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Evidence of a lysosomal pathway for apoptosis induced by the synthetic retinoid CD437 in human leukemia HL-60 cells
CELL DEATH AND DIFFERENTIATION
Retinoids inhibit proliferation of human coronary smooth muscle cells by modulating cell cycle regulators
ARTERIOSCLEROSIS THROMBOSIS AND VASCULAR BIOLOGY
Phenylcyclohexene and phenylcyclohexadiene substituted compounds having retinoid antagonist activity
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Active repression of RAR signaling is required for head formation
GENES & DEVELOPMENT
1,25-dihydroxyvitamin D-3 and retonic acid analogues induce differentiation in breast cancer cells with function- and cell-specific additive effects
BREAST CANCER RESEARCH AND TREATMENT
The synthetic retinoid AGN 193109 but not retinoic acid elevates CYP1A1 levels in mouse embryos and Hepa-1c1c7 cells
TOXICOLOGY AND APPLIED PHARMACOLOGY
New dermatological agents for the treatment of psoriasis
JOURNAL OF MEDICINAL CHEMISTRY
Enantioselective syntheses of potent retinoid X receptor ligands: Differential biological activities of individual antipodes
JOURNAL OF MEDICINAL CHEMISTRY
Regulation of stearoyl coenzyme a desaturase expression in human retinal pigment epithelial cells by retinoic acid
JOURNAL OF BIOLOGICAL CHEMISTRY
Retinoic acid (RA) receptor transcriptional activation correlates with inhibition of 12-O-tetradecanoylphorbol-13-acetate-induced ornithine decarboxylase (ODC) activity by retinoids: A potential role for trans-RA-induced ZBP-89 in ODC inhibition
INTERNATIONAL JOURNAL OF CANCER
Antagonists of retinoic acid receptors (RARs) are potent growth inhibitorsof prostate carcinoma cells
BRITISH JOURNAL OF CANCER
Retinoid X receptor agonist elevation of serum triglycerides in rats by potentiation of retinoic acid receptor agonist induction or by action as single agents
BIOCHEMICAL PHARMACOLOGY
Identification of nuclear receptor interacting proteins using yeast two-hybrid technology - Applications to drug discovery
STEROID RECEPTOR METHODS: PROTOCOLS AND ASSAYS
Recent developments in receptor-selective retinoids
CURRENT PHARMACEUTICAL DESIGN
Therapeutic applications for ligands of retinoid receptors
CURRENT PHARMACEUTICAL DESIGN
Retinoic acid receptor-beta: an endogenous inhibitor of the perinatal formation of pulmonary alveoli
PHYSIOLOGICAL GENOMICS
Expression of a retinoid-inducible tumor suppressor, Tazarotene-inducible gene-3, is decreased in psoriasis and skin cancer
CLINICAL CANCER RESEARCH
Identification of receptor-selective retinoids that are potent inhibitors of the growth of human head and neck squamous cell carcinoma cells
CLINICAL CANCER RESEARCH
Role of retinoic acid in lens regeneration
DEVELOPMENTAL DYNAMICS
The carboxy-terminal hydrophobic domain of TIG3, a class II tumor suppressor protein, is required for appropriate cellular localization and optimal biological activity
INTERNATIONAL JOURNAL OF ONCOLOGY
Dual mechanisms of action of the retinoid CD437: Nuclear retinoic acid receptor-mediated suppression of squamous differentiation and receptor-independent induction of apoptosis in UMSCC22B human head and neck squamous cell carcinoma cells
MOLECULAR PHARMACOLOGY
13-cis retinoic acid exerts its specific activity on human sebocytes through selective intracellular isomerization to all-trans retinoic acid and binding to retinoid acid receptors
JOURNAL OF INVESTIGATIVE DERMATOLOGY
Regulation of skeletal progenitor differentiation by the BMP and retinoid signaling pathways
JOURNAL OF CELL BIOLOGY
Recruitment of nuclear receptor corepressor and coactivator to the retinoic acid receptor by retinoid ligands - Influence of DNA-heterodimer interactions
JOURNAL OF BIOLOGICAL CHEMISTRY
Peroxisome proliferator-activated receptor and retinoid X receptor ligandsinhibit monocyte chemotactic protein-1-directed migration of monocytes
EUROPEAN JOURNAL OF PHARMACOLOGY
Novel approaches for the treatment of psoriasis
DRUG DISCOVERY TODAY
Differential responses of normal, premalignant, and malignant human bronchial epithelial cells to receptor-selective retinoids
CLINICAL CANCER RESEARCH
Mannose 6-phosphate/insulin-like growth factor II receptor mediates the growth-inhibitory effects of retinoids
CELL GROWTH & DIFFERENTIATION
Cell type and gene-specific activity of the retinoid inverse agonist AGN 193109: Divergent effects from agonist at retinoic acid receptor gamma in human keratinocytes
CELL GROWTH & DIFFERENTIATION
Synthesis and biological activity of high-affinity retinoic acid receptor antagonists
BIOORGANIC & MEDICINAL CHEMISTRY
A new class of RAR subtype selective retinoids: Correlation of pharmacological effects with receptor activity
BIOORGANIC & MEDICINAL CHEMISTRY
A new class of potent RAR antagonists: Dihydroanthracenyl, benzochromenyl and benzothiochromenyl retinoids
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
High affinity retinoic acid receptor antagonists: Analogs of AGN 193109
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Stereoselective synthesis and receptor activity of conformationally defined retinoid X receptor selective ligands
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
A short and efficient synthesis of 4-[2,2-dimethyl-4(tol-4-yl)benzochrom-3-en-7-yl]benzoic acid - A potent retinoic acid receptor antagonist
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
Retinoid X receptor (RXR) agonist-induced activation of dominant-negative RXR-retinoic acid receptor alpha 403 heterodimers is developmentally regulated during myeloid differentiation
MOLECULAR AND CELLULAR BIOLOGY
Multiple left-right asymmetry defects in Shh(-/-) mutant mice unveil a convergence of the Shh and retinoic acid pathways in the control of Lefty-1
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
Retinoid-dependent recruitment of a histone H1 displacement activity by retinoic acid receptor
JOURNAL OF BIOLOGICAL CHEMISTRY
Retinoid signaling is required for chondrocyte maturation and endochondralbone formation during limb skeletogenesis
DEVELOPMENTAL BIOLOGY
Tazarotene gel is safe and effective in the treatment of acne vulgaris: A multicenter, double-blind, vehicle-controlled study
CUTIS
Retinoic acid increases tyrosine phosphorylation of focal adhesion kinase and paxillin in MCF-7 human breast cancer cells
CANCER RESEARCH
Novel retinoids with receptor selectivity and functional selectivity
BRITISH JOURNAL OF DERMATOLOGY
Vitamin D regulates human ectocervical epithelial cell proliferation and insulin-like growth factor-binding protein-3 level
BIOLOGY OF REPRODUCTION
THE USE OF A RETINOID RECEPTOR ANTAGONIST IN A NEW MODEL TO STUDY VITAMIN-A-DEPENDENT DEVELOPMENTAL EVENTS
The International journal of developmental biology
RATIONAL DESIGN OF RECEPTOR-SELECTIVE RETINOIDS
Journal of the American Academy of Dermatology
FUTURE-TRENDS - A NEW-GENERATION OF RETINOIDS
Journal of the American Academy of Dermatology
ONCE-DAILY TAZAROTENE GEL VERSUS TWICE-DAILY FLUOCINONIDE CREAM IN THE TREATMENT OF PLAQUE PSORIASIS
Journal of the American Academy of Dermatology
RETINOIC ACID ALTERS THE INTRACELLULAR TRAFFICKING OF THE MANNOSE-6-PHOSPHATE INSULIN-LIKE-GROWTH-FACTOR-II RECEPTOR AND LYSOSOMAL-ENZYMES
Proceedings of the National Academy of Sciences of the United Statesof America
Identification and characterization of a retinoid-induced class II tumor suppressor growth regulatory gene
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
LIGAND INDUCTION OF RETINOIC ACID RECEPTORS ALTERS AN ACUTE INFECTIONBY MURINE CYTOMEGALOVIRUS
Journal of virology
THE SAFETY AND EFFICACY OF TAZAROTENE GEL, A TOPICAL ACETYLENIC RETINOID, IN THE TREATMENT OF PSORIASIS
Archives of dermatology
SYNTHESIS AND BIOLOGICAL-ACTIVITY OF 1,2,3,4-TETRAHYDROQUINOLINE AND 3,4-(1H)-DIHYDROQUINOLIN-2-ONE ANALOGS OF RETINOIC ACID
Bioorganic & medicinal chemistry letters
LACK OF INVOLVEMENT OF RETINOIC ACID RECEPTOR-ALPHA IN RETINOID-INDUCED SKIN IRRITATION IN HAIRLESS MICE
Toxicology letters
RETINOID ANTAGONISM OF NF-IL6 - INSIGHT INTO THE MECHANISM OF ANTIPROLIFERATIVE EFFECTS OF RETINOIDS IN KAPOSIS-SARCOMA
Molecular and cellular biology
TAZAROTENE - THE FIRST RECEPTOR-SELECTIVE TOPICAL RETINOID FOR THE TREATMENT OF PSORIASIS
Journal of the American Academy of Dermatology
MOLECULAR MECHANISMS OF TAZAROTENE ACTION IN PSORIASIS
Journal of the American Academy of Dermatology
TAZAROTENE GEL, A NEW RETINOID, FOR TOPICAL THERAPY OF PSORIASIS - VEHICLE-CONTROLLED STUDY OF SAFETY, EFFICACY, AND DURATION OF THERAPEUTIC EFFECT
Journal of the American Academy of Dermatology
RECEPTOR SPECIFICITY OF RETINOID-INDUCED EPIDERMAL HYPERPLASIA - EFFECT OF RXR-SELECTIVE AGONISTS AND CORRELATION WITH TOPICAL IRRITATION
The Journal of pharmacology and experimental therapeutics
IDENTIFICATION OF HIGHLY POTENT RETINOIC ACID RECEPTOR ALPHA-SELECTIVE ANTAGONISTS
Journal of medicinal chemistry
TAZAROTENE-INDUCED-GENE-2 (TIG2), A NOVEL RETINOID-RESPONSIVE GENE INSKIN
Journal of investigative dermatology
INTERFERON-INDUCIBLE PROTEIN-10 IS REDUCED BY TREATMENT WITH RAR SPECIFIC RETINOIDS IN PSORIASIS AND KERATINOCYTE CULTURES
Journal of investigative dermatology
TAZAROTENE AN RAR SELECTIVE RETINOID, AFFECTS THE EXPRESSION OF GENESASSOCIATED WITH ABNORMAL DIFFERENTIATION, HYPERPROLIFERATION AND INFLAMMATION
Journal of investigative dermatology
RETINOID INHIBITION OF MRP-8 VIA ANTAGONISM OF NF-IL6 ENHANCER ACTIVITY - A NOVEL MECHANISM OF GENE-REGULATION
Journal of investigative dermatology
IDENTIFICATION OF RETINOIC ACID RECEPTOR INVERSE AGONISTS AND THEIR POTENTIAL USE AS THERAPEUTIC AGENTS
Journal of investigative dermatology
VITAMIN-D SUPPRESSES HUMAN ECTOCERVICAL KERATINOCYTE PROLIFERATION AND INCREASES INSULIN-LIKE GROWTH-FACTOR BINDING PROTEIN-3 (IGFBP-3)
Journal of investigative dermatology
ANTAGONISM OF TRANSCRIPTION FACTOR ACTION - A MAJOR-MODE OF THERAPEUTIC ACTION OF RETINOIDS
Journal of investigative dermatology
INTERFERON REGULATION OF PROLIFERATION AND INSULIN-LIKE GROWTH-FACTORBINDING-PROTEIN EXPRESSION IN HUMAN ECTOCERVICAL KERATINOCYTES
Journal of investigative dermatology
TAZAROTENE 0.1-PERCENT GEL IS ASSOCIATED WITH ALTERATIONS IN MARKERS OF EPIDERMAL DIFFERENTIATION AND INFLAMMATION IN PSORIATIC PLAQUES
Journal of investigative dermatology
RETINOID AGONISTS AND INVERSE AGONISTS - A NEW-GENERATION
Journal of investigative dermatology
RETINOIC ACID RECEPTOR-NUCLEAR FACTOR-INTERLEUKIN-6 ANTAGONISM - A NOVEL MECHANISM OF RETINOID-DEPENDENT INHIBITION OF A KERATINOCYTE HYPERPROLIFERATIVE DIFFERENTIATION MARKER
The Journal of biological chemistry
DIFFERENTIAL-EFFECTS OF SYNTHETIC NUCLEAR RETINOID RECEPTOR-SELECTIVERETINOIDS ON THE GROWTH OF HUMAN NONSMALL CELL LUNG-CARCINOMA CELLS
Cancer research
RETINOIC ACID RECEPTOR-ALPHA EXPRESSION CORRELATES WITH RETINOID-INDUCED GROWTH-INHIBITION OF HUMAN BREAST-CANCER CELLS REGARDLESS OF ESTROGEN-RECEPTOR STATUS
Cancer research
MITOGENIC EFFECT OF RETINOID-X-RECEPTOR AGONISTS IN RAT-LIVER
Biochemical pharmacology
DIFFERENTIAL REGULATION OF HUMAN ECTOCERVICAL EPITHELIAL-CELL LINE PROLIFERATION AND DIFFERENTIATION BY RETINOID-X-RECEPTOR-SPECIFIC AND RETINOIC ACID RECEPTOR-SPECIFIC RETINOIDS
Cell growth & differentiation
NEGATIVE REGULATION OF 2 HYPERPROLIFERATIVE KERATINOCYTE DIFFERENTIATION MARKERS BY A RETINOIC ACID RECEPTOR-SPECIFIC RETINOID - INSIGHT INTO THE MECHANISM OF RETINOID ACTION IN PSORIASIS
Cell growth & differentiation
SYNTHESIS OF HIGHLY POTENT RXR-SPECIFIC RETINOIDS - THE USE OF A CYCLOPROPYL GROUP AS A DOUBLE-BOND ISOSTERE
Bioorganic & medicinal chemistry letters
RETINOID-INDUCED EPIPHYSEAL PLATE CLOSURE IN GUINEA-PIGS
Fundamental and applied toxicology
RETINOID-INDUCED HYPERTRIGLYCERIDEMIA IN RATS IS MEDIATED BY RETINOICACID RECEPTORS
Fundamental and applied toxicology
RETINOID-REGULATED EXPRESSION OF BCL-2 AND TISSUE TRANSGLUTAMINASE DURING THE DIFFERENTIATION AND APOPTOSIS OF HUMAN MYELOID-LEUKEMIA (HL-60) CELLS
Leukemia research
SPECIFIC ANTAGONIST OF RETINOID TOXICITY IN MICE
Toxicology and applied pharmacology
SELECTIVE CONVERSION OF ALPHA-TETRALONES TO DIHYDRONAPHTHALENES
Tetrahedron letters
IDENTIFICATION OF RETINOIC ACID RECEPTOR-BETA SUBTYPE-SPECIFIC AGONISTS
Journal of medicinal chemistry
SYNTHESIS AND STRUCTURE-ACTIVITY-RELATIONSHIPS OF RETINOID-X RECEPTOR-SELECTIVE DIARYL SULFIDE ANALOGS OF RETINOIC ACID
Journal of medicinal chemistry
IDENTIFICATION OF A RETINOIC ACID RECEPTOR-ALPHA SUBTYPE-SPECIFIC AGONIST
Journal of medicinal chemistry
TIG1 AND TIG2 (TAZAROTENE INDUCED GENE-1 AND GENE-2) ARE NOVEL RETINOIC ACID RECEPTOR-RESPONSIVE GENES IN SKIN
Journal of investigative dermatology
AGN193109 IS A PURE ANTAGONIST OF RETINOID ACTION IN HUMAN ECTOCERVICAL KERATINOCYTES
Journal of investigative dermatology
RXR-SPECIFIC RETINOIDS INHIBIT THE ABILITY OF RAR-SPECIFIC RETINOIDS TO INCREASE THE LEVEL OF INSULIN-LIKE GROWTH-FACTOR BINDING PROTEIN-9 (IGFBP-3) IN HUMAN ECTOCERVICAL EPITHELIAL-CELLS
Journal of investigative dermatology
COORDINATE REGULATION OF KERATINOCYTE DIFFERENTIATION MARKERS BY RETINOIDS IN CELL-CULTURE AND IN PSORIASIS
Journal of investigative dermatology
THE USE OF A RETINOIC ACID RECEPTOR ANTAGONIST TO PREVENT RETINOID-INDUCED SKIN IRRITATION
Journal of investigative dermatology
TAZAROTENE-INDUCED GENE-1 (TIG1), A NOVEL RETINOIC ACID RECEPTOR-RESPONSIVE GENE IN SKIN
Journal of investigative dermatology
IDENTIFICATION AND CHARACTERIZATION OF A VERSATILE RETINOID RESPONSE ELEMENT (RETINOIC ACID RECEPTOR RESPONSE ELEMENT-RETINOID-X-RECEPTOR RESPONSE ELEMENT) IN THE MOUSE-TISSUE TRANSGLUTAMINASE GENE PROMOTER
The Journal of biological chemistry
AGN193109 IS A HIGHLY EFFECTIVE ANTAGONIST OF RETINOID ACTION IN HUMAN ECTOCERVICAL EPITHELIAL-CELLS
The Journal of biological chemistry
DIFFERENTIAL TERATOGENIC RESPONSE OF MOUSE EMBRYOS TO RECEPTOR-SELECTIVE ANALOGS OF RETINOIC ACID
Chemico-biological interactions
RETINOID-X RECEPTOR-SPECIFIC RETINOIDS INHIBIT THE ABILITY OF RETINOIC ACID RECEPTOR-SPECIFIC RETINOIDS TO INCREASE THE LEVEL OF INSULIN-LIKE GROWTH-FACTOR BINDING PROTEIN-3 IN HUMAN ECTOCERVICAL EPITHELIAL-CELLS
Cancer research
TAZAROTENE - FIRST OF A NEW-GENERATION OF RECEPTOR-SELECTIVE RETINOIDS
British journal of dermatology
INDISPENSABLE ROLE OF VITAMIN-A SIGNALING IN NORMAL VERTEBRATE DEVELOPMENT
Molecular biology of the cell
SYNTHESIS AND PHARMACOLOGICAL ACTIVITY OF CONFORMATIONALLY RESTRICTED, ACETYLENIC RETINOID ANALOGS
Bioorganic & medicinal chemistry letters
DIFFERENTIAL RXR AND RAR ACTIVITY OF STILBENE RETINOID ANALOGS BEARING THIAZOLE AND IMIDAZOLE CARBOXYLIC-ACIDS
Bioorganic & medicinal chemistry letters
ACTIVATION OF RETINOID-X RECEPTORS INDUCES APOPTOSIS IN HL-60 CELL-LINES
Molecular and cellular biology
DEVELOPMENT OF RAR SUBTYPE-SELECTIVE RETINOIDS FOR DERMATOLOGICAL DISEASES
European journal of medicinal chemistry