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Parallel synthesis and pharmacological screening oi nonpeptide ligands of the neuropeptide Y receptor subtype Y-5
JOURNAL OF PEPTIDE RESEARCH
From peptide libraries to optimized nonpeptide ligands in the search for S-farnesyltransferase inhibitors
JOURNAL OF PEPTIDE RESEARCH
Regulation of murine airway responsiveness by endothelial nitric oxide synthase
AMERICAN JOURNAL OF PHYSIOLOGY-LUNG CELLULAR AND MOLECULAR PHYSIOLOGY
Reduced food intake in response to CCP 71683A may be due to mechanisms other than NPYY5 receptor blockade
INTERNATIONAL JOURNAL OF OBESITY
Genomic organization and characterization of splice variants of the human histamine H-3 receptor
BIOCHEMICAL JOURNAL
Role of a pineal cAMP-operated arylalkylamine N-acetyltransferase/14-3-3-binding switch in melatonin synthesis (vol 98, pg 8083, 2001)
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
Role of a pineal cAMP-operated arylalkylamine N-acetyltransferase/14-3-3-binding switch in melatonin synthesis
PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA
Cloning and molecular characterization of the novel human melanin-concentrating hormone receptor MCH2
MOLECULAR PHARMACOLOGY
SLC-1 receptor mediates effect of melanin-concentrating hormone on feedingbehavior in rat: A structure-activity study
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Antiparkinsonian agent piribedil displays antagonist properties at native,rat, and cloned, human alpha(2)-adrenoceptors: Cellular and functional characterization
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Structure-activity relationship studies of melanin-concentrating hormone (MCH)-related peptide ligands at SLC-1, the human MCH receptor
JOURNAL OF BIOLOGICAL CHEMISTRY
Binding of prostaglandins to human PPAR gamma: tool assessment and new natural ligands
EUROPEAN JOURNAL OF PHARMACOLOGY
Development of new assays and improved procedures for the purification of recombinant human chymase
EUROPEAN JOURNAL OF BIOCHEMISTRY
[I-125]-S36057: a new and highly potent radioligand for the melanin-concentrating hormone receptor
BRITISH JOURNAL OF PHARMACOLOGY
Comparative pharmacological studies of melatonin receptors: MT1, MT2 and MT3/QR2. Tissue distribution of MT3/QR2
BIOCHEMICAL PHARMACOLOGY
Structure and expression of the human histamine H-4-receptor gene
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS
High-capacity screening of arylalkylamine N-acetyltransferase inhibitors using a high-performance liquid chromatography system
JOURNAL OF BIOMOLECULAR SCREENING
Screening of ligand binding on melatonin receptor using non-peptide combinatorial libraries
JOURNAL OF RECEPTOR AND SIGNAL TRANSDUCTION RESEARCH
Synthesis of a small library of phenylalkylamide derivatives as melatoninergic ligands for human mt(1) and MT2 receptors
BIOORGANIC & MEDICINAL CHEMISTRY
Agonist and antagonist actions of yohimbine as compared to fluparoxan at alpha(2)-adrenergic receptors (AR)s, serotonin (5-HT)(1A), 5-HT1B, 5-HT1D and dopamine D-2 and D-3 receptors. Significance for the modulation of frontocortical monoaminergic transmission and depressive states
SYNAPSE
Antagonist properties of the novel antipsychotic, S16924, at cloned, humanserotonin 5-HT2C receptors: a parallel phosphatidylinositol and calcium accumulation comparison with clozapine and haloperidol
NAUNYN-SCHMIEDEBERGS ARCHIVES OF PHARMACOLOGY
S18616, a highly potent, spiroimidazoline agonist at alpha(2)-adrenoceptors: I. Receptor profile, antinociceptive and hypothermic actions in comparison with dexmedetomidine and clonidine
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
S18327 (1-{2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)piperid-1-yl]ethyl}3-phenyl imidazolin-2-one), a novel, potential antipsychotic displaying marked antagonist properties at alpha(1) and alpha(2)-adrenergic receptors: I. Receptorial, neurochemical, and electrophysiological profile
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
Synthesis of phenalene and acenaphthene derivatives as new conformationally restricted ligands for melatonin receptors
JOURNAL OF MEDICINAL CHEMISTRY
Substrate specificity and inhibition studies of human serotonin N-acetyltransferase (vol 275, pg 8794, 2000)
JOURNAL OF BIOLOGICAL CHEMISTRY
Identification of the melatonin-binding site MT3 as the quinone reductase 2
JOURNAL OF BIOLOGICAL CHEMISTRY
Substrate specificity and inhibition studies of human serotonin N-acetyltransferase
JOURNAL OF BIOLOGICAL CHEMISTRY
Food intake regulation in rodents: Y-5 or Y1NPY receptors or both?
CANADIAN JOURNAL OF PHYSIOLOGY AND PHARMACOLOGY
Physico-chemical and biological analysis of true combinatorial libraries
JOURNAL OF CHROMATOGRAPHY B
INVESTIGATION OF S-FARNESYL TRANSFERASE SUBSTRATE-SPECIFICITY WITH COMBINATORIAL TETRAPEPTIDE LIBRARIES
Cellular signalling
Truncated isoforms inhibit [H-3]prazosin binding and cellular trafficking of native human alpha(1A)-adrenoceptors
BIOCHEMICAL JOURNAL
Characterization of 2-[I-125]iodomelatonin binding sites in syrian hamsterperipheral organs
JOURNAL OF PHARMACOLOGY AND EXPERIMENTAL THERAPEUTICS
NPY receptor subtype in the rabbit isolated ileum
BRITISH JOURNAL OF PHARMACOLOGY
Cloning and characterization of the 5 ' flanking region of the human uncoupling protein 3 (UCP3) gene
BIOCHEMICAL AND BIOPHYSICAL RESEARCH COMMUNICATIONS
Combinatorial chemistry for the generation of molecular diversity and the discovery of bioactive leads
CHEMOMETRICS AND INTELLIGENT LABORATORY SYSTEMS
NPY RECEPTOR SUBTYPES INVOLVED IN THE CONTRACTION OF THE PROXIMAL COLON OF THE RAT
Regulatory peptides
A ZINC CHELATOR INHIBITING GELATINASES EXERTS POTENT IN-VITRO ANTI-INVASIVE EFFECTS
European journal of pharmacology
CHROMATOGRAPHIC ASSAY AND PEPTIDE SUBSTRATE CHARACTERIZATION OF PARTIALLY PURIFIED FARNESYLGERANYLTRANSFERASES AND GERANYLGERANYLTRANSFERASES FROM RAT-BRAIN CYTOSOL
Archives of biochemistry and biophysics
LIMITATIONS OF THE COUPLING OF AMINO-ACID MIXTURES FOR THE PREPARATION OF EQUIMOLAR PEPTIDE LIBRARIES
Molecular diversity
SELECTION OF A HISTIDINE-CONTAINING INHIBITOR OF GELATINASES THROUGH DECONVOLUTION OF COMBINATORIAL TETRAPEPTIDE LIBRARIES
Molecular diversity
EVALUATION OF HIGH-PERFORMANCE LIQUID-CHROMATOGRAPHY ELECTROSPRAY MASS-SPECTROMETRY WITH SELECTED-ION MONITORING FOR THE ANALYSIS OF LARGE SYNTHETIC COMBINATORIAL PEPTIDE LIBRARIES
Rapid communications in mass spectrometry
MYRISTOYLATION
Cellular signalling
SEEKING FOR NEW RAT-BRAIN FARNESYL SUBSTRAINTS BY USE OF SYNTHETIC COMBINATORIAL TETRAPEPTIDE LIBRANES
The FASEB journal
COMBINATORIAL CHEMISTRY - STATE-OF-THE-AR T, ANALYTICAL NEEDS AND FUTURE EVOLUTIONS
Analusis
PEPTIDE AND NONPEPTIDE LEAD DISCOVERY USING ROBOTICALLY SYNTHESIZED SOLUBLE LIBRARIES
Canadian journal of physiology and pharmacology
TYROSINE PROTEIN-KINASE ASSAYS
Journal of chromatography B. Biomedical applications
COMBINATORIAL PEPTIDE LIBRARIES - ROBOTIC SYNTHESIS AND ANALYSIS BY NUCLEAR-MAGNETIC-RESONANCE, MASS-SPECTROMETRY, TANDEM MASS-SPECTROMETRY, AND HIGH-PERFORMANCE CAPILLARY ELECTROPHORESIS TECHNIQUES
Analytical biochemistry
COMBINATORIAL PEPTIDE-SYNTHESIS - STATISTICAL EVALUATION OF PEPTIDE DISTRIBUTION
Trends in pharmacological sciences
SUBSTRATE PHOSPHORYLATION CAPACITIES OF THE MAJOR TYROSINE PROTEIN-KINASE FROM THE HUMAN PROMYELOCYTIC CELL-LINE, HL-60
International journal of peptide & protein research
HETEROGENEITY OF HEPATIC-MICROSOMAL UDP-GLUCURONOSYLTRANSFERASE(S) ACTIVITIES - A NEW KINETIC APPROACH FOR THE STUDY OF INDUCTION AND SPECIFICITY
Journal of pharmaceutical sciences
TYROSINE PROTEIN-KINASE INHIBITION AND CANCER
International Journal of Biochemistry
HETEROGENEITY OF HEPATIC UDP-GLUCURONOSYLTRANSFERASE ACTIVITIES - INVESTIGATIONS OF ISOENZYMES INVOLVED IN P-NITROPHENOL GLUCURONIDATION
Comparative biochemistry and physiology. C. Comparative pharmacologyand toxicology
IN-VIVO AND IN-VITRO GLUCURONIDATION OF THE FLAVONOID DIOSMETIN IN RATS
Drug metabolism and disposition
MYRISTOYL-COA-PROTEIN N-MYRISTOYLTRANSFERASE ACTIVITY IN CANCER-CELLS- PURIFICATION AND CHARACTERIZATION OF A CYTOSOLIC ISOFORM FROM THE MURINE LEUKEMIA-CELL LINE L1210
European journal of biochemistry
PURIFICATION AND CHARACTERIZATION OF THE MAJOR TYROSINE PROTEIN-KINASE FROM THE HUMAN PROMYELOCYTIC CELL-LINE, HL-60
European journal of biochemistry
INTEGRATED SYSTEM FOR THE SCREENING OF THE SPECIFICITY OF PROTEIN-KINASE INHIBITORS
Biochemical pharmacology