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1. Cooper, LC; Chicchi, GG; Dinnell, K; Elliott, JM; Hollingworth, GJ; Kurtz, MM; Locker, KL; Morrison, D; Shaw, DE; Tsao, KL; Watt, AP; Williams, AR; Swain, CJ
   2-aryl indole NK1 receptor antagonists: Optimisation of indole substitution
   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
   
   L.C. Cooper et al., "2-aryl indole NK1 receptor antagonists: Optimisation of indole substitution", BIOORG MED, 11(9), 2001, pp. 1233-1236
2. Dinnell, K; Chicchi, GG; Dhar, MJ; Elliott, JM; Hollingworth, GJ; Kurtz, MM; Ridgill, MP; Rycroft, W; Tsao, KL; Williams, AR; Swain, CJ
   2-aryl indole NK1 receptor antagonists: Optimisation of the 2-aryl ring and the indole nitrogen substituent
   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
   
   K. Dinnell et al., "2-aryl indole NK1 receptor antagonists: Optimisation of the 2-aryl ring and the indole nitrogen substituent", BIOORG MED, 11(9), 2001, pp. 1237-1240
3. Shaw, D; Chicchi, GG; Elliott, JM; Kurtz, M; Morrison, D; Ridgill, MP; Szeto, N; Watt, AP; Williams, AR; Swain, CJ
   2-aryl indole NK1 antagonists: Optimisation of the amide substituent
   BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
   
   D. Shaw et al., "2-aryl indole NK1 antagonists: Optimisation of the amide substituent", BIOORG MED, 11(23), 2001, pp. 3031-3034
4. Harrison, T; Owens, AP; Williams, BJ; Swain, CJ; Williams, A; Carlson, EJ; Rycroft, W; Tattersall, FD; Cascieri, MA; Chicchi, GG; Sadowski, S; Rupniak, NMJ; Hargreaves, RJ
   An orally active, water-soluble neurokinin-1 receptor antagonist suitable for both intravenous and oral clinical administration
   JOURNAL OF MEDICINAL CHEMISTRY
   
   T. Harrison et al., "An orally active, water-soluble neurokinin-1 receptor antagonist suitable for both intravenous and oral clinical administration", J MED CHEM, 44(24), 2001, pp. 4296-4299
5. Hale, JJ; Mills, SG; MacCoss, M; Dorn, CP; Finke, PE; Budhu, RJ; Reamer, RA; Huskey, SEW; Luffer-Atlas, D; Dean, BJ; McGowan, EM; Feeney, WP; Chiu, SHL; Cascieri, MA; Chicchi, GG; Kurtz, MM; Sadowski, S; Ber, E; Tattersall, FD; Rupniak, NMJ; Williams, AR; Rycroft, W; Hargreaves, R; Metzger, JM; MacIntyre, DE
   Phosphorylated morpholine acetal human neurokinin-1 receptor antagonists as water-soluble prodrugs
   JOURNAL OF MEDICINAL CHEMISTRY
   
   J.J. Hale et al., "Phosphorylated morpholine acetal human neurokinin-1 receptor antagonists as water-soluble prodrugs", J MED CHEM, 43(6), 2000, pp. 1234-1241
6. Cascieri, MA; Koch, GE; Ber, E; Sadowski, SJ; Louizides, D; de Laszlo, SE; Hacker, C; Hagmann, WK; MacCoss, M; Chicchi, GG; Vicario, PP
   Characterization of a novel, non-peptidyl antagonist of the human glucagonreceptor
   JOURNAL OF BIOLOGICAL CHEMISTRY
   
   M.A. Cascieri et al., "Characterization of a novel, non-peptidyl antagonist of the human glucagonreceptor", J BIOL CHEM, 274(13), 1999, pp. 8694-8697
7. KRAMER MS; CUTLER N; FEIGHNER J; SHRIVASTAVA R; CARMAN J; SRAMEK JJ; REINES SA; LIU GH; SNAVELY D; WYATTKNOWLES E; HALE JJ; MILLS SG; MACCOSS M; SWAIN CJ; HARRISON T; HILL RG; HEFTI F; SCOLNICK EM; CASCIERI MA; CHICCHI GG; SADOWSKI S; WILLIAMS AR; HEWSON L; SMITH D; CARLSON EJ; HARGREAVES RJ; RUPNIAK NMJ
   DISTINCT MECHANISM FOR ANTIDEPRESSANT ACTIVITY BY BLOCKADE OF CENTRALSUBSTANCE-P RECEPTORS
   Science
   
   M.S. Kramer et al., "DISTINCT MECHANISM FOR ANTIDEPRESSANT ACTIVITY BY BLOCKADE OF CENTRALSUBSTANCE-P RECEPTORS", Science, 281(5383), 1998, pp. 1640-1645
8. HALE JJ; MILLS SG; MACCOSS M; FINKE PE; CASCIERI MA; SADOWSKI S; BER E; CHICCHI GG; KURTZ M; METZGER J; EIERMANN G; TSOU NN; TATTERSALL FD; RUPNIAK NMJ; WILLIAMS AR; RYCROFT W; HARGREAVES R; MACINTYRE DE
   STRUCTURAL OPTIMIZATION AFFORDING ENYL-4-(3-OXO-1,2,4-TRIAZOL-5-YL)METHYLMORPHOLINE, A POTENT, ORALLY-ACTIVE, LONG-ACTING MORPHOLINE ACETALHUMAN NK-1 RECEPTOR ANTAGONIST
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   J.J. Hale et al., "STRUCTURAL OPTIMIZATION AFFORDING ENYL-4-(3-OXO-1,2,4-TRIAZOL-5-YL)METHYLMORPHOLINE, A POTENT, ORALLY-ACTIVE, LONG-ACTING MORPHOLINE ACETALHUMAN NK-1 RECEPTOR ANTAGONIST", Journal of medicinal chemistry, 41(23), 1998, pp. 4607-4614
9. STEVENSON GI; HUSCROFT I; MACLEOD AM; SWAIN CJ; CASCIERI MA; CHICCHI GG; GRAHAM MI; HARRISON T; KELLEHER FJ; KURTZ M; LADDUWAHETTY T; MERCHANT KJ; METZGER JM; MACINTYRE DE; SADOWSKI S; SOHAL B; OWENS AP
   4,4-DISUBSTITUTED PIPERIDINE HIGH-AFFINITY NK1 ANTAGONISTS - STRUCTURE-ACTIVITY-RELATIONSHIPS AND IN-VIVO ACTIVITY
   Journal of medicinal chemistry
   
   G.I. Stevenson et al., "4,4-DISUBSTITUTED PIPERIDINE HIGH-AFFINITY NK1 ANTAGONISTS - STRUCTURE-ACTIVITY-RELATIONSHIPS AND IN-VIVO ACTIVITY", Journal of medicinal chemistry, 41(23), 1998, pp. 4623-4635
10. CHICCHI GG; CASCIERI MA; GRAZIANO MP; CALAHAN T; TOTA MR
    FLUORESCEIN-TRP(25)-EXENDIN-4, A BIOLOGICALLY-ACTIVE FLUORESCENT-PROBE FOR THE HUMAN GLP-1 RECEPTOR
    Peptides
    
    G.G. Chicchi et al., "FLUORESCEIN-TRP(25)-EXENDIN-4, A BIOLOGICALLY-ACTIVE FLUORESCENT-PROBE FOR THE HUMAN GLP-1 RECEPTOR", Peptides, 18(2), 1997, pp. 319-321
11. CHICCHI GG; GRAZIANO MP; KOCH G; HEY P; SULLIVAN K; VICARIO PP; CASCIERI MA
    ALTERATIONS IN RECEPTOR ACTIVATION AND DIVALENT-CATION ACTIVATION OF AGONIST BINDING BY DELETION OF INTRACELLULAR DOMAINS OF THE GLUCAGON RECEPTOR
    The Journal of biological chemistry
    
    G.G. Chicchi et al., "ALTERATIONS IN RECEPTOR ACTIVATION AND DIVALENT-CATION ACTIVATION OF AGONIST BINDING BY DELETION OF INTRACELLULAR DOMAINS OF THE GLUCAGON RECEPTOR", The Journal of biological chemistry, 272(12), 1997, pp. 7765-7769
12. CHICCHI GG; CASCIERI MA; GRAZIANO MP; TOTA MR
    FLUORESCEIN-TRP(25)-EXENDIN-4, A NOVEL PROBE FOR THE HUMAN GLUCAGON-LIKE PEPTIDE-1 RECEPTOR
    Diabetes
    
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13. GRAZIANO MP; HEY PJ; BORKOWSKI D; CHICCHI GG; STRADER CD
    CLONING AND FUNCTIONAL EXPRESSION OF A HUMAN GLUCAGON-LIKE PEPTIDE-1 RECEPTOR
    Journal of cellular biochemistry
    
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14. GRAZIANO MP; HEY PJ; BORKOWSKI D; CHICCHI GG; STRADER CD
    CLONING AND FUNCTIONAL EXPRESSION OF A HUMAN GLUCAGON-LIKE PEPTIDE-1-RECEPTOR
    Biochemical and biophysical research communications
    
    M.P. Graziano et al., "CLONING AND FUNCTIONAL EXPRESSION OF A HUMAN GLUCAGON-LIKE PEPTIDE-1-RECEPTOR", Biochemical and biophysical research communications, 196(1), 1993, pp. 141-146