF RTI-55 FROM THE DOPAMINE TRANSPORTER BY COCAINE
European journal of pharmacology
TEMPORAL RELATIONSHIPS BETWEEN THE PHARMACOKINETICS OF METHYLPHENIDATE IN THE HUMAN BRAIN AND ITS BEHAVIORAL AND CARDIOVASCULAR EFFECTS
Psychopharmacology
IODINE-123-LABELED GLUCOSE ANALOGS - PROSPECTS FOR A SINGLE-PHOTON-EMITTING ANALOG OF FLUORINE-18-LABELED DEOXYGLUCOSE
Nuclear medicine and biology
PLASMA INPUT FUNCTION DETERMINATION FOR PET USING A COMMERCIAL LABORATORY ROBOT
Nuclear medicine and biology
SENSITIVITY OF STRIATAL [C-11] COCAINE BINDING TO DECREASES IN SYNAPTIC DOPAMINE
Synapse
LONG-LASTING INHIBITION OF IN-VIVO COCAINE BINDING TO DOPAMINE TRANSPORTERS BY 3-BETA-(4-IODOPHENYL)TROPANE-2-CARBOXYLIC ACID METHYL-ESTER - RTI-55 OR BETA-CIT
Synapse
C-11 LABELED N-METHYLSPIPERONE AND OTHER RADIOPHARMACEUTICALS FOR PETSTUDIES OF HIGH-AFFINITY BINDING-SITES
Pharmacopeial forum
CARBON-11-COCAINE BINDING COMPARED AT SUBPHARMACOLOGICAL AND PHARMACOLOGICAL DOSES - A PET STUDY
The Journal of nuclear medicine
A NEW PET LIGAND FOR THE DOPAMINE TRANSPORTER - STUDIES IN THE HUMAN BRAIN
The Journal of nuclear medicine
CARBON-11-D-THREO-METHYLPHENIDATE BINDING TO DOPAMINE TRANSPORTER IN BABOON BRAIN
The Journal of nuclear medicine
MAPPING CATECHOL-O-METHYLTRANSFERASE IN-VIVO - INITIAL STUDIES WITH [F-18] RO41-0960
Life sciences
COMPARISON OF 2 PET RADIOLIGANDS FOR IMAGING EXTRASTRIATAL DOPAMINE TRANSPORTERS IN HUMAN BRAIN
Life sciences
MECHANISTIC POSITRON EMISSION TOMOGRAPHY STUDIES OF 6-[F-18] FLUORODOPAMINE IN LIVING BABOON HEART - SELECTIVE IMAGING AND CONTROL OF RADIOTRACER METABOLISM USING THE DEUTERIUM-ISOTOPE EFFECT
Journal of neurochemistry
BINDING OF D-THREO-[C-11]METHYLPHENIDATE TO THE DOPAMINE TRANSPORTER IN-VIVO - INSENSITIVITY TO SYNAPTIC DOPAMINE
European journal of pharmacology
PHARMACOKINETICS AND IN-VIVO SPECIFICITY OF [C-11] DL-THREO-METHYLPHENIDATE FOR THE PRESYNAPTIC DOPAMINERGIC NEURON
Synapse
PET STUDIES OF COCAINE INHIBITION OF MYOCARDIAL NOREPINEPHRINE UPTAKE
Synapse
EFFECTS OF BLOOD-FLOW ON [C-11] RACLOPRIDE BINDING IN THE BRAIN - MODEL SIMULATIONS AND KINETIC-ANALYSIS OF PET DATA
Journal of cerebral blood flow and metabolism
DRUG PHARMACOKINETICS AND PHARMACODYNAMICS - PET AND MICRODIALYSIS STUDIES OF SR 46349B, SELECTIVE 5HT2 ANTAGONIST
The Journal of nuclear medicine